Abstract 1342: Development and preclinical evaluation of unique first-in-class small molecule inhibitors of the anti-apoptotic protein FLIP by Higgins, Catherine A., Fox, Jennifer, Roberts, Jamie, Doherty, Declan, Perrior, Trevor, Boffey, Ray, Harrison, Tim, Longley, Daniel B.

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Abstract 5220: Development of first-in-class small molecule inhibitors of FLIP which activate caspase-8, the nodal regulator of apoptosis, necroptosis and pyroptosis by Longley, Daniel B., Higgins, Catherine, Fox, Jennifer, Roberts, Jamie Z., Boffey, Ray, Williams, Sophie, Perrior, Trevor, Page, Martin J., Harrison, Tim

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Abstract 382: Development and pre-clinical assessment of a first-in-class small molecule inhibitor of FLIP by Higgins, Catherine A., Fox, Jennifer, Majkut, Joanna, Fiedler, Greti E., Roberts, Jamie, Humphreys, Luke, Boffey, Ray J., Perrior, Trevor R., Harrison, Timothy, Longley, Daniel B.

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Abstract B129: Development and preclinical assessment of a first-in-class small-molecule inhibitor of FLIP by Higgins, Catherine A., Majkut, Joanna, Fox, Jennifer, Humphreys, Luke, Fiedler, Greti Espona, Boffey, Ray J., Perrior, Trevor R., Haigh, David, Harrison, Timothy, Longley, Daniel B.

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Abstract LB-037: Development and preclinical assessment of a first-in-class small molecule inhibitor of the major cell death regulator protein FLIP by Majkut, Joanna, Higgins, Catherine, Malik, Adnan, Nemeth, Zsusannah, Blurton, Peter, Boffey, Ray, Perrior, Trevor R., Johnston, Patrick G., Haigh, David, Harrison, Timothy, Longley, Daniel B.

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Synthesis and SAR studies of analogues of 4-(3,3-dimethyl-butyrylamino)-3,5-difluoro-N-thiazol-2-yl-benzamide (Lu AA41063) as adenosine A2A receptor ligands with improved aqueous s... by Mikkelsen, Gitte Kobberøe, Langgård, Morten, Schrøder, Tenna Juul, Kreilgaard, Mads, Jørgensen, Erling B., Brandt, Guillaume, Griffon, Yann, Boffey, Ray, Bang-Andersen, Benny

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Abstract C5: FLIP protein-protein interaction inhibitors enhance sensitivity of colorectal cancer cells to chemotherapy and TRAIL by Fox, Jennifer P., Majkut, Joanna, Higgins, Catherine, Nemeth, Zsuzsanna, Malik, Adnan, Scott, Christopher J., Blurton, Peter, Boffey, Ray J., Perrior, Trevor R., Harrison, Timothy, Longley, Daniel B.

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Abstract C4: Development and pre-clinical assessment of a first-in-class small molecule inhibitor of FLIP for treatment of NSCLC by Majkut, Joanna, Higgins, Catherine, Malik, Adnan, Nemeth, Zsusannah, Blurton, Peter, Boffey, Ray J., Perrior, Trevor R., Haigh, David, Harrison, Timothy, Longley, Daniel B.

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Design and discovery of 3-aryl-5-substituted-isoquinolin-1-ones as potent tankyrase inhibitors by Elliott, Richard J. R., Jarvis, Ashley, Rajasekaran, Mohan B., Menon, Malini, Bowers, Leandra, Boffey, Ray, Bayford, Melanie, Firth-Clark, Stuart, Key, Rebekah, Aqil, Rehan, Kirton, Stewart B., Niculescu-Duvaz, Dan, Fish, Laura, Lopes, Filipa, McLeary, Robert, Trindade, Ines, Vendrell, Elisenda, Munkonge, Felix, Porter, Rod, Perrior, Trevor, Springer, Caroline, Oliver, Antony W., Pearl, Laurence H., Ashworth, Alan, Lord, Christopher J.

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Design and discovery of 3-aryl-5-substituted-isoquinolin-1-ones as potent tankyrase inhibitorsElectronic supplementary information (ESI) available: For complete experimental detail... by Elliott, Richard J. R, Jarvis, Ashley, Rajasekaran, Mohan B, Menon, Malini, Bowers, Leandra, Boffey, Ray, Bayford, Melanie, Firth-Clark, Stuart, Key, Rebekah, Aqil, Rehan, Kirton, Stewart B, Niculescu-Duvaz, Dan, Fish, Laura, Lopes, Filipa, McLeary, Robert, Trindade, Ines, Vendrell, Elisenda, Munkonge, Felix, Porter, Rod, Perrior, Trevor, Springer, Caroline, Oliver, Antony W, Pearl, Laurence H, Ashworth, Alan, Lord, Christopher J

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Design, synthesis and characterization of a novel class of coumarin-based inhibitors of inducible nitric oxide synthase by Jackson, Sharon A., Sahni, Sukhveen, Lee, Lan, Luo, Yongyi, Nieduzak, Thaddeus R., Liang, Guyan, Chiang, Yulin, Collar, Nicola, Fink, David, He, Wei, Laoui, Abdelazize, Merrill, Jean, Boffey, Ray, Crackett, Peter, Rees, Bryan, Wong, Melanie, Guilloteau, Jean-Pierre, Mathieu, Magali, Rebello, Sam S.

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