Nonsteroidal Dissociated Glucocorticoid Agonists Containing Azaindoles as Steroid A-Ring Mimetics by Riether, Doris, Harcken, Christian, Razavi, Hossein, Kuzmich, Daniel, Gilmore, Thomas, Bentzien, Jörg, Pack, Edward J, Souza, Donald, Nelson, Richard M, Kukulka, Alison, Fadra, Tazmeen N, Zuvela-Jelaska, Ljiljana, Pelletier, Josephine, Dinallo, Roger, Panzenbeck, Mark, Torcellini, Carol, Nabozny, Gerald H, Thomson, David S

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Trifluoromethyl group as a pharmacophore : Effect of replacing a CF3 group on binding and agonist activity of a glucocorticoid receptor ligand by BETAGERI, Raj, YAN ZHANG, PAW, Zofia, SHIH, Daw-Tsun, SHIH, Cheng-Kon, ZUVELA-JELASKA, Ljiljana, NABOZNY, Gerald, THOMSON, David S, ZINDELL, Renee M, KUZMICH, Daniel, KIRRANE, Thomas M, BENTZIEN, Jörg, CARDOZO, Mario, CAPOLINO, Alison J, FADRA, Tazmeen N, NELSON, Richard M

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Non-steroidal dissociated glucocorticoid agonists: indoles as A-ring mimetics and function-regulating pharmacophores by Betageri, Raj, Gilmore, Thomas, Kuzmich, Daniel, Kirrane, Thomas M., Bentzien, Jörg, Wiedenmayer, Dieter, Bekkali, Younes, Regan, John, Berry, Angela, Latli, Bachir, Kukulka, Alison J., Fadra, Tazmeen N., Nelson, Richard M., Goldrick, Susan, Zuvela-Jelaska, Ljiljana, Souza, Don, Pelletier, Josephine, Dinallo, Roger, Panzenbeck, Mark, Torcellini, Carol, Lee, Heewon, Pack, Edward, Harcken, Christian, Nabozny, Gerald, Thomson, David S.

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Identification of Highly Efficacious Glucocorticoid Receptor Agonists with a Potential for Reduced Clinical Bone Side Effects by Harcken, Christian, Riether, Doris, Kuzmich, Daniel, Liu, Pingrong, Betageri, Raj, Ralph, Mark, Emmanuel, Michel, Reeves, Jonathan T, Berry, Angela, Souza, Donald, Nelson, Richard M, Kukulka, Alison, Fadra, Tazmeen N, Zuvela-Jelaska, Ljiljana, Dinallo, Roger, Bentzien, Jörg, Nabozny, Gerald H, Thomson, David S

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Discovery of a potent and dissociated non-steroidal glucocorticoid receptor agonist containing an alkyl carbinol pharmacophore by Razavi, Hossein, Riether, Doris, Harcken, Christian, Bentzien, Jörg, Dinallo, Roger M, Souza, Donald, Nelson, Richard M, Kukulka, Alison, Fadra-Khan, Tazmeen N, Pack, Jr, Edward J, Zuvela-Jelaska, Ljiljana, Pelletier, Josephine, Panzenbeck, Mark, Torcellini, Carol A, Proudfoot, John R, Nabozny, Gerald H, Thomson, David S

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Optimization of Drug-Like Properties of Nonsteroidal Glucocorticoid Mimetics and Identification of a Clinical Candidate by Harcken, Christian, Riether, Doris, Liu, Pingrong, Razavi, Hossein, Patel, Usha, Lee, Thomas, Bosanac, Todd, Ward, Yancey, Ralph, Mark, Chen, Zhidong, Souza, Donald, Nelson, Richard M, Kukulka, Alison, Fadra-Khan, Tazmeen N, Zuvela-Jelaska, Ljiljana, Patel, Mita, Thomson, David S, Nabozny, Gerald H

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Trifluoromethyl group as a pharmacophore: Effect of replacing a CF 3 group on binding and agonist activity of a glucocorticoid receptor ligand by Betageri, Raj, Zhang, Yan, Zindell, Renee M., Kuzmich, Daniel, Kirrane, Thomas M., Bentzien, Jörg, Cardozo, Mario, Capolino, Alison J., Fadra, Tazmeen N., Nelson, Richard M., Paw, Zofia, Shih, Daw-Tsun, Shih, Cheng-Kon, Zuvela-Jelaska, Ljiljana, Nabozny, Gerald, Thomson, David S.

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