Development of Highly Potent Inhibitors of Ras Farnesyltransferase Possessing Cellular and in Vivo Activity by Leftheris, Katerina, Kline, Toni, Vite, Gregory D, Cho, Young H, Bhide, Rajeev S, Patel, Dinesh V, Patel, Manorama M, Schmidt, Robert J, Weller, Harold N, Andahazy, Mary L, Carboni, Joan M, Gullo-Brown, Johnni L, Lee, Francis Y. F, Ricca, Carol, Rose, William C, Yan, Ning, Barbacid, Mariano, Hunt, John T, Meyers, Chester A, Seizinger, Bernd R, Zahler, Robert, Manne, Veeraswamy

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Phosphinyl acid-based bisubstrate analog inhibitors of ras farnesyl protein transferase by PATEL, D. V, GORDON, E. M, RICCA, C, ROBINSON, S, SEIZINGER, B. R, TUOMARI, A. V, MANNE, V, SCHMIDT, R. J, WELLER, H. N, YOUNG, M. G, ZAHLER, R, BARBACID, M, CARBONI, J. M, GULLO-BROWN, J. L, HUNIHAN, L

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Discovery of N-(4-(2-Amino-3-chloropyridin-4-yloxy)-3-fluorophenyl)-4-ethoxy-1-(4-fluorophenyl)-2-oxo-1,2-dihydropyridine-3-carboxamide (BMS-777607), a Selective and Orally Efficac... by Schroeder, Gretchen M, An, Yongmi, Cai, Zhen-Wei, Chen, Xiao-Tao, Clark, Cheryl, Cornelius, Lyndon A. M, Dai, Jun, Gullo-Brown, Johnni, Gupta, Ashok, Henley, Benjamin, Hunt, John T, Jeyaseelan, Robert, Kamath, Amrita, Kim, Kyoung, Lippy, Jonathan, Lombardo, Louis J, Manne, Veeraswamy, Oppenheimer, Simone, Sack, John S, Schmidt, Robert J, Shen, Guoxiang, Stefanski, Kevin, Tokarski, John S, Trainor, George L, Wautlet, Barri S, Wei, Donna, Williams, David K, Zhang, Yingru, Zhang, Yueping, Fargnoli, Joseph, Borzilleri, Robert M

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Discovery of Pyrrolopyridine−Pyridone Based Inhibitors of Met Kinase: Synthesis, X-ray Crystallographic Analysis, and Biological Activities by Kim, Kyoung Soon, Zhang, Liping, Schmidt, Robert, Cai, Zhen-Wei, Wei, Donna, Williams, David K, Lombardo, Louis J, Trainor, George L, Xie, Dianlin, Zhang, Yaquan, An, Yongmi, Sack, John S, Tokarski, John S, Darienzo, Celia, Kamath, Amrita, Marathe, Punit, Zhang, Yueping, Lippy, Jonathan, Jeyaseelan, Robert, Wautlet, Barri, Henley, Benjamin, Gullo-Brown, Johnni, Manne, Veeraswamy, Hunt, John T, Fargnoli, Joseph, Borzilleri, Robert M

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Design, synthesis, and structure–activity relationships of tetrahydroquinoline-based farnesyltransferase inhibitors by Lombardo, Louis J., Camuso, Amy, Clark, John, Fager, Krista, Gullo-Brown, Johnni, Hunt, John T., Inigo, Ivan, Kan, David, Koplowitz, Barry, Lee, Francis, McGlinchey, Kelly, Qian, Ligang, Ricca, Carolyn, Rovnyak, George, Traeger, Sarah, Tokarski, John, Williams, David K., Wu, Laurence I., Zhao, Yufen, Manne, Veeraswamy, Bhide, Rajeev S.

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Apoptotic and cytostatic farnesyltransferase inhibitors have distinct pharmacology and efficacy profiles in tumor models by MANNE, Veeraswamy, LEE, Francis Y. F, TAI WAI WONG, HUNT, John T, BOL, David K, GULLO-BROWN, Johnni, FAIRCHILD, Craig R, LOMBARDO, Louis J, SMYKLA, Richard A, VITE, Gregory D, WEN, Mei-Li D, YU, Chiang

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Design, synthesis and structure–activity relationships of novel biarylamine-based Met kinase inhibitors by Williams, David K., Chen, Xiao-Tao, Tarby, Christine, Kaltenbach, Robert, Cai, Zhen-Wei, Tokarski, John S., An, Yongmi, Sack, John S., Wautlet, Barri, Gullo-Brown, Johnni, Henley, Benjamin J., Jeyaseelan, Robert, Kellar, Kristen, Manne, Veeraswamy, Trainor, George L., Lombardo, Louis J., Fargnoli, Joseph, Borzilleri, Robert M.

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Phosphinyl Acid-Based Bisubstrate Analog Inhibitors of Farnesyl Protein Transferase by Patel, Dinesh V, Gordon, Eric M, Schmidt, Robert J, Weller, Harold N, Young, Marian G, Zahler, Robert, Barbacid, Mariano, Carboni, Joan M, Gullo-Brown, Johnni L, Hunihan, Lisa, Ricca, Carol, Robinson, Simon, Seizinger, Bernd R, Tuomari, Anne V, Manne, Veeraswamy

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