Assessment of the antinociceptive, respiratory-depressant, and reinforcing effects of the low pKa fluorinated fentanyl analogs, FF3 and NFEPP by Edwards, Shelley R., Blough, Bruce E., Cowart, Kristian, Howell, Grace H., Araujo, Aaron A., Haskell, Jacob P., Huskinson, Sally L., Rowlett, James K., Brackeen, Marcus F., Freeman, Kevin B.

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Assessment of the Antinociceptive, Respiratory-Depressant, and Reinforcing Effects of the Low pK a Fluorinated Fentanyl Analogs, FF3 and NFEPP by Edwards, Shelley R, Blough, Bruce E, Cowart, Kristian, Howell, Grace H, Araujo, Aaron A, Haskell, Jacob P, Huskinson, Sally L, Rowlett, James K, Brackeen, Marcus F, Freeman, Kevin B

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Identification of a Potent Human Trace Amine-Associated Receptor 1 Antagonist by Decker, Ann M, Brackeen, Marcus F, Mohammadkhani, Aida, Kormos, Chad M, Hesk, David, Borgland, Stephanie L, Blough, Bruce E

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Design and Synthesis of Conformationally Constrained Analogs of 4-(3-Butoxy-4-methoxybenzyl)imidazolidin-2-one (Ro 20-1724) as Potent Inhibitors of cAMP-Specific Phosphodiesterase by Brackeen, Marcus F, Stafford, Jeffrey A, Cowan, David J, Brown, Peter J, Domanico, Paul L, Feldman, Paul L, Rose, Dudley, Strickland, Alan B, Veal, James M, Verghese, Margrith

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Design, synthesis, and pharmacological evaluation of ultrashort- to long-acting opioid analgesics by Feldman, Paul L, James, Michael K, Brackeen, Marcus F, Bilotta, Joanne M, Schuster, Suzanne V, Lahey, Avis P, Lutz, Michael W, Johnson, M. Ross, Leighton, H. Jeff

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Phosphodiesterase Type IV Inhibition. Structure-Activity Relationships of 1,3-Disubstituted Pyrrolidines by Feldman, Paul L, Brackeen, Marcus F, Cowan, David J, Marron, Brian E, Schoenen, Frank J, Stafford, Jeffrey A, Suh, Edward M, Domanico, Paul L, Rose, Dudley

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N-(2-Benzoylphenyl)-l-tyrosine PPARγ Agonists. 1. Discovery of a Novel Series of Potent Antihyperglycemic and Antihyperlipidemic Agents by Henke, Brad R, Blanchard, Steven G, Brackeen, Marcus F, Brown, Kathleen K, Cobb, Jeff E, Collins, Jon L, Harrington, W. Wallace, Hashim, Mir A, Hull-Ryde, Emily A, Kaldor, Istvan, Kliewer, Steven A, Lake, Debra H, Leesnitzer, Lisa M, Lehmann, Jürgen M, Lenhard, James M, Orband-Miller, Lisa A, Miller, John F, Mook, Robert A, Noble, Stewart A, Oliver, William, Parks, Derek J, Plunket, Kelli D, Szewczyk, Jerzy R, Willson, Timothy M

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Introduction of a conformational switching element on a pyrrolidine ring. Synthesis and evaluation of methyl (R,R)-(.+-.)-3-acetyl-4-[3- (cyclopentyloxy)-4-methoxyphenyl]-3- methyl... by Stafford, Jeffrey A, Veal, James M, Feldman, Paul L, Valvano, Nicole L, Baer, Philip G, Brackeen, Marcus F, Brawley, E. Sloan, Connolly, Kevin M, Domanico, Paul L

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Design, synthesis, and pharmacological evaluation of ultrashort- to long-acting opioid analgetics by FELDMAN, P. L, JAMES, M. K, BRACKEEN, M. F, BILOTTA, J. M, SCHUSTER, S. V, LAHEY, A. P, LUTZ, M. W, JOHNSON, M. R, LEIGHTON, H. J

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A novel route to the 4-anilido-4-(methoxycarbonyl)piperidine class of analgetics by Feldman, Paul L., Brackeen, Marcus F.

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Evaluation of cannabimimetic effects of selected minor cannabinoids and Terpenoids in mice by Wiley, Jenny L., Marusich, Julie A., Blough, Bruce E., Namjoshi, Ojas, Brackeen, Marcus, Akinfiresoye, Luli R., Walker, Teneille D., Prioleau, Cassandra, Barrus, Daniel G., Gamage, Thomas F.

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Conformationally Constrained Analogues of N-(Piperidinyl)-5-(4-Chlorophenyl)-1-(2,4- Dichlorophenyl)-4-Methyl-1H-Pyrazole-3-Carboxamide (SR141716): Design, Synthesis, Computational... by Zhang, Yanan, Burgess, Jason P, Brackeen, Marcus, Gilliam, Anne, Mascarella, S. Wayne, Page, Kevin, Seltzman, Herbert H, Thomas, Brian F

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Conformationally Constrained Analogues of N -(Piperidinyl)-5-(4-Chlorophenyl)-1-(2,4- Dichlorophenyl)-4-Methyl-1 H -Pyrazole-3-Carboxamide (SR141716): Design, Synthesis, Computatio... by Zhang, Yanan, Burgess, Jason P., Brackeen, Marcus, Gilliam, Anne, Mascarella, S. Wayne, Page, Kevin, Seltzman, Herbert H., Thomas, Brian F.

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Conformational characteristics of the interaction of SR141716A with the CB1 cannabinoid receptor as determined through the use of conformationally constrained analogs by Thomas, Brian F, Zhang, Yanan, Brackeen, Marcus, Page, Kevin M, Mascarella, S Wayne, Seltzman, Herbert H

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