Identification of a series of 4-[3-(quinolin-2-yl)-1,2,4-oxadiazol-5-yl]piperazinyl ureas as potent smoothened antagonist hedgehog pathway inhibitors by Ontoria, Jesus M., Bufi, Laura Llauger, Torrisi, Caterina, Bresciani, Alberto, Giomini, Claudia, Rowley, Michael, Serafini, Sergio, Bin, Hu, Hao, Wu, Steinkühler, Christian, Jones, Philip

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Identification and SAR of novel pyrrolo[1,2- a]pyrazin-1(2 H)-one derivatives as inhibitors of poly(ADP-ribose) polymerase-1 (PARP-1) by Pescatore, Giovanna, Branca, Danila, Fiore, Fabrizio, Kinzel, Olaf, Bufi, Laura Llauger, Muraglia, Ester, Orvieto, Federica, Rowley, Michael, Toniatti, Carlo, Torrisi, Caterina, Jones, Philip

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N-(2-alkylaminoethyl)-4-(1,2,4-oxadiazol-5-yl)piperazine-1-carboxamides as highly potent smoothened antagonists by Muraglia, Ester, Ontoria, Jesus M., Branca, Danila, Dessole, Gabriella, Bresciani, Alberto, Fonsi, Massimiliano, Giuliano, Claudio, Llauger Bufi, Laura, Monteagudo, Edith, Palumbi, Maria Cecilia, Torrisi, Caterina, Rowley, Michael, Steinkühler, Christian, Jones, Philip

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Development of substituted 6-[4-fluoro-3-(piperazin-1-ylcarbonyl)benzyl]-4,5-dimethylpyridazin-3(2 H)-ones as potent poly(ADP–ribose) polymerase-1 (PARP-1) inhibitors active in BRC... by Ferrigno, Federica, Branca, Danila, Kinzel, Olaf, Lillini, Samuele, Llauger Bufi, Laura, Monteagudo, Edith, Muraglia, Ester, Rowley, Michael, Schultz-Fademrecht, Carsten, Toniatti, Carlo, Torrisi, Caterina, Jones, Philip

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Synthesis of novel fluorescent probes for the molecular chaperone Hsp90 by Llauger-Bufi, Laura, Felts, Sara J, Huezo, Henri, Rosen, Neal, Chiosis, Gabriela

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Discovery of a Potent Class I Selective Ketone Histone Deacetylase Inhibitor with Antitumor Activity in Vivo and Optimized Pharmacokinetic Properties by Kinzel, Olaf, Llauger-Bufi, Laura, Pescatore, Giovanna, Rowley, Michael, Schultz-Fademrecht, Carsten, Monteagudo, Edith, Fonsi, Massimiliano, Gonzalez Paz, Odalys, Fiore, Fabrizio, Steinkühler, Christian, Jones, Philip

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N-(2-alkylaminoethyl)-4-(1,2,4-oxadiazol-5-yl)piperazine-1-carboxa mide s as highly potent smoothened antagonists by Muraglia, Ester, Ontoria, Jesus M, Branca, Danila, Dessole, Gabriella, Bresciani, Alberto, Fonsi, Massimiliano, Giuliano, Claudio, Bufi, Laura Llauger, Monteagudo, Edith, Palumbi, Maria Cecilia, Torrisi, Caterina, Rowley, Michael, Steinkuehler, Christian, Jones, Philip

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Development of substituted 6-[4-fluoro-3-(piperazin-1-ylcarbonyl)benzyl]-4,5-dimethylpyridazi n -3(2H)-ones as potent poly(ADP-ribose) polymerase-1 (PARP-1) inhibitors active in BR... by Ferrigno, Federica, Branca, Danila, Kinzel, Olaf, Lillini, Samuele, Bufi, Laura Llauger, Monteagudo, Edith, Muraglia, Ester, Rowley, Michael, Schultz-Fademrecht, Carsten, Toniatti, Carlo, Torrisi, Caterina, Jones, Philip

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