Structure–Activity Study of Bioisosteric Trifluoromethyl and Pentafluorosulfanyl Indole Inhibitors of the AAA ATPase p97 by Alverez, Celeste, Arkin, Michelle R, Bulfer, Stacie L, Colombo, Raffaele, Kovaliov, Marina, LaPorte, Matthew G, Lim, Chaemin, Liang, Mary, Moore, William J, Neitz, R. Jeffrey, Yan, Yongzhao, Yue, Zhizhou, Huryn, Donna M, Wipf, Peter

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Validation of HDAC8 Inhibitors as Drug Discovery Starting Points to Treat Acute Kidney Injury by Long, Keith, Vaughn, Zoe, McDaniels, Michael David, Joyasawal, Sipak, Przepiorski, Aneta, Parasky, Emily, Sander, Veronika, Close, David, Johnston, Paul A, Davidson, Alan J, de Caestecker, Mark, Hukriede, Neil A, Huryn, Donna M

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A threonine turnstile defines a dynamic amphiphilic binding motif in the AAA ATPase p97 allosteric binding site by Burnett, James C, Lim, Chaemin, Peyser, Brian D, Samankumara, Lalith P, Kovaliov, Marina, Colombo, Raffaele, Bulfer, Stacie L, LaPorte, Matthew G, Hermone, Ann R, McGrath, Connor F, Arkin, Michelle R, Gussio, Rick, Huryn, Donna M, Wipf, Peter

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Cyclopentane-1,3-dione: A Novel Isostere for the Carboxylic Acid Functional Group. Application to the Design of Potent Thromboxane (A2) Receptor Antagonists by Ballatore, Carlo, Soper, James H, Piscitelli, Francesco, James, Michael, Huang, Longchuan, Atasoylu, Onur, Huryn, Donna M, Trojanowski, John Q, Lee, Virginia M.-Y, Brunden, Kurt R, Smith, Amos B

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Optimization of Phenyl Indole Inhibitors of the AAA+ ATPase p97 by LaPorte, Matthew G, Burnett, James C, Colombo, Raffaele, Bulfer, Stacie L, Alverez, Celeste, Chou, Tsui-Fen, Neitz, R. Jeffrey, Green, Neal, Moore, William J, Yue, Zhizhou, Li, Shan, Arkin, Michelle R, Wipf, Peter, Huryn, Donna M

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Contributions of Academic Laboratories to the Discovery and Development of Chemical Biology Tools: Miniperspective by Huryn, Donna M, Resnick, Lynn O, Wipf, Peter

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Allosteric Indole Amide Inhibitors of p97: Identification of a Novel Probe of the Ubiquitin Pathway by Alverez, Celeste, Bulfer, Stacie L, Chakrasali, Ramappa, Chimenti, Michael. S, Deshaies, Raymond J, Green, Neal, Kelly, Mark, LaPorte, Matthew G, Lewis, Taber S, Liang, Mary, Moore, William J, Neitz, R. Jeffrey, Peshkov, Vsevolod A, Walters, Michael A, Zhang, Feng, Arkin, Michelle R, Wipf, Peter, Huryn, Donna M

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Virtual Special Issue: Epigenetics 2022 by Aldrich, Courtney C., Calderón, Félix, Conway, Stuart J., He, Chuan, Hooker, Jacob M., Huryn, Donna M., Lindsley, Craig W., Liotta, Dennis C., Müller, Christa E.

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Identification of Aminothienopyridazine Inhibitors of Tau Assembly by Quantitative High-Throughput Screening by Crowe, Alex, Huang, Wenwei, Ballatore, Carlo, Johnson, Ronald L, Hogan, Anne-Marie L, Huang, Ruili, Wichterman, Jennifer, McCoy, Joshua, Huryn, Donna, Auld, Douglas S, Smith, Amos B, Inglese, James, Trojanowski, John Q, Austin, Christopher P, Brunden, Kurt R, Lee, Virginia M.-Y

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Pyrimidinone-peptoid hybrid molecules with distinct effects on molecular chaperone function and cell proliferation by Wright, Christine M., Chovatiya, Raj J., Jameson, Nora E., Turner, David M., Zhu, Guangyu, Werner, Stefan, Huryn, Donna M., Pipas, James M., Day, Billy W., Wipf, Peter, Brodsky, Jeffrey L.

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Toxicity, pharmacokinetics and metabolism of a novel inhibitor of IL-6-induced STAT3 activation by Kiesel, Brian F., Parise, Robert A., Guo, Jianxia, Huryn, Donna M., Johnston, Paul A., Colombo, Raffaele, Sen, Malabika, Grandis, Jennifer R., Beumer, Jan H., Eiseman, Julie L.

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Virtual Special Issue: Epigenetics 2022 by Aldrich, Courtney C., Calderón, Félix, Conway, Stuart J., He, Chuan, Hooker, Jacob M., Huryn, Donna M., Lindsley, Craig W., Liotta, Dennis C., Müller, Christa E.

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2-Guanidinoquinazolines as new inhibitors of the STAT3 pathway by LaPorte, Matthew G., da Paz Lima, Dimas José, Zhang, Feng, Sen, Malabika, Grandis, Jennifer R., Camarco, Daniel, Hua, Yun, Johnston, Paul A., Lazo, John S., Resnick, Lynn O., Wipf, Peter, Huryn, Donna M.

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Abstract 2083: Toxicity, bioavailability, pharmacokinetics, tissue distribution and metabolism of a novel small molecule inhibitor of IL-6-induced STAT3 activation by Kiesel, Brian F., Parise, Robert A., Guo, Jianxia, Huryn, Donna M., Johnston, Paul A., Colombo, Rafaelle, Sen, Malabika, Grandis, Jennifer, Eiseman, Julie L., Beumer, Jan H.

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AIDS-driven nucleoside chemistry by Huryn, Donna M, Okabe, Masami

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Our Scope Expansion to Include Biologics by Maryanoff, Bruce E, Huryn, Donna M

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Kinetic Characterization and Molecular Docking of a Novel, Potent, and Selective Slow-Binding Inhibitor of Human Cathepsin L by Shah, Parag P, Myers, Michael C, Beavers, Mary Pat, Purvis, Jeremy E, Jing, Huiyan, Grieser, Heather J, Sharlow, Elizabeth R, Napper, Andrew D, Huryn, Donna M, Cooperman, Barry S, Smith, 3rd, Amos B, Diamond, Scott L

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Screening of 5-HT1A Receptor Antagonists using Molecularly Imprinted Polymers by O'Connor, Naphtali A, Paisner, David A, Huryn, Donna, Shea, Kenneth J

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Pharmaceutical profiling method for lipophilicity and integrity using liquid chromatography–mass spectrometry by Kerns, Edward H., Di, Li, Petusky, Susan, Kleintop, Teresa, Huryn, Donna, McConnell, Oliver, Carter, Guy

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Mechanism of action of selective inhibitors of IL-6 induced STAT3 pathway in head and neck cancer cell lines by Sen, Malabika, Johnston, Paul A., Pollock, Netanya I., DeGrave, Kara, Joyce, Sonali C., Freilino, Maria L., Hua, Yun, Camarco, Daniel P., Close, David A., Huryn, Donna M., Wipf, Peter, Grandis, Jennifer R.

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