Discovery of Brivanib Alaninate ((S)-((R)-1-(4-(4-Fluoro-2-methyl-1H-indol-5-yloxy)-5-methylpyrrolo[2,1-f][1,2,4]triazin-6-yloxy)propan-2-yl)2-aminopropanoate), A Novel Prodrug of... by Cai, Zhen-wei, Zhang, Yongzheng, Borzilleri, Robert M, Qian, Ligang, Barbosa, Stephanie, Wei, Donna, Zheng, Xiaoping, Wu, Lawrence, Fan, Junying, Shi, Zhongping, Wautlet, Barri S, Mortillo, Steve, Jeyaseelan, Robert, Kukral, Daniel W, Kamath, Amrita, Marathe, Punit, D’Arienzo, Celia, Derbin, George, Barrish, Joel C, Robl, Jeffrey A, Hunt, John T, Lombardo, Louis J, Fargnoli, Joseph, Bhide, Rajeev S

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Role of Self-Association and Supersaturation in Oral Absorption of a Poorly Soluble Weakly Basic Drug by Narang, Ajit S., Badawy, Sherif, Ye, Qingmei, Patel, Dhaval, Vincent, Maria, Raghavan, Krishnaswamy, Huang, Yande, Yamniuk, Aaron, Vig, Balvinder, Crison, John, Derbin, George, Xu, Yan, Ramirez, Antonio, Galella, Michael, Rinaldi, Frank A.

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Discovery and Preclinical Studies of (R)-1-(4-(4-Fluoro-2-methyl-1H-indol-5-yloxy)-5- methylpyrrolo[2,1-f][1,2,4]triazin-6-yloxy)propan- 2-ol (BMS-540215), an In Vivo Active Potent... by Bhide, Rajeev S, Cai, Zhen-Wei, Zhang, Yong-Zheng, Qian, Ligang, Wei, Donna, Barbosa, Stephanie, Lombardo, Louis J, Borzilleri, Robert M, Zheng, Xiaoping, Wu, Laurence I, Barrish, Joel C, Kim, Soong-Hoon, Leavitt, Kenneth, Mathur, Arvind, Leith, Leslie, Chao, Sam, Wautlet, Barri, Mortillo, Steven, Jeyaseelan, Robert, Kukral, Daniel, Hunt, John T, Kamath, Amrita, Fura, Aberra, Vyas, Viral, Marathe, Punit, D'Arienzo, Celia, Derbin, George, Fargnoli, Joseph

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Food Increased the Bioavailability of BMS-690514, an Orally Active EGFR/HER2/VEGF Receptor Kinase Inhibitor, in Healthy Subjects by Vakkalagadda, Blisse, Park, Jong-Soon, Ahlers, Christoph M., Dorizio, Stephanie, Has, Teresa, Roongta, Vikram, Heller, Kevin N., Derbin, George M., Zhang, Steven

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Discovery and Evaluation of N-Cyclopropyl- 2,4-difluoro-5-((2-(pyridin-2-ylamino)thiazol-5- ylmethyl)amino)benzamide (BMS-605541), a Selective and Orally Efficacious Inhibitor of V... by Borzilleri, Robert M, Bhide, Rajeev S, Barrish, Joel C, D'Arienzo, Celia J, Derbin, George M, Fargnoli, Joseph, Hunt, John T, Jeyaseelan, Robert, Kamath, Amrita, Kukral, Daniel W, Marathe, Punit, Mortillo, Steve, Qian, Ligang, Tokarski, John S, Wautlet, Barri S, Zheng, Xiaoping, Lombardo, Louis J

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Development of a Canine Model to Enable the Preclinical Assessment of Ph-dependent Absorption of Test Compounds by Fancher, R. Marcus, Zhang, Hongjian, Sleczka, Bogdan, Derbin, George, Rockar, Richard, Marathe, Punit

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Acid-Catalyzed Hydrolysis of BMS-582664: Degradation Product Identification and Mechanism Elucidation by Zhao, Fang, Derbin, George, Miller, Scott, Badawy, Sherif, Hussain, Munir

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Discovery and preclinical studies of 5-isopropyl-6-(5-methyl-1,3,4-oxadiazol-2-yl)- N-(2-methyl-1 H-pyrrolo[2,3- b]pyridin-5-yl)pyrrolo[2,1- f][1,2,4]triazin-4-amine (BMS-645737),... by Ruel, Réjean, Thibeault, Carl, L’Heureux, Alexandre, Martel, Alain, Cai, Zhen-Wei, Wei, Donna, Qian, Ligang, Barrish, Joel C., Mathur, Arvind, D’Arienzo, Celia, Hunt, John T., Kamath, Amrita, Marathe, Punit, Zhang, Yueping, Derbin, George, Wautlet, Barri, Mortillo, Steven, Jeyaseelan, Robert, Henley, Benjamin, Tejwani, Ravindra, Bhide, Rajeev S., Trainor, George L., Fargnoli, Joseph, Lombardo, Louis J.

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Discovery of Brivanib Alaninate (S)-(R)-1-(4-(4-Fluoro-2-methyl-1H-indol-5-yloxy)-5-methylpyrrolo[2,1-f][1,2,4]triazin-6-yloxy)propan-2-yl2-aminopropanoate, A Novel Prodrug of Dual... by CAI, Zhen-Wei, YONGZHENG ZHANG, WAUTLET, Barri S, MORTILLO, Steve, JEYASEELAN, Robert, KUKRAL, Daniel W, KAMATH, Amrita, MARATHE, Punit, D'ARIENZO, Celia, DERBIN, George, BARRISH, Joel C, ROBL, Jeffrey A, BORZILLERI, Robert M, HUNT, John T, LOMBARDO, Louis J, FARGNOLI, Joseph, BHIDE, Rajeev S, LIGANG QIAN, BARBOSA, Stephanie, WEI, Donna, XIAOPING ZHENG, WU, Lawrence, JUNYING FAN, ZHONGPING SHI

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Discovery and evaluation of N-cyclopropyl-2,4-difluoro-5-(2-(pyridin-2-ylamino)thiazol-5-ylmethyl)aminobenzamide (BMS-605541), a selective and orally efficacious inhibitor of vascu... by BORZILLERI, Robert M, BHIDE, Rajeev S, MARATHE, Punit, MORTILLO, Steve, LIGANG QIAN, TOKARSKI, John S, WAUTLET, Barri S, XIAOPING ZHENG, LOMBARDO, Louis J, BARRISH, Joel C, D'ARIENZO, Celia J, DERBIN, George M, FARGNOLI, Joseph, HUNT, John T, JEYASEELAN, Robert, KAMATH, Amrita, KUKRAL, Daniel W

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Discovery and preclinical studies of (R)-1-(4-(4-fluoro-2-methyl- 1H-indol-5-yloxy)-5-methylpyrrolo[2,1-/][1,2,4]triazin-6-yloxy)propan2-ol (BMS-540215), an in vivo active potent V... by BHIDE, Rajeev S, CAI, Zhen-Wei, BARRISH, Joel C, KIM, Soong-Hoon, LEAVITT, Kenneth, MATHUR, Arvind, LEITH, Leslie, CHAO, Sam, WAUTLET, Barri, MORTILLO, Steven, JEYASEELAN, Robert, KUKRAL, Daniel, ZHANG, Yong-Zheng, HUNT, John T, KAMATH, Amrita, FURA, Aberra, VYAS, Viral, MARATHE, Punit, D'ARIENZO, Celia, DERBIN, George, FARGNOLI, Joseph, LIGANG QIAN, WEI, Donna, BARBOSA, Stephanie, LOMBARDO, Louis J, BORZILLERI, Robert M, XIAOPING ZHENG, WU, Laurence I

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