Discovery of heterocyclic ureas as a new class of raf kinase inhibitors: identification of a second generation lead by a combinatorial chemistry approach by Smith, Roger A, Barbosa, James, Blum, Cheri L, Bobko, Mark A, Caringal, Yolanda V, Dally, Robert, Johnson, Jeffrey S, Katz, Michael E, Kennure, Nancy, Kingery-Wood, Jill, Lee, Wendy, Lowinger, Timothy B, Lyons, John, Marsh, Vivienne, Rogers, Daniel H, Swartz, Stephen, Walling, Tracy, Wild, Hanno

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Discovery of (( S )-5-(Methoxymethyl)-7-(1-methyl-1 H -indol-2-yl)-2-(trifluoromethyl)-4,7-dihydropyrazolo[1,5- a ]pyrimidin-6-yl)(( S )-2-(3-methylisoxazol-5-yl)pyrrolidin-1-yl)me... by Finlay, Heather J., Lloyd, John, Vaccaro, Wayne, Kover, Alexander, Yan, Lin, Bhave, Gauri, Prol, Joseph, Huynh, Tram, Bhandaru, Rao, Caringal, Yolanda, DiMarco, John, Gan, Jinping, Harper, Tim, Huang, Christine, Conder, Mary Lee, Sun, Huabin, Levesque, Paul, Blanar, Michael, Atwal, Karnail, Wexler, Ruth

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Triazolo and imidazo dihydropyrazolopyrimidine potassium channel antagonists by Finlay, Heather J., Jiang, Ji, Caringal, Yolanda, Kover, Alexander, Conder, Mary Lee, Xing, Dezhi, Levesque, Paul, Harper, Timothy, Hsueh, Mei Mann, Atwal, Karnail, Blanar, Michael, Wexler, Ruth, Lloyd, John

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Correction to Discovery of (( S )-5-(Methoxymethyl)-7-(1-methyl-1 H -indol-2-yl)-2-(trifluoromethyl)-4,7-dihydropyrazolo[1,5- a ]pyrimidin-6-yl)(( S )-2-(3-methylisoxazol-5-yl)pyrr... by Finlay, Heather J., Lloyd, John, Vaccaro, Wayne, Kover, Alexander, Yan, Lin, Bhave, Gauri, Prol, Joseph, Huynh, Tram, Bhandaru, Rao, Caringal, Yolanda, DiMarco, John, Gan, Jinping, Harper, Tim, Huang, Christine, Conder, Mary Lee, Sun, Huabin, Levesque, Paul, Blanar, Michael, Atwal, Karnail, Wexler, Ruth

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A new route to benzo[a]naphthacene-8,13-diones: synthesis and revision of the structure proposed for G2N by Hauser, Frank M, Caringal, Yolanda

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Omega-carboxypyridyl substituted ureas as Raf kinase inhibitors: SAR of the amide substituent by Khire, Uday R., Bankston, Donald, Barbosa, James, Brittelli, David R., Caringal, Yolanda, Carlson, Robert, Dumas, Jacques, Gane, Todd, Heald, Sarah L., Hibner, Barbara, Johnson, Jeffrey S., Katz, Michael E., Kennure, Nancy, Kingery-Wood, Jill, Lee, Wendy, Liu, Xiao-Gao, Lowinger, Timothy B., McAlexander, Ian, Monahan, Mary-Katherine, Natero, Reina, Renick, Joel, Riedl, Bernd, Rong, Hong, Sibley, Robert N., Smith, Roger A., Wolanin, Donald

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Thyroid receptor ligands. Part 8: Thyromimetics derived from N-acylated-α-amino acid derivatives displaying modulated pharmacological selectivity compared with KB-141 by Garg, Neeraj, Li, Yi-Lin, Garcia Collazo, Ana Maria, Litten, Chris, Ryono, Denis E., Zhang, Minsheng, Caringal, Yolanda, Brigance, Robert P., Meng, Wei, Washburn, William N., Agback, Peter, Mellström, Karin, Rehnmark, Stefan, Rahimi-Ghadim, Mahmoud, Norin, Thomas, Grynfarb, Marlena, Sandberg, Johnny, Grover, Gary, Malm, Johan

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p38 Kinase inhibitors for the treatment of arthritis and osteoporosis: thienyl, furyl, and pyrrolyl ureas by Redman, Anikó M, Johnson, Jeffrey S, Dally, Robert, Swartz, Steve, Wild, Hanno, Paulsen, Holger, Caringal, Yolanda, Gunn, David, Renick, Joel, Osterhout, Martin, Kingery-Wood, Jill, Smith, Roger A, Lee, Wendy, Dumas, Jacques, Wilhelm, Scott M, Housley, Timothy J, Bhargava, Ajay, Ranges, Gerald E, Shrikhande, Alka, Young, Deborah, Bombara, Michael, Scott, William J

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Discovery of ((S)-5-(methoxymethyl)-7-(1-methyl-1H-indol-2-yl)-2-(trifluoromethyl)-4,7-dihydropyrazolo[1,5-a]pyrimidin-6-yl)((S)-2-(3-methylisoxazol-5-yl)pyrrolidin-1-yl)methanone... by Finlay, Heather J, Lloyd, John, Vaccaro, Wayne, Kover, Alexander, Yan, Lin, Bhave, Gauri, Prol, Joseph, Huynh, Tram, Bhandaru, Rao, Caringal, Yolanda, DiMarco, John, Gan, Jinping, Harper, Tim, Huang, Christine, Conder, Mary Lee, Sun, Huabin, Levesque, Paul, Blanar, Michael, Atwal, Karnail, Wexler, Ruth

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Synthesis and pharmacological characterization of a potent, orally active p38 kinase inhibitor by Dumas, Jacques, Hatoum-Mokdad, Holia, Sibley, Robert N, Smith, Roger A, Scott, William J, Khire, Uday, Lee, Wendy, Wood, Jill, Wolanin, Donald, Cooley, Jeffrey, Bankston, Donald, Redman, Aniko M, Schoenleber, Robert, Caringal, Yolanda, Gunn, David, Romero, Romulo, Osterhout, Martin, Paulsen, Holger, Housley, Timothy J, Wilhelm, Scott M, Pirro, John, Chien, Du-Shieng, Ranges, Gerald E, Shrikhande, Alka, Muzsi, Andrew, Bortolon, Elizabeth, Wakefield, Jean, Gianpaolo Ostravage, Cynthia, Bhargava, Ajay, Chau, Thuy

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Correction to Discovery of ((S)‑5-(Methoxymethyl)-7-(1-methyl‑1H‑indol-2-yl)-2-(trifluoromethyl)-4,7-dihydropyrazolo[1,5‑a]pyrimidin-6-yl)((S)‑2-(3-methylisoxazol-5-yl)pyrrolidin-1... by Finlay, Heather J, Lloyd, John, Vaccaro, Wayne, Kover, Alexander, Yan, Lin, Bhave, Gauri, Prol, Joseph, Huynh, Tram, Bhandaru, Rao, Caringal, Yolanda, DiMarco, John, Gan, Jinping, Harper, Tim, Huang, Christine, Conder, Mary Lee, Sun, Huabin, Levesque, Paul, Blanar, Michael, Atwal, Karnail, Wexler, Ruth

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Omega-carboxypyridyl substituted ureas as Raf kinase inhibitors by Khire, Uday R., Bankston, Donald, Barbosa, James, Brittelli, David R., Caringal, Yolanda, Carlson, Robert, Dumas, Jacques, Gane, Todd, Heald, Sarah L., Hibner, Barbara, Johnson, Jeffrey S., Katz, Michael E., Kennure, Nancy, Kingery-Wood, Jill, Lee, Wendy, Liu, Xiao-Gao, Lowinger, Timothy B., McAlexander, Ian, Monahan, Mary-Katherine, Natero, Reina, Renick, Joel, Riedl, Bernd, Rong, Hong, Sibley, Robert N., Smith, Roger A., Wolanin, Donald

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Discovery of ((S)-5-(Methoxymethyl)-7-(1-methyl-1H-indol-2-yl)-2-(trifluoromethyl)-4,7-dihydropyrazolo[1,5-a]pyrimidin-6-yl)((S)-2-(3-methylisoxazol-5-yl)pyrrolidin-1-yl)methanone... by Finlay, Heather J, Lloyd, John, Vaccaro, Wayne, Kover, Alexander, Yan, Lin, Bhave, Gauri, Prol, Joseph, Huynh, Tram, Bhandaru, Rao, Caringal, Yolanda, DiMarco, John, Gan, Jinping, Harper, Tim, Huang, Christine, Conder, Mary Lee, Sun, Huabin, Levesque, Paul, Blanar, Michael, Atwal, Karnail, Wexler, Ruth

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