Discovery of JNJ-64264681: A Potent and Selective Covalent Inhibitor of Bruton’s Tyrosine Kinase by Tichenor, Mark S., Wiener, John J. M., Rao, Navin L., Bacani, Genesis M., Wei, Jianmei, Pooley Deckhut, Charlotte, Barbay, J. Kent, Kreutter, Kevin D., Chang, Leon, Clancy, Kathleen W., Murrey, Heather E., Wang, Weixue, Ahn, Kay, Huber, Michael, Rex, Elizabeth, Coe, Kevin J., Wu, Jiejun, Rui, Haopeng, Sepassi, Kia, Gaudiano, Marcello, Bekkers, Mariette, Cornelissen, Ivo, Packman, Kathryn, Seierstad, Mark, Xiouras, Christos, Bembenek, Scott D., Alexander, Richard, Milligan, Cynthia, Balasubramanian, Sriram, Lebsack, Alec D., Venable, Jennifer D., Philippar, Ulrike, Edwards, James P., Hirst, Gavin

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Discovery of a Potent and Selective Covalent Inhibitor of Bruton’s Tyrosine Kinase with Oral Anti-Inflammatory Activity by Tichenor, Mark S, Wiener, John J. M, Rao, Navin L, Pooley Deckhut, Charlotte, Barbay, J. Kent, Kreutter, Kevin D, Bacani, Genesis M, Wei, Jianmei, Chang, Leon, Murrey, Heather E, Wang, Weixue, Ahn, Kay, Huber, Michael, Rex, Elizabeth, Coe, Kevin J, Wu, JieJun, Seierstad, Mark, Bembenek, Scott D, Leonard, Kristi A, Lebsack, Alec D, Venable, Jennifer D, Edwards, James P

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Potent, nonsteroidal selective androgen receptor modulators (SARMs) based on 8H-[1,4 ]oxazino [2,3 -f] quinolin-8-ones by HIGUCHI, Robert I, THOMPSON, Anthony W, ADAM KALLEL, E, KARANEWSKY, Donald S, SCHRADER, William T, MARSCHKE, Keith B, LIN ZHI, CHEN, Jyun-Hung, CAFERRO, Thomas R, CUMMINGS, Marquis L, DECKHUT, Charlotte P, ADAMS, Mark E, TEGLEY, Christopher M, EDWARDS, James P, LOPEZ, Francisco J

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5 (Z) -Benzylidene -1,2 -dihydro -9 -hydroxy -10 -methoxy -2,2, 4 -trimethyl -5H-1 -aza -6 -oxa -chrysenes as non-steroidal glucocorticoid receptor modulators by ARDECKY, Robert J, HUDSON, Andrew R, LOPEZ, Francisco J, MARSCHKE, Keith B, MINER, Jeffrey N, KARANEWSKY, Donald S, NEGRO-VILAR, Andrés, LIN ZHI, PHILLIPS, Dean P, TYHONAS, John S, DECKHUT, Charlotte, LAU, Thomas L, YONGKAI LI, MARTINBOROUGH, Esther A, ROACH, Steven L, HIGUCHI, Robert I

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Potent, nonsteroidal selective androgen receptor modulators (SARMs) based on 8 H-[1,4]oxazino[2,3- f]quinolin-8-ones by Higuchi, Robert I., Thompson, Anthony W., Chen, Jyun-Hung, Caferro, Thomas R., Cummings, Marquis L., Deckhut, Charlotte P., Adams, Mark E., Tegley, Christopher M., Edwards, James P., López, Francisco J., Kallel, E. Adam, Karanewsky, Donald S., Schrader, William T., Marschke, Keith B., Zhi, Lin

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5( Z)-Benzylidene-1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5 H-1-aza-6-oxa-chrysenes as non-steroidal glucocorticoid receptor modulators by Ardecky, Robert J., Hudson, Andrew R., Phillips, Dean P., Tyhonas, John S., Deckhut, Charlotte, Lau, Thomas L., Li, Yongkai, Martinborough, Esther A., Roach, Steven L., Higuchi, Robert I., Lopez, Francisco J., Marschke, Keith B., Miner, Jeffrey N., Karanewsky, Donald S., Negro-Vilar, Andrés, Zhi, Lin

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