Azepino-indazoles as calcitonin gene-related peptide (CGRP) receptor antagonists by Mercer, Stephen E., Chaturvedula, Prasad V., Conway, Charles M., Cook, Deborah A., Davis, Carl D., Pin, Sokhom S., Macci, Robert, Schartman, Richard, Signor, Laura J., Widmann, Kimberly A., Whiterock, Valerie J., Chen, Ping, Xu, Cen, Herbst, John J., Kostich, Walter A., Thalody, George, Macor, John E., Dubowchik, Gene M.

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Discovery of (R)-N-(3-(7-methyl-1H-indazol-5-yl)-1-(4-(1-methylpiperidin-4-yl)-1-oxopropan-2-yl)-4-(2-oxo-1,2-dihydroquinolin-3-yl)piperidine-1-carboxamide (BMS-742413): A potent h... by Chaturvedula, Prasad V., Mercer, Stephen E., Pin, Sokhom S., Thalody, George, Xu, Cen, Conway, Charlie M., Keavy, Deborah, Signor, Laura, Cantor, Glenn H., Mathias, Neil, Moench, Paul, Denton, Rex, Macci, Robert, Schartman, Richard, Whiterock, Valerie, Davis, Carl, Macor, John E., Dubowchik, Gene M.

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Synthesis and SAR of calcitonin gene-related peptide (CGRP) antagonists containing substituted aryl-piperazines and piperidines by Civiello, Rita L., Han, Xiaojun, Beno, Brett R., Chaturvedula, Prasad V., Herbst, John J., Xu, Cen, Conway, Charles M., Macor, John E., Dubowchik, Gene M.

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Design and synthesis of potent antagonists containing rigid spirocyclic privileged structures for the CGRP receptor by Chaturvedula, Prasad V., Pin, Sokhom, Tholady, George, Conway, Charlie M., Macor, John E., Dubowchik, Gene M.

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Discovery of (R)-4-(8-Fluoro-2-oxo-1,2-dihydroquinazolin-3(4H)-yl)-N-(3-(7-methyl-1H-indazol-5-yl)-1-oxo-1-(4-(piperidin-1-yl)piperidin-1-yl)propan-2-yl)piperidine-1-carboxamide (B... by Degnan, Andrew P, Chaturvedula, Prasad V, Conway, Charles M, Cook, Deborah A, Davis, Carl D, Denton, Rex, Han, Xiaojun, Macci, Robert, Mathias, Neil R, Moench, Paul, Pin, Sokhom S, Ren, Shelly X, Schartman, Richard, Signor, Laura J, Thalody, George, Widmann, Kimberly A, Xu, Cen, Macor, John E, Dubowchik, Gene M

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Enantioselective synthesis of constrained phenylalanine analogues by Chaturvedula, Prasad V., Mercer, Stephen E., Guernon, Leatte, Macor, John E., Dubowchik, Gene M.

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Catalytic Asymmetric Syntheses of α-Amino and α-Hydroxyl Acid Derivatives by Han, Xiaojun, Jiang, Xiang-Jun, Civiello, Rita L, Degnan, Andrew P, Chaturvedula, Prasad V, Macor, John E, Dubowchik, Gene M

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The synthesis and SAR of calcitonin gene-related peptide (CGRP) receptor antagonists derived from tyrosine surrogates. Part 1 by Han, Xiaojun, Civiello, Rita L., Conway, Charles M., Cook, Deborah A., Davis, Carl D., Macci, Robert, Pin, Sokhom S., Ren, Shelly X., Schartman, Richard, Signor, Laura J., Thalody, George, Widmann, Kimberly A., Xu, Cen, Chaturvedula, Prasad V., Macor, John E., Dubowchik, Gene M.

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Catalytic Asymmetric Syntheses of Tyrosine Surrogates by Han, Xiaojun, Civiello, Rita L, Fang, Haiquang, Wu, Dedong, Gao, Qi, Chaturvedula, Prasad V, Macor, John E, Dubowchik, Gene M

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Discovery of (R)-4-(8-Fluoro-2-oxo-1,2-dihydroquinazolin-3(4H)-yl)-N-3-(7-methyl-1H-indazol-5-yl)-1-oxo-1-(4-(piperidm-1-yl)piperidin-1-yl)propan-2-ylpiperidine-1-carboxamide (BMS-... by DEGNAN, Andrew P, CHATURVEDULA, Prasad V, PIN, Sokhom S, REN, Shelly X, SCHARTMAN, Richard, SIGNOR, Laura J, THALODY, George, WIDMANN, Kimberly A, CEN XU, MACOR, John E, DUBOWCHIK, Gene M, CONWAY, Charles M, COOK, Deborah A, DAVIS, Carl D, DENTON, Rex, XIAOJUN HAN, MACCI, Robert, MATHIAS, Neil R, MOENCH, Paul

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P2-122 Detection of Nβ peptide and quantitation of its inhibition by γ-secretase inhibitors by Toyn, Jeremy, Fiedler, Tracey, Guss, Valerie L., Polson, Craig, Meredith, Jere E., Seiffert, Dietmar, Olson, Richard E., Chaturvedula, Prasad V., Smith, David W.

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