A Focused Library of Tetrahydropyrimidinone Amides via a Tandem Biginelli-Ugi Multi-Component Process by Werner, Stefan, Turner, David M., Lyon, Michael A., Huryn, Donna M., Wipf, Peter

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Experimental Design on Single-Time-Point High-Throughput Microsomal Stability Assay by Di, Li, Kerns, Edward H., Gao, Ning, Li, Susan Q., Huang, Youping, Bourassa, Jim L., Huryn, Donna M.

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Optimization of a Higher Throughput Microsomal Stability Screening Assay for Profiling Drug Discovery Candidates by Di, Li, Kerns, Edward H., Hong, Yan, Kleintop, Teresa A., Mc Connell, Oliver J., Huryn, Donna M.

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Studies toward the discovery of the next generation of antidepressants. Part 6: Dual 5-HT1A receptor and serotonin transporter affinity within a class of arylpiperazinyl-cyclohexyl... by DAHUI ZHOU, PING ZHOU, SMITH, Deborah L, ANDREE, Terrance H, MEWSHAW, Richard E, EVRARD, Deborah A, MEAGHER, Kristin, WEBB, Michael, HARRISON, Boyd L, HURYN, Donna M, GOLEMBIESKI, Jeannette, HOMBY, Geoffrey A, SCHECHTER, Lee E

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Identification and characterization of 3-substituted pyrazolyl esters as alternate substrates for cathepsin B: The confounding effects of DTT and cysteine in biological assays by Myers, Michael C., Napper, Andrew D., Motlekar, Nuzhat, Shah, Parag P., Chiu, Chun-Hao, Beavers, Mary Pat, Diamond, Scott L., Huryn, Donna M., Smith, Amos B.

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Molecular Docking of Cathepsin L Inhibitors in the Binding Site of Papain by Beavers, Mary Pat, Myers, Michael C, Shah, Parag P, Purvis, Jeremy E, Diamond, Scott L, Cooperman, Barry S, Huryn, Donna M, Smith, Amos B

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Identification and synthesis of a unique thiocarbazate cathepsin L inhibitor by Myers, Michael C., Shah, Parag P., Diamond, Scott L., Huryn, Donna M., Smith, Amos B.

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Empowering Women in Organic Chemistry (EWOC) at Five Years: Giving Back and Getting Back by Cantor, Elinor H., Faul, Margaret M., Huryn, Donna M., Kallander, Lara, Ruck, Rebecca T., Watson, Mary P.

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Empowering Women in Organic Chemistry (EWOC) at Five Years: Giving Back and Getting Back by Cantor, Elinor H., Faul, Margaret M., Huryn, Donna M., Kallander, Lara, Ruck, Rebecca T., Watson, Mary P.

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Empowering Women in Organic Chemistry (EWOC) at Five Years: Giving Back and Getting Back by Cantor, Elinor H., Faul, Margaret M., Huryn, Donna M., Kallander, Lara, Ruck, Rebecca T., Watson, Mary P.

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Design, synthesis, and evaluation of inhibitors of cathepsin L: Exploiting a unique thiocarbazate chemotype by Myers, Michael C., Shah, Parag P., Beavers, Mary Pat, Napper, Andrew D., Diamond, Scott L., Smith, Amos B., Huryn, Donna M.

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Molecular Docking of Cathepsin L Inhibitors in the Binding Site of Papain by Beavers, Mary Pat, Myers, Michael C, Shah, Parag P, Purvis, Jeremy E, Diamond, Scott L, Cooperman, Barry S, Huryn, Donna M, Smith, Amos B

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Pharmacological Validation of HDAC8 as a Therapeutic Target for AKI: PO0331 by Huryn, Donna M., Long, Keith E., McDaniels, Michael D., Delgado, Rachel, Vaughn, Zoe, Iyer, Prema C., Sander, Veronika, Davidson, Alan J., de Caestecker, Mark P., Hukriede, Neil A.

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Synthesis and Biological Activity of a Focused Library of Mitogen-activated Protein Kinase Phosphatase Inhibitors by Arnold, David M., Foster, Caleb, Huryn, Donna M., Lazo, John S., Johnston, Paul A., Wipf, Peter

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Synthesis and Biological Evaluation of Benzodioxanylpiperazine Derivatives as Potent Serotonin 5-HT1A Antagonists:  The Discovery of Lecozotan by Childers, Wayne E, Abou-Gharbia, Magid A, Kelly, Michael G, Andree, Terrance H, Harrison, Boyd L, Ho, Douglas M, Hornby, Geoffrey, Huryn, Donna M, Potestio, Lisa, Rosenzweig-Lipson, Sharon J, Schmid, Jean, Smith, Deborah L, Sukoff, Stacey J, Zhang, Gan, Schechter, Lee E

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Virtual Special Issue: Epigenetics 2022 by Aldrich, Courtney C., Calderón, Félix, Conway, Stuart J., He, Chuan, Hooker, Jacob M., Huryn, Donna M., Lindsley, Craig W., Liotta, Dennis C., Müller, Christa E.

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Contributions of Academic Labs to the Discovery and Development of Chemical Biology Tools by Huryn, Donna M., Resnick, Lynn O., Wipf, Peter

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Begacestat (GSI-953): a novel, selective thiophene sulfonamide inhibitor of amyloid precursor protein gamma-secretase for the treatment of Alzheimer's disease by Martone, Robert L, Zhou, Hua, Atchison, Kevin, Comery, Thomas, Xu, Jane Z, Huang, Xinyi, Gong, Xioahai, Jin, Mei, Kreft, Anthony, Harrison, Boyd, Mayer, Scott C, Aschmies, Suzan, Gonzales, Cathleen, Zaleska, Margaret M, Riddell, David R, Wagner, Erik, Lu, Peimin, Sun, Shaiu-Ching, Sonnenberg-Reines, June, Oganesian, Aram, Adkins, Karissa, Leach, Michael W, Clarke, David W, Huryn, Donna, Abou-Gharbia, Magid, Magolda, Ronald, Bard, Jonathan, Frick, Glen, Raje, Sangeeta, Forlow, S Bradley, Balliet, Carrie, Burczynski, Michael E, Reinhart, Peter H, Wan, Hong I, Pangalos, Menelas N, Jacobsen, J Steven

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A threonine turnstile defines a dynamic amphiphilic binding motif in the AAA ATPase p97 allosteric binding siteElectronic supplementary information (ESI) available: Copies of 1H an... by Burnett, James C, Lim, Chaemin, Peyser, Brian D, Samankumara, Lalith P, Kovaliov, Marina, Colombo, Raffaele, Bulfer, Stacie L, LaPorte, Matthew G, Hermone, Ann R, McGrath, Connor F, Arkin, Michelle R, Gussio, Rick, Huryn, Donna M, Wipf, Peter

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Synthesis, characterization and evaluation of pro-drugs of VLA-4 antagonists by Huryn, Donna M, Ashwell, Susan, Baudy, Reinhardt, Dressen, Darren B, Gallaway, William, Grant, Francine S, Konradi, Andrei, Ley, Robert W, Petusky, Susan, Pleiss, Michael A, Sarantakis, Dimitri, Semko, Christopher M, Sherman, Mary M, Tio, Cesar, Zhang, Lu

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