Crystal Structures of Human Factor Xa Complexed with Potent Inhibitors by Maignan, Sébastien, Guilloteau, Jean-Pierre, Pouzieux, Stéphanie, Choi-Sledeski, Yong Mi, Becker, Michael R, Klein, Scott I, Ewing, William R, Pauls, Henry W, Spada, Alfred P, Mikol, Vincent

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Aminoisoquinolines: Design and synthesis of an orally active benzamidine isostere for the inhibition of factor XA by Choi-Sledeski, Y.M., Becker, M.R., Green, D.M., Davis, R., Ewing, W.R., Mason, H.J., Ly, C., Spada, A., Liang, G., Cheney, D., Barton, J., Chu, V., Brown, K., Colussi, D., Bentley, R., Leadley, R., Dunwiddie, C., Pauls, H.W.

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Design and Structure−Activity Relationships of Potent and Selective Inhibitors of Blood Coagulation Factor Xa by Ewing, William R, Becker, Michael R, Manetta, Vincent E, Davis, Roderick S, Pauls, Henry W, Mason, Helen, Choi-Sledeski, Yong Mi, Green, Daniel, Cha, Don, Spada, Alfred P, Cheney, Daniel L, Mason, Jonathan S, Maignan, Sebastien, Guilloteau, Jean-Pierre, Brown, Karen, Colussi, Dennis, Bentley, Ross, Bostwick, Jeff, Kasiewski, Charles J, Morgan, Suzanne R, Leadley, Robert J, Dunwiddie, Christopher T, Perrone, Mark H, Chu, Valeria

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Synthesis, SAR and in vivo activity of novel thienopyridine sulfonamide pyrrolidinones as factor Xa inhibitors by Becker, Michael R., Ewing, William R., Davis, Roderick S., Pauls, Henry W., Ly, Cuong, Li, Aiwen, Mason, Helen J., Choi-Sledeski, Yong Mi, Spada, Alfred P., Chu, Valeria, Brown, Karen D., Colussi, Dennis J., Leadley, Robert J., Bentley, Ross, Bostwick, Jeff, Kasiewski, Charles, Morgan, Suzanne

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Solid-phase parallel synthesis of azarene pyrrolidinones as factor Xa inhibitors by Gong, Y, Becker, M, Choi-Sledeski, Y M, Davis, R S, Salvino, J M, Chu, V, Brown, K D, Pauls, H W

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Synthesis of Functionalized Aromatic Oligomers from a Versatile Diphenylmethane Template by Bruno, J. G, Chang, M. N, Choi-Sledeski, Y. M, Green, D. M, McGarry, D. G, Regan, J. R, Volz, F. A

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Discovery of an Orally Efficacious Inhibitor of Coagulation Factor Xa Which Incorporates a Neutral P 1 Ligand by Choi-Sledeski, Yong Mi, Kearney, Robert, Poli, Gregory, Pauls, Henry, Gardner, Charles, Gong, Yong, Becker, Michael, Davis, Roderick, Spada, Alfred, Liang, Guyan, Chu, Valeria, Brown, Karen, Collussi, Dennis, Leadley, Robert, Rebello, Sam, Moxey, Phillip, Morgan, Suzanne, Bentley, Ross, Kasiewski, Charles, Maignan, Sebastien, Guilloteau, Jean-Pierre, Mikol, Vincent

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Sulfonamidopyrrolidinone Factor Xa Inhibitors:  Potency and Selectivity Enhancements via P-1 and P-4 Optimization by Choi-Sledeski, Yong Mi, McGarry, Daniel G, Green, Daniel M, Mason, Helen J, Becker, Michael R, Davis, Roderick S, Ewing, William R, Dankulich, William P, Manetta, Vincent E, Morris, Robert L, Spada, Alfred P, Cheney, Daniel L, Brown, Karen D, Colussi, Dennis J, Chu, Valeria, Heran, Christopher L, Morgan, Suzanne R, Bentley, Ross G, Leadley, Robert J, Maignan, Sebastien, Guilloteau, Jean-Pierre, Dunwiddie, Christopher T, Pauls, Henry W

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Molecular Structures of Human Factor Xa Complexed with Ketopiperazine Inhibitors:  Preference for a Neutral Group in the S1 Pocket by Maignan, Sébastien, Guilloteau, Jean-Pierre, Choi-Sledeski, Yong Mi, Becker, Michael R, Ewing, William R, Pauls, Henry W, Spada, Alfred P, Mikol, Vincent

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