Identification and Preliminary Characterization of a Potent, Safe, and Orally Efficacious Inhibitor of Acyl-CoA:Diacylglycerol Acyltransferase 1 by Yeh, Vince S. C, Beno, David W. A, Brodjian, Sevan, Brune, Michael E, Cullen, Steven C, Dayton, Brian D, Dhaon, Madhup K, Falls, Hugh D, Gao, Ju, Grihalde, Nelson, Hajduk, Philip, Hansen, T. Matthew, Judd, Andrew S, King, Andrew J, Klix, Russel C, Larson, Kelly J, Lau, Yau Y, Marsh, Kennan C, Mittelstadt, Scott W, Plata, Dan, Rozema, Michael J, Segreti, Jason A, Stoner, Eric J, Voorbach, Martin J, Wang, Xiaojun, Xin, Xili, Zhao, Gang, Collins, Christine A, Cox, Bryan F, Reilly, Regina M, Kym, Philip R, Souers, Andrew J

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Normal phase and reverse phase HPLC-UV-MS analysis of process impurities for rapamycin analog ABT-578: Application to active pharmaceutical ingredient process development by Chen, Yong, Brill, Gregory M., Benz, Nancy J., Leanna, M. Robert, Dhaon, Madhup K., Rasmussen, Michael, Zhou, Casey Chun, Bruzek, James A., Bellettini, John R.

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An intramolecular ionic hydrogen bond stabilizes a cis amide bond rotamer of a ring-opened rapamycin-degradation product by Zhou, Casey Chun, Stewart, Kent D., Dhaon, Madhup K.

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BOP-Cl mediated synthesis of the cyclosporine A 8-11 tetrapeptide fragment by Tung, Roger D, Dhaon, Madhup K, Rich, Daniel H

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Synthesis and antimitogenic activities of four analogs of cyclosporin A modified in the 1-position by Rich, Daniel H, Dhaon, Madhup K, Dunlap, Brian, Miller, Stephen P. F

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Esterification of N-protected .alpha.-amino acids with alcohol/carbodiimide/4-(dimethylamino)pyridine. Racemization of aspartic and glutamic acid derivatives by Dhaon, Madhup K, Olsen, Richard K, Ramasamy, K

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Synthesis, isolation, and characterization of ABT-578 equilibrium isomers by Dhaon, Madhup K., Zhou, Casey C., Chemburkar, Sanjay, Morton, Howard

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Synthesis of (MeAla)TANDEM, the bis(N-methylalanine) analog of des-N-tetramethyltriostin A by Dhaon, Madhup K, Olsen, Richard K

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A short synthesis of enantiomerically pure (2S,3R,4R,6E)-3-hydroxy-4-methyl-2-(methylamino)-6-octenoic acid, the unusual C9 amino acid found in the immunosuppressive peptide cyclos... by Aebi, Johannes D, Dhaon, Madhup K, Rich, Daniel H

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Derivatives of 2-methyl-1,4-naphthoquinone as substrates and inhibitors of the vitamin K-dependent carboxylase by Dhaon, Madhup K, Lehrman, S. R, Rich, D. H, Engelke, J. A, Suttie, J. W

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A short synthesis of enantiomerically pure (2S,3R,4R,6E)-3-hydroxy-4-methyl-2-(methylamino)-6-octenoic acid, the unusual C-9 amino acid found in the immunosuppressive peptide cyclo... by AEBI, J. D, DHAON, M. K, RICH, D. H

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