Encoded Library Technology as a Source of Hits for the Discovery and Lead Optimization of a Potent and Selective Class of Bactericidal Direct Inhibitors of Mycobacterium tuberculos... by Encinas, Lourdes, O’Keefe, Heather, Neu, Margarete, Remuiñán, Modesto J, Patel, Amish M, Guardia, Ana, Davie, Christopher P, Pérez-Macías, Natalia, Yang, Hongfang, Convery, Maire A, Messer, Jeff A, Pérez-Herrán, Esther, Centrella, Paolo A, Álvarez-Gómez, Daniel, Clark, Matthew A, Huss, Sophie, O’Donovan, Gary K, Ortega-Muro, Fátima, McDowell, William, Castañeda, Pablo, Arico-Muendel, Christopher C, Pajk, Stane, Rullás, Joaquín, Angulo-Barturen, Iñigo, Álvarez-Ruíz, Emilio, Mendoza-Losana, Alfonso, Ballell Pages, Lluís, Castro-Pichel, Julia, Evindar, Ghotas

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The repurposing of Tebipenem pivoxil as alternative therapy for severe gastrointestinal infections caused by extensively drug-resistant Shigella spp by Fernández Álvaro, Elena, Voong Vinh, Phat, de Cozar, Cristina, Willé, David R, Urones, Beatriz, Cortés, Alvaro, Price, Alan, Tran Do Hoang, Nhu, Ha Thanh, Tuyen, McCloskey, Molly, Shaheen, Shareef, Dayao, Denise, Martinot, Amanda, de Mercado, Jaime, Castañeda, Pablo, García-Perez, Adolfo, Singa, Benson, Pavlinac, Patricia, Walson, Judd, Martínez-Martínez, Maria Santos, Arnold, Samuel L M, Tzipori, Saul, Ballell Pages, Lluis, Baker, Stephen

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N-Benzyl-4-((heteroaryl)methyl)benzamides: A New Class of Direct NADH-Dependent 2-trans Enoyl-Acyl Carrier Protein Reductase (InhA) Inhibitors with Antitubercular Activity by Guardia, Ana, Gulten, Gulcin, Fernandez, Raquel, Gómez, Jesus, Wang, Feng, Convery, Maire, Blanco, Delia, Martínez, María, Pérez-Herrán, Esther, Alonso, Marta, Ortega, Fátima, Rullás, Joaquín, Calvo, David, Mata, Lydia, Young, Robert, Sacchettini, James C., Mendoza-Losana, Alfonso, Remuiñán, Modesto, Ballell Pages, Lluís, Castro-Pichel, Julia

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Correction: The repurposing of Tebipenem pivoxil as alternative therapy for severe gastrointestinal infections caused by extensively drug-resistant Shigella spp by Fernández Álvaro, Elena, Voong Vinh, Phat, de Cozar, Cristina, Willé, David R, Urones, Beatriz, Cortés, Alvaro, Price, Alan, Tran Do Hoang, Nhu, Ha Thanh, Tuyen, McCloskey, Molly, Shaheen, Shareef, Dayao, Denise, Martinot, Amanda, de Mercado, Jaime, Castañeda, Pablo, García-Perez, Adolfo, Singa, Benson, Pavlinac, Patricia, Walson, Judd, Martínez-Martínez, Maria Santos, Arnold, Samuel LM, Tzipori, Saul, Pages, Lluis Ballell, Baker, Stephen

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Design, Synthesis, and Evaluation of New Thiadiazole-Based Direct Inhibitors of Enoyl Acyl Carrier Protein Reductase (InhA) for the Treatment of Tuberculosis by Šink, Roman, Sosič, Izidor, Živec, Matej, Fernandez-Menendez, Raquel, Turk, Samo, Pajk, Stane, Alvarez-Gomez, Daniel, Lopez-Roman, Eva Maria, Gonzales-Cortez, Carolina, Rullas-Triconado, Joaquin, Angulo-Barturen, Inigo, Barros, David, Ballell-Pages, Lluís, Young, Robert J, Encinas, Lourdes, Gobec, Stanislav

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Design, synthesis and structure-activity relationship study of wollamide B; a new potential anti TB agent by Asfaw, Henok, Laqua, Katja, Walkowska, Anna Maria, Cunningham, Fraser, Martinez-Martinez, Maria Santos, Cuevas-Zurita, Juan Carlos, Ballell-Pages, Lluís, Imming, Peter

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High-content screening technology combined with a human granuloma model as a new approach to evaluate the activities of drugs against Mycobacterium tuberculosis by Silva-Miranda, Mayra, Ekaza, Euloge, Breiman, Adrien, Asehnoune, Karim, Barros-Aguirre, David, Pethe, Kevin, Ewann, Fanny, Brodin, Priscille, Ballell-Pages, Lluís, Altare, Frédéric

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Testing tuberculosis drug efficacy in a zebrafish high-throughput translational medicine screen by Ordas, Anita, Raterink, Robert-Jan, Cunningham, Fraser, Jansen, Hans J, Wiweger, Malgorzata I, Jong-Raadsen, Susanne, Bos, Sabine, Bates, Robert H, Barros, David, Meijer, Annemarie H, Vreeken, Rob J, Ballell-Pages, Lluís, Dirks, Ron P, Hankemeier, Thomas, Spaink, Herman P

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New direct inhibitors of InhA with antimycobacterial activity based on a tetrahydropyran scaffold by Pajk, Stane, Živec, Matej, Šink, Roman, Sosič, Izidor, Neu, Margarete, Chung, Chun-wa, Martínez-Hoyos, María, Pérez-Herrán, Esther, Álvarez-Gómez, Daniel, Álvarez-Ruíz, Emilio, Mendoza-Losana, Alfonso, Castro-Pichel, Julia, Barros, David, Ballell-Pages, Lluís, Young, Robert J., Convery, Maire A., Encinas, Lourdes, Gobec, Stanislav

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A Developability-Focused Optimization Approach Allows Identification of in Vivo Fast-Acting Antimalarials: N‑[3-[(Benzimidazol-2-yl)amino]propyl]amides by Keurulainen, Leena, Vahermo, Mikko, Puente-Felipe, Margarita, Sandoval-Izquierdo, Elena, Crespo-Fernández, Benigno, Guijarro-López, Laura, Huertas-Valentín, Leticia, de las Heras-Dueña, Laura, Leino, Teppo O, Siiskonen, Antti, Ballell-Pages, Lluís, Sanz, Laura M, Castañeda-Casado, Pablo, Jiménez-Díaz, M. Belén, Martínez-Martínez, María S, Viera, Sara, Kiuru, Paula, Calderón, Félix, Yli-Kauhaluoma, Jari

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Carbamoyl Triazoles, Known Serine Protease Inhibitors, Are a Potent New Class of Antimalarials by McConville, Matthew, Fernández, Jorge, Angulo-Barturen, Íñigo, Bahamontes-Rosa, Noemi, Ballell-Pages, Lluis, Castañeda, Pablo, de Cózar, Cristina, Crespo, Benigno, Guijarro, Laura, Jiménez-Díaz, María Belén, Martínez-Martínez, Maria S, de Mercado, Jaime, Santos-Villarejo, Ángel, Sanz, Laura M, Frigerio, Micol, Washbourn, Gina, Ward, Stephen A, Nixon, Gemma L, Biagini, Giancarlo A, Berry, Neil G, Blackman, Michael J, Calderón, Félix, O’Neill, Paul M

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