Galantamine-memantine hybrids for Alzheimer's disease: The influence of linker rigidity in biological activity and pharmacokinetic properties by Basagni, Filippo, Ortega, Jose A., Bertozzi, Sine M., Armirotti, Andrea, Summa, Maria, Bertorelli, Rosalia, Bartolini, Manuela, Mellor, Ian R., Bedeschi, Martina, Bottegoni, Giovanni, Lembo, Vittorio, Minarini, Anna, Cavalli, Andrea, Rosini, Michela

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Anterior insula stimulation suppresses appetitive behavior while inducing forebrain activation in alcohol-preferring rats by Haaranen, Mia, Scuppa, Giulia, Tambalo, Stefano, Järvi, Vilja, Bertozzi, Sine M., Armirotti, Andrea, Sommer, Wolfgang H., Bifone, Angelo, Hyytiä, Petri

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Structural determinants of peripheral O-arylcarbamate FAAH inhibitors render them dual substrates for Abcb1 and Abcg2 and restrict their access to the brain by Moreno-Sanz, Guillermo, Barrera, Borja, Armirotti, Andrea, Bertozzi, Sine M., Scarpelli, Rita, Bandiera, Tiziano, Prieto, Julio G., Duranti, Andrea, Tarzia, Giorgio, Merino, Gracia, Piomelli, Daniele

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Discovery of a class of calcium sensing receptor positive allosteric modulators; 1-(benzothiazol-2-yl)-1-phenylethanols by Gustafsson, Magnus, Jensen, Jacob, Bertozzi, Sine M., Currier, Erika A., Ma, Jian-Nong, Burstein, Ethan S., Olsson, Roger

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Identification of novel selective v2 receptor non-peptide agonists by DEL TREDID, Andria L, VANOVER, Kim E, MOHELL, Nina, OLSSON, Roger, PIN, Fabrice, KNAPP, Anne E, BERTOZZI, Sine M, NASH, Norman R, BURSTEIN, Ethan S, LAMEH, Jelveh, CURRIER, Erika A, DAVIS, Robert E, BRANN, Mark R

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Identification of novel selective V 2 receptor non-peptide agonists by Del Tredici, Andria L., Vanover, Kim E., Knapp, Anne E., Bertozzi, Sine M., Nash, Norman R., Burstein, Ethan S., Lameh, Jelveh, Currier, Erika A., Davis, Robert E., Brann, Mark R., Mohell, Nina, Olsson, Roger, Piu, Fabrice

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Structure-based design of CDC42 effector interaction inhibitors for the treatment of cancer by Jahid, Sohail, Ortega, Jose A., Vuong, Linh M., Acquistapace, Isabella Maria, Hachey, Stephanie J., Flesher, Jessica L., La Serra, Maria Antonietta, Brindani, Nicoletta, La Sala, Giuseppina, Manigrasso, Jacopo, Arencibia, Jose M., Bertozzi, Sine Mandrup, Summa, Maria, Bertorelli, Rosalia, Armirotti, Andrea, Jin, Rongsheng, Liu, Zheng, Chen, Chi-Fen, Edwards, Robert, Hughes, Christopher C.W., De Vivo, Marco, Ganesan, Anand K.

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Design, Synthesis, In Vitro and In Vivo Characterization of CDC42 GTPase Interaction Inhibitors for the Treatment of Cancer by Brindani, Nicoletta, Vuong, Linh M., Acquistapace, Isabella Maria, La Serra, Maria Antonietta, Ortega, José Antonio, Veronesi, Marina, Bertozzi, Sine Mandrup, Summa, Maria, Girotto, Stefania, Bertorelli, Rosalia, Armirotti, Andrea, Ganesan, Anand K., De Vivo, Marco

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Discovery of CDC42 Inhibitors with a Favorable Pharmacokinetic Profile and Anticancer In Vivo Efficacy by Brindani, Nicoletta, Vuong, Linh M., La Serra, Maria Antonietta, Salvador, Noel, Menichetti, Andrea, Acquistapace, Isabella Maria, Ortega, Jose Antonio, Veronesi, Marina, Bertozzi, Sine Mandrup, Summa, Maria, Girotto, Stefania, Bertorelli, Rosalia, Armirotti, Andrea, Ganesan, Anand K., De Vivo, Marco

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Novel, Potent, and Druglike Tetrahydroquinazoline Inhibitor That Is Highly Selective for Human Topoisomerase II α over β by Ortega, Jose Antonio, Arencibia, Jose M, Minniti, Elirosa, Byl, Jo Ann W, Franco-Ulloa, Sebastian, Borgogno, Marco, Genna, Vito, Summa, Maria, Bertozzi, Sine Mandrup, Bertorelli, Rosalia, Armirotti, Andrea, Minarini, Anna, Sissi, Claudia, Osheroff, Neil, De Vivo, Marco

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Design, Synthesis, Dynamic Docking, Biochemical Characterization, and in Vivo Pharmacokinetics Studies of Novel Topoisomerase II Poisons with Promising Antiproliferative Activity by Arencibia, Jose M, Brindani, Nicoletta, Franco-Ulloa, Sebastian, Nigro, Michela, Kuriappan, Jissy Akkarapattiakal, Ottonello, Giuliana, Bertozzi, Sine Mandrup, Summa, Maria, Girotto, Stefania, Bertorelli, Rosalia, Armirotti, Andrea, De Vivo, Marco

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Structure-based design of CDC42 effector interaction inhibitors for the treatment of cancer by Jahid, Sohail, Ortega, Jose A., Vuong, Linh M., Acquistapace, Isabella Maria, Hachey, Stephanie J., Flesher, Jessica L., La Serra, Maria Antonietta, Brindani, Nicoletta, La Sala, Giuseppina, Manigrasso, Jacopo, Arencibia, Jose M., Bertozzi, Sine Mandrup, Summa, Maria, Bertorelli, Rosalia, Armirotti, Andrea, Jin, Rongsheng, Liu, Zheng, Chen, Chi-Fen, Edwards, Robert, Hughes, Christopher C.W., De Vivo, Marco, Ganesan, Anand K.

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