Imidazopyridine-Based 5-HT 6 Receptor Neutral Antagonists: Impact of N 1 -Benzyl and N 1 -Phenylsulfonyl Fragments on Different Receptor Conformational States by Vanda, David, Canale, Vittorio, Chaumont-Dubel, Severine, Kurczab, Rafał, Satała, Grzegorz, Koczurkiewicz-Adamczyk, Paulina, Krawczyk, Martyna, Pietruś, Wojciech, Blicharz, Klaudia, Pękala, Elżbieta, Bojarski, Andrzej J, Popik, Piotr, Marin, Philippe, Soural, Miroslav, Zajdel, Paweł

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1-(Arylsulfonyl-isoindol-2-yl)piperazines as 5-HT6R Antagonists: Mechanochemical Synthesis, In Vitro Pharmacological Properties and Glioprotective Activity by Canale, Vittorio, Trybała, Wojciech, Chaumont-Dubel, Séverine, Koczurkiewicz-Adamczyk, Paulina, Satała, Grzegorz, Bento, Ophélie, Blicharz-Futera, Klaudia, Bantreil, Xavier, Pękala, Elżbieta, Bojarski, Andrzej J., Lamaty, Frédéric, Marin, Philippe, Zajdel, Paweł

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Imidazopyridine-Based 5‑HT6 Receptor Neutral Antagonists: Impact of N 1‑Benzyl and N 1‑Phenylsulfonyl Fragments on Different Receptor Conformational States by Vanda, David, Canale, Vittorio, Chaumont-Dubel, Severine, Kurczab, Rafał, Satała, Grzegorz, Koczurkiewicz-Adamczyk, Paulina, Krawczyk, Martyna, Pietruś, Wojciech, Blicharz, Klaudia, Pękala, Elżbieta, Bojarski, Andrzej J, Popik, Piotr, Marin, Philippe, Soural, Miroslav, Zajdel, Paweł

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A dual-acting 5-HT6 receptor inverse agonist/MAO-B inhibitor displays glioprotective and pro-cognitive properties by Canale, Vittorio, Grychowska, Katarzyna, Kurczab, Rafał, Ryng, Mateusz, Keeri, Abdul Raheem, Satała, Grzegorz, Olejarz-Maciej, Agnieszka, Koczurkiewicz, Paulina, Drop, Marcin, Blicharz, Klaudia, Piska, Kamil, Pękala, Elżbieta, Janiszewska, Paulina, Krawczyk, Martyna, Walczak, Maria, Chaumont-Dubel, Severine, Bojarski, Andrzej J., Marin, Philippe, Popik, Piotr, Zajdel, Paweł

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Overcoming undesirable hERG affinity by incorporating fluorine atoms: A case of MAO-B inhibitors derived from 1 H-pyrrolo-[3,2-c]quinolines by Grychowska, Katarzyna, Olejarz-Maciej, Agnieszka, Blicharz, Klaudia, Pietruś, Wojciech, Karcz, Tadeusz, Kurczab, Rafał, Koczurkiewicz, Paulina, Doroz-Płonka, Agata, Latacz, Gniewomir, Keeri, Abdul Raheem, Piska, Kamil, Satała, Grzegorz, Pęgiel, Joanna, Trybała, Wojciech, Jastrzębska-Więsek, Magdalena, Bojarski, Andrzej J., Lamaty, Frédéric, Partyka, Anna, Walczak, Maria, Krawczyk, Martyna, Malikowska-Racia, Natalia, Popik, Piotr, Zajdel, Paweł

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A dual-acting 5-HT 6 receptor inverse agonist/MAO-B inhibitor displays glioprotective and pro-cognitive properties by Canale, Vittorio, Grychowska, Katarzyna, Kurczab, Rafał, Ryng, Mateusz, Keeri, Abdul Raheem, Keeri, Abdul Raheem, Satała, Grzegorz, Olejarz-Maciej, Agnieszka, Koczurkiewicz, Paulina, Drop, Marcin, Blicharz, Klaudia, Piska, Kamil, Pękala, Elżbieta, Janiszewska, Paulina, Krawczyk, Martyna, Walczak, Maria, Chaumont-Dubel, Séverine, Bojarski, Andrzej J, Marin, Philippe, Popik, Piotr, Zajdel, Paweł

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5-HT6 receptor neutral antagonists protect astrocytes: A lesson from 2-phenylpyrrole derivatives by Drop, Marcin, Koczurkiewicz-Adamczyk, Paulina, Bento, Ophélie, Pietruś, Wojciech, Satała, Grzegorz, Blicharz-Futera, Klaudia, Canale, Vittorio, Grychowska, Katarzyna, Bantreil, Xavier, Pękala, Elżbieta, Kurczab, Rafał, Bojarski, Andrzej J., Chaumont-Dubel, Severine, Marin, Philippe, Lamaty, Frédéric, Zajdel, Paweł

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Superiority of the Triple-Acting 5-HT 6 R/5-HT 3 R Antagonist and MAO-B Reversible Inhibitor PZ-1922 over 5-HT 6 R Antagonist Intepirdine in Alleviation of Cognitive Deficits in Ra... by Grychowska, Katarzyna, López-Sánchez, Uriel, Vitalis, Mathieu, Canet, Geoffrey, Satała, Grzegorz, Olejarz-Maciej, Agnieszka, Gołębiowska, Joanna, Kurczab, Rafał, Pietruś, Wojciech, Kubacka, Monika, Moreau, Christophe, Walczak, Maria, Blicharz-Futera, Klaudia, Bento, Ophélie, Bantreil, Xavier, Subra, Gilles, Bojarski, Andrzej J., Lamaty, Frédéric, Becamel, Carine, Zussy, Charleine, Chaumont-Dubel, Séverine, Popik, Piotr, Nury, Hugues, Marin, Philippe, Givalois, Laurent, Zajdel, Paweł

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Superiority of the Triple-Acting 5‑HT6R/5-HT3R Antagonist and MAO‑B Reversible Inhibitor PZ-1922 over 5‑HT6R Antagonist Intepirdine in Alleviation of Cognitive Deficits in Rats... by Grychowska, Katarzyna, López-Sánchez, Uriel, Vitalis, Mathieu, Canet, Geoffrey, Satała, Grzegorz, Olejarz-Maciej, Agnieszka, Gołębiowska, Joanna, Kurczab, Rafał, Pietruś, Wojciech, Kubacka, Monika, Moreau, Christophe, Walczak, Maria, Blicharz-Futera, Klaudia, Bento, Ophélie, Bantreil, Xavier, Subra, Gilles, Bojarski, Andrzej J., Lamaty, Frédéric, Becamel, Carine, Zussy, Charleine, Chaumont-Dubel, Séverine, Popik, Piotr, Nury, Hugues, Marin, Philippe, Givalois, Laurent, Zajdel, Paweł

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5-HT 6 receptor neutral antagonists protect astrocytes: A lesson from 2-phenylpyrrole derivatives by Drop, Marcin, Koczurkiewicz-Adamczyk, Paulina, Bento, Ophélie, Pietruś, Wojciech, Satała, Grzegorz, Blicharz-Futera, Klaudia, Canale, Vittorio, Grychowska, Katarzyna, Bantreil, Xavier, Pękala, Elżbieta, Kurczab, Rafał, Bojarski, Andrzej J, Chaumont-Dubel, Severine, Marin, Philippe, Lamaty, Frédéric, Zajdel, Paweł

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1-(Arylsulfonyl-isoindol-2-yl)piperazines as 5-HT 6 R Antagonists: Mechanochemical Synthesis, In Vitro Pharmacological Properties and Glioprotective Activity by Canale, Vittorio, Trybała, Wojciech, Chaumont-Dubel, Séverine, Koczurkiewicz-Adamczyk, Paulina, Satała, Grzegorz, Bento, Ophélie, Blicharz-Futera, Klaudia, Bantreil, Xavier, Pękala, Elżbieta, Bojarski, Andrzej J, Lamaty, Frédéric, Marin, Philippe, Zajdel, Paweł

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