Pharmacological characterization of GLPG1972/S201086, a potent and selective small-molecule inhibitor of ADAMTS5 by Clement-Lacroix, P., Little, C.B., Smith, M.M., Cottereaux, C., Merciris, D., Meurisse, S., Mollat, P., Touitou, R., Brebion, F., Gosmini, R., De Ceuninck, F., Botez, I., Lepescheux, L., van der Aar, E., Christophe, T., Vandervoort, N., Blanqué, R., Comas, D., Deprez, P., Amantini, D.

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GLPG1972: a potent, selective, orally available adamts-5 inhibitor for the treatment of OA by Clement-Lacroix, P, Little, C, Meurisse, S, Blanqué, R, Mollat, P, Brebion, F, Gosmini, R, De Ceuninck, F, Botez, I, Lepescheux, L, van der Aar, E, Christophe, T, Vandervoort, N, Cottereaux, C, Comas, D, Deprez, P, Amantini, D

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New cartilage quality evaluation using bio-indentation: effect of a tool dmoad compound active in the rat MNX model by Lavet, C, Clement-Lacroix, P, Merciris, D, Meurisse, S, Lepescheux, L, Gaillard, V, Pastoureau, P, Deprez, P, Amantini, D, Ammann, P

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Efficient O-Trimethylsilylation of Alcohols and Phenols with Trimethylsilyl Azide Catalyzed by Tetrabutylammonium Bromide under Neat Conditions by Amantini, David, Fringuelli, Francesco, Pizzo, Ferdinando, Vaccaro, Luigi

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Bromolysis and Iodolysis of α,β-Epoxycarboxylic Acids in Water Catalyzed by Indium Halides by Amantini, David, Fringuelli, Francesco, Pizzo, Ferdinando, Vaccaro, Luigi

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Synthesis of 4-Aryl-1H-1,2,3-triazoles through TBAF-Catalyzed [3 + 2] Cycloaddition of 2-Aryl-1-nitroethenes with TMSN3 under Solvent-Free Conditions by Amantini, David, Fringuelli, Francesco, Piermatti, Oriana, Pizzo, Ferdinando, Zunino, Ennio, Vaccaro, Luigi

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ADAMTS-5 inhibitor GLPG1972, a potential new treatment in osteoarthritis, shows favorable safety, pharmacokinetics and pharmacodynamics in healthy subjects by van der Aar, E.M., Desrivot, J., Fagard, L., Amantini, D., Larsson, S., Struglics, A., Lohmander, S., Vanhoutte, F., Dupont, S.

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SELECTED METHODS FOR THE REDUCTION OF THE AZIDO GROUP by Amantini, D., Fringuelli, F., Pizza, F., Vaccaro, L.

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ADAMTS-5 inhibition with the potent and highly selective inhibitor GLPG1972 results in strong disease-modifying OA drug effects in the rat meniscectomy model by Clement-Lacroix, P., Meurisse, S., Lepescheux, L., Merciris, D., Borgonovi, M., Cottereaux, C., Mollat, P., Brebion, F., Gosmini, R., De Ceuninck, F., Botez, I., Christophe, T., van der Aar, E.E., Vandervoort, N., Blanqué, R., Comas, D., Deprez, P., Amantini, D.

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3-Nitrocoumarins as Dienophiles in the Diels−Alder Reaction in Water. An Approach to the Synthesis of Nitrotetrahydrobenzo[c]chromenones and Dihydrodibenzo[b,d]furans by Amantini, David, Fringuelli, Francesco, Piermatti, Oriana, Pizzo, Ferdinando, Vaccaro, Luigi

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Uncatalyzed [4 + 2] Cycloadditions of 3-Nitrocoumarins with Vinyl Ethers in Solventless Conditions. A New Entry to Chromene Derivatives by Amantini, David, Fringuelli, Francesco, Pizzo, Ferdinando

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ZnCl2 as an Efficient Catalyst in the Thiolysis of 1,2-Epoxides by Thiophenol in Aqueous Medium by Amantini, David, Fringuelli, Francesco, Pizzo, Ferdinando, Tortoioli, Simone, Vaccaro, Luigi

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Blepharo-cheilo-dontic (BCD) syndrome: Report on four new patients by Guion-Almeida, M.L., Rodini, E.S.O., Kokitsu-Nakata, N.M., Bologna-Amantini, D.

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Nucleophilic ring opening of 1,2-epoxides in aqueous medium by Amantini, David, Fringuelli, Francesco, Piermatti, Oriana, Tortoioli, Simone, Vaccaro, Luigi

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Cortical Blindness After Cardiac Surgery: Just an Ischemic Mechanism? by Scarpino, Maenia, MD, Olivo, Giuseppe, MD, Quilghini, Pietro, MD, Lanzo, Giovanni, Phd, Moretti, Marco, MD, Carrai, Riccardo, MD, Fontanari, Paolo, MD, Amantini, Aldo, MD, Grippo, Antonello, MD

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Extracellular Vesicles in the Cornea: Insights from Other Tissues by McKay, Tina B., Yeung, Vincent, Hutcheon, Audrey E. K., Guo, Xiaoqing, Zieske, James D., Ciolino, Joseph B.

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The CAESAR Project for the ASI Space Weather Infrastructure by Laurenza, M., Del Moro, D., Alberti, T., Battiston, R., Benella, S., Benvenuto, F., Berrilli, F., Bertello, I., Bertucci, B., Biasiotti, L., Campi, C., Carbone, V., Casolino, M., Cecchi Pestellini, C., Chiappetta, F., Coco, I., Colombo, S., Consolini, G., D’Amicis, R., De Gasperis, G., De Marco, R., Del Corpo, A., Diego, P., Di Felice, V., Di Fino, L., Di Geronimo, C., Faldi, F., Ferrente, F., Feruglio, C., Fiandrini, E., Fiore, F., Foldes, R., Formato, V., Francisco, G., Giannattasio, F., Giardino, M., Giobbi, P., Giovannelli, L., Giusti, M., Gorgi, A., Heilig, B., Iafrate, G., Ivanovski, S. L., Jerse, G., Korsos, M. B., Lepreti, F., Locci, D., Magnafico, C., Mangano, V., Marcucci, M. F., Martucci, M., Massetti, S., Micela, G., Milillo, A., Miteva, R., Molinaro, M., Mugatwala, R., Mura, A., Napoletano, G., Narici, L., Neubüser, C., Nisticò, G., Pauluzzi, M., Perfetti, A., Perri, S., Petralia, A., Pezzopane, M., Piersanti, M., Pietropaolo, E., Pignalberi, A., Plainaki, C., Polenta, G., Primavera, L., Romoli, G., Rossi, M., Santarelli, L., Santi Amantini, G., Siciliano, F., Sindoni, G., Spadoni, S., Sparvoli, R., Stumpo, M., Tomassetti, N., Tozzi, R., Vagelli, V., Vasantharaju, N., Vecchio, A., Vellante, M., Vernetto, S., Vigorito, C., West, M. J., Zimbardo, G., Zucca, P., Zuccarello, F., Zuccon, P.

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Guidelines for the use and interpretation of assays for monitoring autophagy (4th edition) by Klionsky, Daniel, Abdel-Aziz, Amal Kamal, Abdelfatah, Sara, Abdellatif, Mahmoud, Abdoli, Asghar, Abel, Steffen, Abeliovich, Hagai, Abildgaard, Marie, Abudu, Yakubu Princely, Acevedo-Arozena, Abraham, Adamopoulos, Iannis, Adeli, Khosrow, Adolph, Timon, Adornetto, Annagrazia, Aflaki, Elma, Agam, Galila, Agarwal, Anupam, Aggarwal, Bharat, Agnello, Maria, Agostinis, Patrizia, Agrewala, Javed, Agrotis, Alexander, Aguilar, Patricia, Ahmad, S. Tariq, Ahmed, Zubair, Ahumada-Castro, Ulises, Aits, Sonja, Aizawa, Shu, Akkoc, Yunus, Akoumianaki, Tonia, Akpinar, Hafize Aysin, Al-Abd, Ahmed, Al-Akra, Lina, Al-Gharaibeh, Abeer, Alaoui-Jamali, Moulay, Alberti, Simon, Alcocer-Gómez, Elísabet, Alessandri, Cristiano, Ali, Muhammad, Alim Al-Bari, M. Abdul, Aliwaini, Saeb, Alizadeh, Javad, Almacellas, Eugènia, Almasan, Alexandru, Alonso, Alicia, Alonso, Guillermo, Altan-Bonnet, Nihal, Altieri, Dario, Álvarez, Élida, Alves, Sara, Alves da Costa, Cristine, Alzaharna, Mazen, Amadio, Marialaura, Amantini, Consuelo, Amaral, Cristina, Ambrosio, Susanna, Amer, Amal, Ammanathan, Veena, An, Zhenyi, Andersen, Stig, Andrabi, Shaida, Andrade-Silva, Magaiver, Andres, Allen, Angelini, Sabrina, Ann, David, Anozie, Uche, Ansari, Mohammad, Antas, Pedro, Antebi, Adam, Antón, Zuriñe, Anwar, Tahira, Apetoh, Lionel, Apostolova, Nadezda, Araki, Toshiyuki, Araki, Yasuhiro, Arasaki, Kohei, Araújo, Wagner, Araya, Jun, Arden, Catherine, Arévalo, Maria-Angeles, Arguelles, Sandro, Arias, Esperanza, Arikkath, Jyothi, Arimoto, Hirokazu, Ariosa, Aileen, Armstrong-James, Darius, Arnauné-Pelloquin, Laetitia, Aroca, Angeles, Arroyo, Daniela, Arsov, Ivica, Artero, Rubén, Asaro, Dalia Maria Lucia, Aschner, Michael, Ashrafizadeh, Milad, Ashur-Fabian, Osnat, Atanasov, Atanas, Au, Alicia, Auberger, Patrick, Auner, Holger, Aurelian, Laure

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The Italian technical/administrative recommendations for telemedicine in clinical neurophysiology by Stipa, G., Gabbrielli, F., Rabbito, C., Di Lazzaro, V., Amantini, A., Grippo, A., Carrai, R., Pasqui, R., Barloscio, D., Olivi, D., Lori, S.

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Radiation measurements in the International Space Station, Columbus module, in 2020–2022 with the LIDAL detector by Di Fino, L., Romoli, G., Santi Amantini, G., Boretti, V., Lunati, L., Berucci, C., Messi, R., Rizzo, A., Albicocco, P., De Donato, C., Masciantonio, G., Morone, M.C., Nobili, G., Baiocco, G., Mentana, A., Pullia, M., Tommasino, F., Carrubba, E., Bardi, A., Passerai, M., Castagnolo, D., Mascetti, G., Crisconio, M., Matthiä, D., Narici, L.

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