Food Increased the Bioavailability of BMS-690514, an Orally Active EGFR/HER2/VEGF Receptor Kinase Inhibitor, in Healthy Subjects by Vakkalagadda, Blisse, Park, Jong-Soon, Ahlers, Christoph M., Dorizio, Stephanie, Has, Teresa, Roongta, Vikram, Heller, Kevin N., Derbin, George M., Zhang, Steven

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Discovery and Evaluation of N-Cyclopropyl- 2,4-difluoro-5-((2-(pyridin-2-ylamino)thiazol-5- ylmethyl)amino)benzamide (BMS-605541), a Selective and Orally Efficacious Inhibitor of V... by Borzilleri, Robert M, Bhide, Rajeev S, Barrish, Joel C, D'Arienzo, Celia J, Derbin, George M, Fargnoli, Joseph, Hunt, John T, Jeyaseelan, Robert, Kamath, Amrita, Kukral, Daniel W, Marathe, Punit, Mortillo, Steve, Qian, Ligang, Tokarski, John S, Wautlet, Barri S, Zheng, Xiaoping, Lombardo, Louis J

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Discovery and evaluation of N-cyclopropyl-2,4-difluoro-5-(2-(pyridin-2-ylamino)thiazol-5-ylmethyl)aminobenzamide (BMS-605541), a selective and orally efficacious inhibitor of vascu... by BORZILLERI, Robert M, BHIDE, Rajeev S, MARATHE, Punit, MORTILLO, Steve, LIGANG QIAN, TOKARSKI, John S, WAUTLET, Barri S, XIAOPING ZHENG, LOMBARDO, Louis J, BARRISH, Joel C, D'ARIENZO, Celia J, DERBIN, George M, FARGNOLI, Joseph, HUNT, John T, JEYASEELAN, Robert, KAMATH, Amrita, KUKRAL, Daniel W

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Discovery and Preclinical Studies of (R)-1-(4-(4-Fluoro-2-methyl-1H-indol-5-yloxy)-5- methylpyrrolo[2,1-f][1,2,4]triazin-6-yloxy)propan- 2-ol (BMS-540215), an In Vivo Active Potent... by Bhide, Rajeev S, Cai, Zhen-Wei, Zhang, Yong-Zheng, Qian, Ligang, Wei, Donna, Barbosa, Stephanie, Lombardo, Louis J, Borzilleri, Robert M, Zheng, Xiaoping, Wu, Laurence I, Barrish, Joel C, Kim, Soong-Hoon, Leavitt, Kenneth, Mathur, Arvind, Leith, Leslie, Chao, Sam, Wautlet, Barri, Mortillo, Steven, Jeyaseelan, Robert, Kukral, Daniel, Hunt, John T, Kamath, Amrita, Fura, Aberra, Vyas, Viral, Marathe, Punit, D'Arienzo, Celia, Derbin, George, Fargnoli, Joseph

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Discovery of Brivanib Alaninate ((S)-((R)-1-(4-(4-Fluoro-2-methyl-1H-indol-5-yloxy)-5-methylpyrrolo[2,1-f][1,2,4]triazin-6-yloxy)propan-2-yl)2-aminopropanoate), A Novel Prodrug of... by Cai, Zhen-wei, Zhang, Yongzheng, Borzilleri, Robert M, Qian, Ligang, Barbosa, Stephanie, Wei, Donna, Zheng, Xiaoping, Wu, Lawrence, Fan, Junying, Shi, Zhongping, Wautlet, Barri S, Mortillo, Steve, Jeyaseelan, Robert, Kukral, Daniel W, Kamath, Amrita, Marathe, Punit, D’Arienzo, Celia, Derbin, George, Barrish, Joel C, Robl, Jeffrey A, Hunt, John T, Lombardo, Louis J, Fargnoli, Joseph, Bhide, Rajeev S

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Discovery of Brivanib Alaninate (S)-(R)-1-(4-(4-Fluoro-2-methyl-1H-indol-5-yloxy)-5-methylpyrrolo[2,1-f][1,2,4]triazin-6-yloxy)propan-2-yl2-aminopropanoate, A Novel Prodrug of Dual... by CAI, Zhen-Wei, YONGZHENG ZHANG, WAUTLET, Barri S, MORTILLO, Steve, JEYASEELAN, Robert, KUKRAL, Daniel W, KAMATH, Amrita, MARATHE, Punit, D'ARIENZO, Celia, DERBIN, George, BARRISH, Joel C, ROBL, Jeffrey A, BORZILLERI, Robert M, HUNT, John T, LOMBARDO, Louis J, FARGNOLI, Joseph, BHIDE, Rajeev S, LIGANG QIAN, BARBOSA, Stephanie, WEI, Donna, XIAOPING ZHENG, WU, Lawrence, JUNYING FAN, ZHONGPING SHI

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Discovery and preclinical studies of (R)-1-(4-(4-fluoro-2-methyl- 1H-indol-5-yloxy)-5-methylpyrrolo[2,1-/][1,2,4]triazin-6-yloxy)propan2-ol (BMS-540215), an in vivo active potent V... by BHIDE, Rajeev S, CAI, Zhen-Wei, BARRISH, Joel C, KIM, Soong-Hoon, LEAVITT, Kenneth, MATHUR, Arvind, LEITH, Leslie, CHAO, Sam, WAUTLET, Barri, MORTILLO, Steven, JEYASEELAN, Robert, KUKRAL, Daniel, ZHANG, Yong-Zheng, HUNT, John T, KAMATH, Amrita, FURA, Aberra, VYAS, Viral, MARATHE, Punit, D'ARIENZO, Celia, DERBIN, George, FARGNOLI, Joseph, LIGANG QIAN, WEI, Donna, BARBOSA, Stephanie, LOMBARDO, Louis J, BORZILLERI, Robert M, XIAOPING ZHENG, WU, Laurence I

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