Molecular tuning of farnesoid X receptor partial agonism by Merk, Daniel, Sreeramulu, Sridhar, Kudlinzki, Denis, Saxena, Krishna, Linhard, Verena, Gande, Santosh L., Hiller, Fabian, Lamers, Christina, Nilsson, Ewa, Aagaard, Anna, Wissler, Lisa, Dekker, Niek, Bamberg, Krister, Schubert-Zsilavecz, Manfred, Schwalbe, Harald

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Chemiluminescence Biosensor for the Determination of Cardiac Troponin I (cTnI) by Tannenberg, Robert, Paul, Martin, Röder, Bettina, Gande, Santosh L, Sreeramulu, Sridhar, Saxena, Krishna, Richter, Christian, Schwalbe, Harald, Swart, Claudia, Weller, Michael G

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Light Dynamics of the Retinal‐Disease‐Relevant G90D Bovine Rhodopsin Mutant by Kubatova, Nina, Mao, Jiafei, Eckert, Carl Elias, Saxena, Krishna, Gande, Santosh L., Wachtveitl, Josef, Glaubitz, Clemens, Schwalbe, Harald

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Optimization of the Lead Compound NVP‐BHG712 as a Colorectal Cancer Inhibitor by Tröster, Alix, DiPrima, Michael, Jores, Nathalie, Kudlinzki, Denis, Sreeramulu, Sridhar, Gande, Santosh L., Linhard, Verena, Ludig, Damian, Schug, Alexander, Saxena, Krishna, Reinecke, Maria, Heinzlmeir, Stephanie, Leisegang, Matthias S., Wollenhaupt, Jan, Lennartz, Frank, Weiss, Manfred S., Kuster, Bernhard, Tosato, Giovanna, Schwalbe, Harald

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Binding Adaptation of GS-441524 Diversifies Macro Domains and Downregulates SARS-CoV-2 de-MARylation Capacity by Tsika, Aikaterini C., Gallo, Angelo, Fourkiotis, Nikolaos K., Argyriou, Aikaterini I., Sreeramulu, Sridhar, Löhr, Frank, Rogov, Vladimir V., Richter, Christian, Linhard, Verena, Gande, Santosh L., Altincekic, Nadide, Krishnathas, Robin, Elamri, Isam, Schwalbe, Harald, Wollenhaupt, Jan, Weiss, Manfred S., Spyroulias, Georgios A.

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Mechanistic Impact of Different Ligand Scaffolds on FXR Modulation Suggests Avenues to Selective Modulators by Heering, Jan, Jores, Nathalie, Kilu, Whitney, Schallmayer, Espen, Peelen, Evelyn, Muehler, Andreas, Kohlhof, Hella, Vitt, Daniel, Linhard, Verena, Gande, Santosh L., Chaikuad, Apirat, Sreeramulu, Sridhar, Schwalbe, Harald, Merk, Daniel

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Synthesis and in Vitro Evaluation of Novel 5‐Nitroindole Derivatives as c‐Myc G‐Quadruplex Binders with Anticancer Activity by Nimbarte, Vijaykumar D., Wirmer‐Bartoschek, Julia, Gande, Santosh L., Alshamleh, Islam, Seibert, Marcel, Nasiri, Hamid Reza, Schnütgen, Frank, Serve, Hubert, Schwalbe, Harald

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Targeting the Main Protease (Mpro, nsp5) by Growth of Fragment Scaffolds Exploiting Structure-Based Methodologies by Altincekic, Nadide, Jores, Nathalie, Löhr, Frank, Richter, Christian, Ehrhardt, Claus, Blommers, Marcel J. J., Berg, Hannes, Öztürk, Sare, Gande, Santosh L., Linhard, Verena, Orts, Julien, Abi Saad, Marie Jose, Bütikofer, Matthias, Kaderli, Janina, Karlsson, B. Göran, Brath, Ulrika, Hedenström, Mattias, Gröbner, Gerhard, Sauer, Uwe H., Perrakis, Anastassis, Langer, Julian, Banci, Lucia, Cantini, Francesca, Fragai, Marco, Grifagni, Deborah, Barthel, Tatjana, Wollenhaupt, Jan, Weiss, Manfred S., Robertson, Angus, Bax, Adriaan, Sreeramulu, Sridhar, Schwalbe, Harald

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NVP‐BHG712: Effects of Regioisomers on the Affinity and Selectivity toward the EPHrin Family by Tröster, Alix, Heinzlmeir, Stephanie, Berger, Benedict‐Tilman, Gande, Santosh L., Saxena, Krishna, Sreeramulu, Sridhar, Linhard, Verena, Nasiri, Amir H., Bolte, Michael, Müller, Susanne, Kuster, Bernhard, Médard, Guillaume, Kudlinzki, Denis, Schwalbe, Harald

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Structure and Biophysical Characterization of the S-Adenosylmethionine-dependent O-Methyltransferase PaMTH1, a Putative Enzyme Accumulating during Senescence of Podospora anserina by Chatterjee, Deep, Kudlinzki, Denis, Linhard, Verena, Saxena, Krishna, Schieborr, Ulrich, Gande, Santosh L., Wurm, Jan Philip, Wöhnert, Jens, Abele, Rupert, Rogov, Vladimir V., Dötsch, Volker, Osiewacz, Heinz D., Sreeramulu, Sridhar, Schwalbe, Harald

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Modulation of the Allosteric Communication between the Polo-Box Domain and the Catalytic Domain in Plk1 by Small Compounds by Raab, Monika, Sanhaji, Mourad, Pietsch, Larissa, Béquignon, Isabelle, Herbrand, Amanda K, Süß, Evelyn, Gande, Santosh L, Caspar, Birgit, Kudlinzki, Denis, Saxena, Krishna, Sreeramulu, Sridhar, Schwalbe, Harald, Strebhardt, Klaus, Biondi, Ricardo M

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Expression and Purification of EPHA2 Tyrosine Kinase Domain for Crystallographic and NMR Studies by Gande, Santosh L., Saxena, Krishna, Sreeramulu, Sridhar, Linhard, Verena, Kudlinzki, Denis, Heinzlmeir, Stephanie, Reichert, Andreas J., Skerra, Arne, Kuster, Bernhard, Schwalbe, Harald

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Light Dynamics of the Retinal‐Disease‐Relevant G90D Bovine Rhodopsin Mutant by Kubatova, Nina, Mao, Jiafei, Eckert, Carl Elias, Saxena, Krishna, Gande, Santosh L., Wachtveitl, Josef, Glaubitz, Clemens, Schwalbe, Harald

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Cover Feature: Optimization of the Lead Compound NVP‐BHG712 as a Colorectal Cancer Inhibitor (Chem. Eur. J. 23/2023) by Tröster, Alix, DiPrima, Michael, Jores, Nathalie, Kudlinzki, Denis, Sreeramulu, Sridhar, Gande, Santosh L., Linhard, Verena, Ludig, Damian, Schug, Alexander, Saxena, Krishna, Reinecke, Maria, Heinzlmeir, Stephanie, Leisegang, Matthias S., Wollenhaupt, Jan, Lennartz, Frank, Weiss, Manfred S., Kuster, Bernhard, Tosato, Giovanna, Schwalbe, Harald

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Comprehensive Fragment Screening of the SARS‐CoV‐2 Proteome Explores Novel Chemical Space for Drug Development by Berg, Hannes, Wirtz Martin, Maria A., Altincekic, Nadide, Alshamleh, Islam, Kaur Bains, Jasleen, Blechar, Julius, Ceylan, Betül, Jesus, Vanessa, Dhamotharan, Karthikeyan, Fuks, Christin, Gande, Santosh L., Hargittay, Bruno, Hohmann, Katharina F., Hutchison, Marie T., Marianne Korn, Sophie, Krishnathas, Robin, Kutz, Felicitas, Linhard, Verena, Matzel, Tobias, Meiser, Nathalie, Niesteruk, Anna, Pyper, Dennis J., Schulte, Linda, Trucks, Sven, Azzaoui, Kamal, Blommers, Marcel J. J., Gadiya, Yojana, Karki, Reagon, Zaliani, Andrea, Gribbon, Philip, Silva Almeida, Marcius, Dinis Anobom, Cristiane, Bula, Anna L., Bütikofer, Matthias, Putinhon Caruso, Ícaro, Caterina Felli, Isabella, Da Poian, Andrea T., Cardoso de Amorim, Gisele, Fourkiotis, Nikolaos K., Gallo, Angelo, Ghosh, Dhiman, Gomes‐Neto, Francisco, Gorbatyuk, Oksana, Hao, Bing, Kurauskas, Vilius, Lecoq, Lauriane, Li, Yunfeng, Cunha Mebus‐Antunes, Nathane, Mompeán, Miguel, Cristtina Neves‐Martins, Thais, Ninot‐Pedrosa, Martí, Pinheiro, Anderson S., Pontoriero, Letizia, Pustovalova, Yulia, Riek, Roland, Robertson, Angus J., Jose Abi Saad, Marie, Treviño, Miguel Á., Tsika, Aikaterini C., Almeida, Fabio C. L., Bax, Ad, Henzler‐Wildman, Katherine, Hoch, Jeffrey C., Jaudzems, Kristaps, Laurents, Douglas V., Orts, Julien, Pierattelli, Roberta, Spyroulias, Georgios A., Duchardt‐Ferner, Elke, Ferner, Jan, Fürtig, Boris, Hengesbach, Martin, Löhr, Frank, Qureshi, Nusrat, Richter, Christian, Saxena, Krishna, Schlundt, Andreas, Sreeramulu, Sridhar, Wacker, Anna, Weigand, Julia E., Wirmer‐Bartoschek, Julia, Wöhnert, Jens, Schwalbe, Harald

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Comprehensive Fragment Screening of the SARS‐CoV‐2 Proteome Explores Novel Chemical Space for Drug Development by Berg, Hannes, Wirtz Martin, Maria A., Altincekic, Nadide, Alshamleh, Islam, Kaur Bains, Jasleen, Blechar, Julius, Ceylan, Betül, Jesus, Vanessa, Dhamotharan, Karthikeyan, Fuks, Christin, Gande, Santosh L., Hargittay, Bruno, Hohmann, Katharina F., Hutchison, Marie T., Marianne Korn, Sophie, Krishnathas, Robin, Kutz, Felicitas, Linhard, Verena, Matzel, Tobias, Meiser, Nathalie, Niesteruk, Anna, Pyper, Dennis J., Schulte, Linda, Trucks, Sven, Azzaoui, Kamal, Blommers, Marcel J. J., Gadiya, Yojana, Karki, Reagon, Zaliani, Andrea, Gribbon, Philip, Silva Almeida, Marcius, Dinis Anobom, Cristiane, Bula, Anna L., Bütikofer, Matthias, Putinhon Caruso, Ícaro, Caterina Felli, Isabella, Da Poian, Andrea T., Cardoso de Amorim, Gisele, Fourkiotis, Nikolaos K., Gallo, Angelo, Ghosh, Dhiman, Gomes‐Neto, Francisco, Gorbatyuk, Oksana, Hao, Bing, Kurauskas, Vilius, Lecoq, Lauriane, Li, Yunfeng, Cunha Mebus‐Antunes, Nathane, Mompeán, Miguel, Cristtina Neves‐Martins, Thais, Ninot‐Pedrosa, Martí, Pinheiro, Anderson S., Pontoriero, Letizia, Pustovalova, Yulia, Riek, Roland, Robertson, Angus J., Jose Abi Saad, Marie, Treviño, Miguel Á., Tsika, Aikaterini C., Almeida, Fabio C. L., Bax, Ad, Henzler‐Wildman, Katherine, Hoch, Jeffrey C., Jaudzems, Kristaps, Laurents, Douglas V., Orts, Julien, Pierattelli, Roberta, Spyroulias, Georgios A., Duchardt‐Ferner, Elke, Ferner, Jan, Fürtig, Boris, Hengesbach, Martin, Löhr, Frank, Qureshi, Nusrat, Richter, Christian, Saxena, Krishna, Schlundt, Andreas, Sreeramulu, Sridhar, Wacker, Anna, Weigand, Julia E., Wirmer‐Bartoschek, Julia, Wöhnert, Jens, Schwalbe, Harald

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Molecular Characterization of the Human Cα-formylglycine-generating Enzyme by Preusser-Kunze, Andrea, Mariappan, Malaiyalam, Schmidt, Bernhard, Gande, Santosh Lakshmi, Mutenda, Kudzai, Wenzel, Dirk, von Figura, Kurt, Dierks, Thomas

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High-resolution crystal structure of cAMP-dependent protein kinase from Cricetulus griseus by Kudlinzki, Denis, Linhard, Verena L., Saxena, Krishna, Sreeramulu, Sridhar, Gande, Santosh, Schieborr, Ulrich, Dreyer, Matthias, Schwalbe, Harald

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Design and Isolation of Temperature-sensitive Mutants of Gal4 in Yeast and Drosophila by Mondal, Kajari, Dastidar, Antara Ghosh, Singh, Guramrit, Madhusudhanan, S., Gande, Santosh Lakshmi, VijayRaghavan, K., Varadarajan, Raghavan

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Expression, Localization, Structural, and Functional Characterization of pFGE, the Paralog of the Cα-Formylglycine-generating Enzyme by Mariappan, Malaiyalam, Preusser-Kunze, Andrea, Balleininger, Martina, Eiselt, Nicole, Schmidt, Bernhard, Gande, Santosh Lakshmi, Wenzel, Dirk, Dierks, Thomas, von Figura, Kurt

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