Iron-Catalyzed, Fluoroamide-Directed C–H Fluorination by Groendyke, Brian J, AbuSalim, Deyaa I, Cook, Silas P

Get full text

Fenton-Inspired C–H Functionalization: Peroxide-Directed C–H Thioetherification by Groendyke, Brian J, Modak, Atanu, Cook, Silas P

Get full text

Tubulin Resists Degradation by Cereblon-Recruiting PROTACs by Gasic, Ivana, Groendyke, Brian J, Nowak, Radosław P, Yuan, J Christine, Kalabathula, Joann, Fischer, Eric S, Gray, Nathanael S, Mitchison, Timothy J

Get full text

Development and Utility of a PAK1-Selective Degrader by Chow, Hoi-Yee, Karchugina, Sofiia, Groendyke, Brian J., Toenjes, Sean, Hatcher, John, Donovan, Katherine A., Fischer, Eric S., Abalakov, Gleb, Faezov, Bulat, Dunbrack, Roland, Gray, Nathanael S., Chernoff, Jonathan

Get full text

Exploration of the tunability of BRD4 degradation by DCAF16 trans-labelling covalent glues by Hassan, Muhammad Murtaza, Li, Yen-Der, Ma, Michelle W., Teng, Mingxing, Byun, Woong Sub, Puvar, Kedar, Lumpkin, Ryan, Sandoval, Brittany, Rutter, Justine C., Jin, Cyrus Y., Wang, Michelle Y., Xu, Shawn, Schmoker, Anna M., Cheong, Hakyung, Groendyke, Brian J., Qi, Jun, Fischer, Eric S., Ebert, Benjamin L., Gray, Nathanael S.

Get full text

Benzopyrimidodiazepinone inhibitors of TNK2 by Groendyke, Brian J., Powell, Chelsea E., Feru, Frederic, Gero, Thomas W., Li, Zhengnian, Szabo, Hilary, Pang, Kevin, Feutrill, John, Chen, Bailing, Li, Bin, Gray, Nathanael S., Scott, David A.

Get full text

Discovery of a series of benzopyrimidodiazepinone TNK2 inhibitors via scaffold morphing by Li, Zhengnian, Powell, Chelsea E., Groendyke, Brian J., Gero, Thomas W., Feru, Frederic, Feutrill, John, Chen, Bailing, Li, Bin, Szabo, Hilary, Gray, Nathanael S., Scott, David A.

Get full text

Discovery of a Pyrimidothiazolodiazepinone as a Potent and Selective Focal Adhesion Kinase (FAK) Inhibitor by Groendyke, Brian J, Nabet, Behnam, Mohardt, Mikaela L, Zhang, Haisheng, Peng, Ke, Koide, Eriko, Coffey, Calvin R, Che, Jianwei, Scott, David A, Bass, Adam J, Gray, Nathanael S

Get full text

Abstract 3424: Template-assisted covalent modification of DCAF16 enables BRD4 molecular glue degraders by Li, Yen-Der, Ma, Michelle W., Hassan, Muhammad Murtaza, Puvar, Kedar, Teng, Mingxing, Sandoval, Brittany, Lumpkin, Ryan, Ficarro, Scott B., Wang, Michelle Y., Xu, Shawn, Groendyke, Brian J., Sigua, Logan H., Tavares, Isidoro, Zou, Charles, Tsai, Jonathan M., Park, Paul M., Yoon, Hojong, Nowak, Radosław P., Marto, Jarrod A., Qi, Jun, Donovan, Katherine A., Słabicki, Mikołaj, Gray, Nathanael S., Fischer, Eric S., Ebert, Benjamin L.

Get full text

Mapping the Degradable Kinome Provides a Resource for Expedited Degrader Development by Donovan, Katherine A., Ferguson, Fleur M., Bushman, Jonathan W., Eleuteri, Nicholas A., Bhunia, Debabrata, Ryu, SeongShick, Tan, Li, Shi, Kun, Yue, Hong, Liu, Xiaoxi, Dobrovolsky, Dennis, Jiang, Baishan, Wang, Jinhua, Hao, Mingfeng, You, Inchul, Teng, Mingxing, Liang, Yanke, Hatcher, John, Li, Zhengnian, Manz, Theresa D., Groendyke, Brian, Hu, Wanyi, Nam, Yunju, Sengupta, Sandip, Cho, Hanna, Shin, Injae, Agius, Michael P., Ghobrial, Irene M., Ma, Michelle W., Che, Jianwei, Buhrlage, Sara J., Sim, Taebo, Gray, Nathanael S., Fischer, Eric S.

Get full text