Development of Orally Bioavailable Bicyclic Pyrazolones as Inhibitors of Tumor Necrosis Factor-α Production by Clark, Michael P, Laughlin, Steven K, Laufersweiler, Matthew J, Bookland, Roger G, Brugel, Todd A, Golebiowski, Adam, Sabat, Mark P, Townes, Jennifer A, VanRens, John C, Djung, Jane F, Natchus, Michael G, De, Biswanath, Hsieh, Lily C, Xu, Susan C, Walter, Rick L, Mekel, Marlene J, Heitmeyer, Sandra A, Brown, Kimberly K, Juergens, Karen, Taiwo, Yetunde O, Janusz, Michael J

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The development of new isoxazolone based inhibitors of tumor necrosis factor-alpha (TNF-α) production by Laughlin, Steven K., Clark, Michael P., Djung, Jane F., Golebiowski, Adam, Brugel, Todd A., Sabat, Mark, Bookland, Roger G., Laufersweiler, Matthew J., VanRens, John C., Townes, Jennifer A., De, Biswanath, Hsieh, Lily C., Xu, Susan C., Walter, Richard L., Mekel, Marlene J., Janusz, Michael J.

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Intramolecular Diels−Alder Cyclizations of (E)-1-Nitro-1,7,9-decatrienes:  Synthesis of the AB Ring System of Norzoanthamine by Williams, David R, Brugel, Todd A

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Oncologic outcomes, prognostic factor analysis and therapeutic algorithm evaluation of head and neck mucosal melanomas in France by Moya-Plana, A., Aupérin, A., Obongo, R., Baglin, A., Baujat, B., Saroul, N., Casiraghi, O., Vergez, S., Janot, F., Thariat, J., Vérillaud, B., de Gabory, L., Albert, S., Andry, G., Badet, J.-M., Badoual, C., Baglin, A.C., Barry, B., Baujat, B., Bensadoun, R.J., Bertolus, C., Bessède, J.-P., Blanchard, D., Borel, C., Breheret, R., Breton, P., Brugel, L., Cassagnau, E., Castillo, L., Ceruse, P., Chabolle, F., Chevalier, D., Chobaut, J.C., Choussy, O., Cosmidis, A., Costes, V., Darrouzet, V., Demez, P., Dessi, P., Devauchelle, B., Digue, L., Dolivet, G., Dubrulle, F., Duflo, S., Faivre, S., Fakhry, N., Ferron, C., Floret, F., Garrel, R., Geoffrois, L., Giovanni, A., Girod, A., Guerrier, B., Hans, S., Herman, P., Hofman, P., Housset, M., Jankowski, R., Jegoux, F., Juliéron, M., Kaminsky, M.-C., Kolb, F., Lacau St Guily, J., Laccoureye, L., Lallemant, B., Lang, P., Lavieille, J.-P., Lefevre, M., Leroy, X., Malard, O., Mauvais, O., Merol, J.-C., Michel, J., Mom, T., Morinière, S., de Monès, E., Moulin, G., Moya-Plana, A., Noel, G., Poissonnet, G., Prades, J.-M., Reyt, E., Righini, C., Rolland, F., Sarroul, N., Schultz, P., Serrano, E., Sterkers, O., Strunski, V., Tassart, M., Testelin, S., Thariat, J., Timochenko, A., Uro Coste, E., Valette, G., Van den Abbeele, T., Veillon, F., Vergez, S., Vérillaud, B., Wassef, M.

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Beneath HMGA2 alterations in pleomorphic adenomas: Pathological, immunohistochemical, and molecular insights by Lépine, Charles, Descotes, Françoise, Pissaloux, Daniel, Tirode, Franck, Lopez, Jonathan, Philouze, Pierre, Fieux, Maxime, Wassef, Michel, Castain, Claire, Uro-Coste, Emmanuelle, Babin, E., Bach, C., Badoual, C., Baglin, A.C., Bastit, V., Baujat, B., Bensadoun, R.J., Benzerdjeb, N., Bernadach, M., Bozec, L., Grayeli, A.Bozorg, Camby, S., Cassagnau, E., Castelli, J., Chevalier, D., Clatot, F., Constans, J.M., Coste, A., Coste, F., Costes, V., Cottier, J.P., Cristofari, J.P., Cupissol, D., Delgrande, J., Delord, J.P., Digue, L., Dolivet, G., Doré, M., Dufour, X., Eker, E., Even, C., Fabiano, E., Faivre, S., Fakhry, N., Frandon, J., de Gabory, L., Garcier, M., Guihard, S., Halimi, C., Herman, P., Hourseau, M., Jankowski, R., Jeanne, C., Juliéron, M., Kreps, S., Laccoureye, L., Lae, M., Lagarde, F., Lagrange, A., Lamuraglia, M., Lapeyre, M., Cardon, A.Lasne, Lefevre, M., Lelonge, Y., Liem, X., Linassier, C., Maingon, P., Michel, J., Mineur, G., Mirghani, H., Modesto, A., Molinier-Blossier, S., Morinière, S., Moya-Plana, A., Musat, E., Nguyen, F., Obongo-Anga, F.R., Page, C., Pestre, J., Pons, C., J.-M.Prades, Queiros, C., Rambeau, A., Ramin, L., Siegfried, A., Righini, C.A., Saada, E., Salas, S., Simonaggio, A., Sterkers, O., Xu-Shan, S., Taouachi, R., Tassart, M., David, M. Timar, Coste, E. Uro, Valette, G., Varoquaux, A., Vauleon, E., Vulquin, N., Wassef, M.

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Mucoepidermoid carcinoma of salivary glands: A French Network of Rare Head and Neck Tumors (REFCOR) prospective study of 292 cases by Giorgi, Roch, Vergez, Sébastien, Le Taillandier de Gabory, Ludovic, Costes-Martineau, Valérie, Herman, Philippe, Mauvais, Olivier, Malard, Olivier, Garrel, Renaud, Barry, Béatrix, Bach, Christine, Chevalier, Dominique, Mouawad, Francois, Merol, Jean-Claude, Bastit, Vianney, Thariat, Juliette, Dufour, Xavier, Righini, Christian-Adrien, Moya-Plana, Antoine, Radulesco, Thomas, Michel, Justin, Baujat, Bertrand, Andry, G., Badet, J.-M., Badoual, C., Baglin, A.C., Banal, A., Baudin, E., Baujat, B., Bertolus, C., Bessède, J.-P., Blanchard, D., Bozorg-Grayeli, A., Breheret, R., Breton, P., Brugel, L., Calais, G., Casiraghi, O., Castillo, L., Ceruse, P., Chabolle, F., Choussy, O., Coste, A., Costes, V., Crampette, L., Darrouzet, V., Demez, P., Devauchelle, B., Dolivet, G., Dufour, X., Faivre, S., Fakhry, N., Ferron, C., Floret, F., Garrel, R., Geoffrois, L., Gilain, L., Giovanni, A., Girod, A., Hans, S., Hofman, P., Housset, M., Jankowski, R., Jegoux, F., Kaminsky, M.-C., Kolb, F., St Guily, J. Lacau, Laccoureye, L., Lallemant, B., Lang, P., Lartigau, E., Lavieille, J.-P., Lefevre, M., Malard, O., Mauvais, O., Merol, J.-C., Michel, J., Morinière, S., Moulin, G., Poissonnet, G., Prades, J.-M., Radulesco, T., de Raucourt, D., Reyt, E., Righini, C., Robin, Y. Marie, Rolland, F., Sarroul, N., Schultz, P., Sterkers, O., Strunski, V., Tassart, M., Testelin, S., Thariat, J., Timochenko, A., Toussaint, B., Van den Abbeele, T., Varoquaux, A., Veillon, F., Vergez, S., Wassef, M.

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Bicyclo((aryl)methyl)benzamides as inhibitors of GlyT1 by Varnes, Jeffrey G., Xiong, Hui, Forst, Janet M., Holmquist, Christopher R., Ernst, Glen E., Frietze, William, Dembofsky, Bruce, Andisik, Don W., Palmer, William E., Hinkley, Lindsay, Steelman, Gary B., Wilkins, Deidre E., Tian, Gaochao, Jonak, Gerald, Potts, William M., Wang, Xia, Brugel, Todd A., Alhambra, Cristóbal, Wood, Michael W., Veale, Chris A., Albert, Jeffrey S.

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Identification of short-acting κ-opioid receptor antagonists with anxiolytic-like activity by Peters, Matthew F., Zacco, Anna, Gordon, John, Maciag, Carla M., Litwin, Linda C., Thompson, Carolann, Schroeder, Patricia, Sygowski, Linda A., Piser, Timothy M., Brugel, Todd A.

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Impact of facial nerve resection in parotid cancer abutting the facial nerve without preoperative paralysis: A multicentric propensity score-based analysis by Chatelet, Florian, Chevret, Sylvie, Fakhry, Nicolas, Even, Caroline, Mouawad, François, Vergez, Sébastien, Schultz, Philippe, Baudouin, Robin, Atallah, Sarah, Haroun, Fabienne, Paasche, Agnès, Herman, Philippe, Aubry, K., Babin, E., Bach, C., Badoual, C., Baglin, A.C., Bastit, V., Baujat, B., Bensadoun, R.J., Benzerdjeb, N., Bernadach, M., Bodmer, D., Boisselier, P., Brenet, E., Brugel, L., Calugaru, V., Cassagnau, E., Castelli, J., Ceruse, P., Chabolle, F., Chevalier, D., Choussy, O., Colin, E., Cottier, J.P., Coutte, A., Devauchelle, B., Dupin, C., Espitalier, F., Evrard, C., Fabiano, E., Fakhry, N., Frandon, J., Garrel, R., Gilain, L., Guillerm, S., Houessinon, A., Hourseau, M., Jegoux, F., Juliéron, M., de Kermadec, H., Laadhari, M., Laccoureye, L., Lae, M., Lagarde, F., Lagrange, A., Lapeyre, M., Lasne Cardon, A., Le Tourneau, C., Lefebvre, G., Lelonge, Y., Leroy, X., Maingon, P., Malard, O., Marie, J.-P., Maurina, T., Mineur, G., Mirafzal, S., Mirghani, H., Mouawad, F., Nguyen, F., Obongo-Anga, F.R., Onea, M., Page, C., Pestre, J., Pham Dang, N., Prades, J.-M., Prevost, A., Rahmani, A., Rambeau, A., Ramin, L., Renard, S., Righini, C.A., Rolland, F., Sacino, F., Saroul, N., Schultz, P., Strunski, V., Sudaka, A., Xu-Shan, S., Testelin, S., Timar David, M., Timochenko, A., Villa, J., Villepelet, A., Volondat, M., Vulquin, N., Wagner, I., Webert, L., Wong, S.

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Identification of protease-sensitive but not misfolding PNLIP variants in familial and hereditary pancreatitis by Masson, Emmanuelle, Berthet, Stéphanie, Le Gac, Gerald, Le Rhun, Marc, Ka, Chandran, Autret, Sandrine, Gourlaouen, Isabelle, Abrantes, Amandine, Aguilera Munoz, Lina, Albouys, Jérémie, Alric, Laurent, Amiot, Xavier, Archambeaud, Isabelle, Bastide, Laetitia, Baudon, Julien, Bellaiche, Guy, Bertrand, Valérie, Bideau, Karine, Billiemaz, Kareen, Billioud, Claire, Bonnefoy, Sabine, Borderon, Corinne, Bournet, Barbara, Breton, Estelle, Brugel, Mathias, Cadiot, Guillaume, Camus, Marine, Chamouard, Patrick, Chaput, Ulriikka, Cholet, Franck, Ciocan, Dragos Marius, Coffin, Benoit, Coimet-Berger, Laura, Daboussi, Oussama, Dalstein, Véronique, De Mestier, Louis, Degand, Thibault, Denis, Bernard, Desgrippes, Romain, Drouet d'Aubigny, Augustin, Enaud, Raphaël, Fabre, Alexandre, Gelsi, Eve, Gentilcore, Elena, Gincul, Rodica, Ginglinger-Favre, Emmanuelle, Gomercic, Cécile, Gondran, Hannah, Grandval, Philippe, Grasset, Denis, Grimbert, Sylvie, Heissat, Sophie, Hentic, Olivia, Herber-Mayne, Anne, Jacques, Jérémie, Jais, Bénédicte, Kaassis, Mehdi, Koch, Stéphane, Lacaze, Elodie, Lamireau, Thierry, Le Guillou, Xavier, Leblanc, Sarah, Levy, Philippe, Lievre, Astrid, Lorenzo, Diane, Marcel, Kévin, Matias, Clément, Mauillon, Jacques, Morgant, Stéphanie, Moussata, Driffa, Muller, Nelly, Napoleon, Bertrand, Olivier, Anne, Pagenault, Maël, Pelletier, Anne-laure, Pennec, Olivier, Pioche, Mathieu, Prost, Bénédicte, Queneherve, Lucille, Rebours, Vinciane, Rekik, Samia, Riachi, Ghassan, Rohmer, Barbara, Roquelaure, Bertrand, Rosa Hezode, Isabelle, Rostain, Florian, Saurin, Jean-Christophe, Servais, Laure, Stan-Iuga, Roxana, Subtil, Clément, Texier, Charles, Tougeron, David, Tsakiris, Laurent, Vuitton, Lucine, Wallenhorst, Timothée, Wangerme, Marc, Zerbib, Frank, Cooper, David N., Férec, Claude, Chen, Jian-Min

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Nineteen polymorphic microsatellite markers from two African Vanilla species: across-species transferability and diversity in a wild population of V. humblotii from Mayotte by Gigant, R., Brugel, A., De Bruyn, A., Risterucci, A. M., Guiot, V., Viscardi, G., Humeau, L., Grisoni, M., Besse, P.

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N-Functionalization of Poly(ethylene glycol)-Linked Mono- and Bis-dioxocyclams as Potential Ligands for Gd3 by Brugel, Todd A, Hegedus, L. S

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The development of 2-benzimidazole substituted pyrimidine based inhibitors of lymphocyte specific kinase (Lck) by Sabat, Mark, VanRens, John C., Laufersweiler, Matthew J., Brugel, Todd A., Maier, Jennifer, Golebiowski, Adam, De, Biswanath, Easwaran, Vijayasurian, Hsieh, Lily C., Walter, Richard L., Mekel, Marlene J., Evdokimov, Artem, Janusz, Michael J.

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The development of monocyclic pyrazolone based cytokine synthesis inhibitors by Golebiowski, Adam, Townes, Jennifer A., Laufersweiler, Matthew J., Brugel, Todd A., Clark, Michael P., Clark, Cynthia M., Djung, Jane F., Laughlin, Steven K., Sabat, Mark P., Bookland, Roger G., VanRens, John C., De, Biswanath, Hsieh, Lily C., Janusz, Michael J., Walter, Richard L., Webster, Mark E., Mekel, Marlene J.

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Understanding and overcoming the pitfalls in the diagnosis of pleomorphic and carcinoma ex-pleomorphic adenoma of salivary glands by Alsugair, Ziyad, Lépine, Charles, Fieux, Maxime, Descotes, Françoise, Pissaloux, Daniel, Lopez, Jonathan, Russel, Juliette, Céruse, Philippe, Philouze, Pierre, Uro-Coste, Emmanuelle, Siegfried, Aurore, Costes-Martineau, Valérie, Champagnac, Anne, Benzerdjeb, Nazim

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4-Aryl piperazine and piperidine amides as novel mGluR5 positive allosteric modulators by Xiong, Hui, Brugel, Todd A., Balestra, Michael, Brown, Dean G., Brush, Kelly A., Hightower, Caprice, Hinkley, Lindsay, Hoesch, Valerie, Kang, James, Koether, Gerard M., McCauley, John P., McLaren, Francis M., Panko, Laura M., Simpson, Thomas R., Smith, Reed W., Woods, James M., Brockel, Becky, Chhajlani, Vijay, Gadient, Reto A., Spear, Nathan, Sygowski, Linda A., Zhang, Minli, Arora, Jalaj, Breysse, Nathalie, Wilson, Julie M., Isaac, Methvin, Slassi, Abdelmalik, King, Megan M.

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From source terrains of the Eastern Alps to the Molasse Basin: Detrital record of non-steady-state exhumation by Kuhlemann, J., Dunkl, I., Brügel, A., Spiegel, C., Frisch, W.

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SAR development of a series of 8-azabicyclo[3.2.1]octan-3-yloxy-benzamides as kappa opioid receptor antagonists. Part 2 by Brugel, Todd A., Smith, Reed W., Balestra, Michael, Becker, Christopher, Daniels, Thalia, Koether, Gerard M., Throner, Scott R., Panko, Laura M., Brown, Dean G., Liu, Ruifeng, Gordon, John, Peters, Matthew F.

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Development of new pyrrolopyrimidine-based inhibitors of Janus kinase 3 (JAK3) by Clark, Michael P., George, Kelly M., Bookland, Roger G., Chen, Jack, Laughlin, Steven K., Thakur, Kumar D., Lee, Wenlin, Davis, Jan R., Cabrera, Ed J., Brugel, Todd A., VanRens, John C., Laufersweiler, Matthew J., Maier, Jennifer A., Sabat, Mark P., Golebiowski, Adam, Easwaran, Vijay, Webster, Mark E., De, Biswanath, Zhang, George

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Discovery of 8-azabicyclo[3.2.1]octan-3-yloxy-benzamides as selective antagonists of the kappa opioid receptor. Part 1 by Brugel, Todd A., Smith, Reed W., Balestra, Michael, Becker, Christopher, Daniels, Thalia, Hoerter, Tiffany N., Koether, Gerard M., Throner, Scott R., Panko, Laura M., Folmer, James J., Cacciola, Joseph, Hunter, Angela M., Liu, Ruifeng, Edwards, Philip D., Brown, Dean G., Gordon, John, Ledonne, Norman C., Pietras, Mark, Schroeder, Patricia, Sygowski, Linda A., Hirata, Lee T., Zacco, Anna, Peters, Matthew F.

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