Rational design of a new antibiotic class for drug-resistant infections by Durand-Reville, Thomas F., Miller, Alita A., O’Donnell, John P., Wu, Xiaoyun, Sylvester, Mark A., Guler, Satenig, Iyer, Ramkumar, Shapiro, Adam B., Carter, Nicole M., Velez-Vega, Camilo, Moussa, Samir H., McLeod, Sarah M., Chen, April, Tanudra, Angela M., Zhang, Jing, Comita-Prevoir, Janelle, Romero, Jan A., Huynh, Hoan, Ferguson, Andrew D., Horanyi, Peter S., Mayclin, Stephen J., Heine, Henry S., Drusano, George L., Cummings, Jason E., Slayden, Richard A., Tommasi, Ruben A.

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Antibacterial Inhibitors of Gram-Positive Thymidylate Kinase: Structure–Activity Relationships and Chiral Preference of a New Hydrophobic Binding Region by Kawatkar, Sameer P, Keating, Thomas A, Olivier, Nelson B, Breen, John N, Green, Oluyinka M, Guler, Satenig Y, Hentemann, Martin F, Loch, James T, McKenzie, Andrew R, Newman, Joseph V, Otterson, Linda G, Martínez-Botella, Gabriel

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In Vivo Validation of Thymidylate Kinase (TMK) with a Rationally Designed, Selective Antibacterial Compound by Keating, Thomas A, Newman, Joseph V, Olivier, Nelson B, Otterson, Linda G, Andrews, Beth, Boriack-Sjodin, P. Ann, Breen, John N, Doig, Peter, Dumas, Jacques, Gangl, Eric, Green, Oluyinka M, Guler, Satenig Y, Hentemann, Martin F, Joseph-McCarthy, Diane, Kawatkar, Sameer, Kutschke, Amy, Loch, James T, McKenzie, Andrew R, Pradeepan, Selvi, Prasad, Swati, Martínez-Botella, Gabriel

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Discovery of quinazoline HPK1 inhibitors with high cellular potency by Toure, Momar, Johnson, Theresa, Li, Bin, Schmidt, Ralf, Ma, Hong, Neagu, Constantin, Lopez, Andrea Unzue, Wang, Yanping, Guler, Satenig, Xiao, YuFang, Henkes, Renate, Ho, Kevin, Zhang, Susan, Chu, Chia Lin, Gundra, Uma Mahesh, Porichis, Filippos, Li, Long, Maurer, Christine Katharina, Fang, Zhizhou, Musil, Djordje, DiPoto, Maria, Friis, Emily, Jones, Reinaldo, Jones, Christopher, Cummings, James, Chekler, Eugene, Tanzer, Eva Maria, Huck, Bayard, Sherer, Brian

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Selective Wee1 Inhibitors Led to Antitumor Activity In Vitro and Correlated with Myelosuppression by Guler, Satenig, DiPoto, Maria C., Crespo, Alejandro, Caldwell, Richard, Doerfel, Benjamin, Grossmann, Nina, Ho, Kevin, Huck, Bayard, Jones, Christopher CV, Lan, Ruoxi, Musil, Djordje, Potnick, Justin, Schilke, Heike, Sherer, Brian, Simon, Stephanie, Sirrenberg, Christian, Zhang, Zhuo, Liu-Bujalski, Lesley

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Discovery of Selective and Potent Inhibitors of Gram-Positive Bacterial Thymidylate Kinase (TMK) by Martínez-Botella, Gabriel, Breen, John N, Duffy, James E. S, Dumas, Jacques, Geng, Bolin, Gowers, Ian K, Green, Oluyinka M, Guler, Satenig, Hentemann, Martin F, Hernandez-Juan, Felix A, Joseph-McCarthy, Diane, Kawatkar, Sameer, Larsen, Nicholas A, Lazari, Ovadia, Loch, James T, Macritchie, Jacqueline A, McKenzie, Andrew R, Newman, Joseph V, Olivier, Nelson B, Otterson, Linda G, Owens, Andrew P, Read, Jon, Sheppard, David W, Keating, Thomas A

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Selective inhibitors of tumor progression loci-2 (Tpl2) kinase with potent inhibition of TNF-α production in human whole blood by Wu, Junjun, Green, Neal, Hotchandani, Rajeev, Hu, Yonghan, Condon, Jeffrey, Huang, Adrian, Kaila, Neelu, Li, Huan-Qiu, Guler, Satenig, Li, Wei, Tam, Steve Y., Wang, Qin, Pelker, Jeffrey, Marusic, Suzana, Hsu, Sang, Perry Hall, J., Telliez, Jean-Baptiste, Cui, Junqing, Lin, Lih-Ling

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Inhibitors of Tumor Progression Loci-2 (Tpl2) Kinase and Tumor Necrosis Factor α (TNF-α) Production:  Selectivity and in Vivo Antiinflammatory Activity of Novel 8-Substituted-4-ani... by Green, Neal, Hu, Yonghan, Janz, Kristin, Li, Huan-Qiu, Kaila, Neelu, Guler, Satenig, Thomason, Jennifer, Joseph-McCarthy, Diane, Tam, Steve Y, Hotchandani, Rajeev, Wu, Junjun, Huang, Adrian, Wang, Qin, Leung, Louis, Pelker, Jefferey, Marusic, Suzana, Hsu, Sang, Telliez, Jean-Baptiste, Hall, J. Perry, Cuozzo, John W, Lin, Lih-Ling

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Continued exploration of biphenylsulfonamide scaffold as a platform for aggrecanase-1 inhibition by Hu, Yonghan, Xing, Li, Thomason, Jennifer R., Xiang, Jason, Ipek, Manus, Guler, Satenig, Li, Huanqiu, Sabatini, Joshua, Chockalingam, Priya, Reifenberg, Erica, Sheldon, Richard, Morris, Elisabeth A., Georgiadis, Katy E., Tam, Steve

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Inhibitors of tumor progression loci-2 (Tpl2) kinase and tumor necrosis factor a (TNF-α) production : Selectivity and in vivo antiinflammatory activity of novel 8-substituted-4-ani... by GREEN, Neal, YONGHAN HU, JUNJUN WU, HUANG, Adrian, QIN WANG, LEUNG, Louis, PELKER, Jefferey, MARUSIC, Suzana, HSU, Sang, TELLIEZ, Jean-Baptiste, HALL, J. Perry, CUOZZO, John W, JANZ, Kristin, LIN, Lih-Ling, LI, Huan-Qiu, KAILA, Neelu, GULER, Satenig, THOMASON, Jennifer, JOSEPH-MCCARTHY, Diane, TAM, Steve Y, HOTCHANDANI, Rajeev

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