Analysis of Tks4 Knockout Mice Suggests a Role for Tks4 in Adipose Tissue Homeostasis in the Context of Beigeing by Vas, Virag, Háhner, Tamás, Kudlik, Gyöngyi, Ernszt, Dávid, Kvell, Krisztián, Kuti, Dániel, Kovács, Krisztina J, Tóvári, József, Trexler, Mária, Merő, Balázs L, Szeder, Bálint, Koprivanacz, Kitti, Buday, László

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Determination of Ligand-Binding Affinity (K d) Using Transverse Relaxation Rate (R 2) in the Ligand-Observed 1H NMR Experiment and Applications to Fragment-Based Drug Discovery by Liu, Manjuan, Mirza, Amin, McAndrew, P. Craig, Thapaliya, Arjun, Pierrat, Olivier A., Stubbs, Mark, Hahner, Tamas, Chessum, Nicola E. A., Innocenti, Paolo, Caldwell, John, Cheeseman, Matthew D., Bellenie, Benjamin R., van Montfort, Rob L. M., Newton, Gary K., Burke, Rosemary, Collins, Ian, Hoelder, Swen

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A Degron Blocking Strategy Towards Improved CRL4CRBN Recruiting PROTAC Selectivity by Habib Bouguenina, Scarpino, Andrea, O'Hanlon, Jack A, Warne, Justin, Wang, Hannah Z, Laura Chan Wah Hak, Sadok, Amine, McAndrew, P Craig, Stubbs, Mark, Pierrat, Olivier A, Hahner, Tamas, Cabry, Marc P, Yann‐Vaï Le Bihan, Mitsopoulos, Costas, Sialana, Fernando J, Roumeliotis, Theodoros I, Burke, Rosemary, Rob L M van Montfort, Choudhari, Jyoti, Chopra, Rajesh, Caldwell, John J, Collins, Ian

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Front Cover: A Degron Blocking Strategy Towards Improved CRL4 CRBN Recruiting PROTAC Selectivity (ChemBioChem 23/2023) by Bouguenina, Habib, Scarpino, Andrea, O'Hanlon, Jack A., Warne, Justin, Wang, Hannah Z., Wah Hak, Laura Chan, Sadok, Amine, McAndrew, P. Craig, Stubbs, Mark, Pierrat, Olivier A., Hahner, Tamas, Cabry, Marc P., Le Bihan, Yann‐Vaï, Mitsopoulos, Costas, Sialana, Fernando J., Roumeliotis, Theodoros I., Burke, Rosemary, van Montfort, Rob L. M., Choudhari, Jyoti, Chopra, Rajesh, Caldwell, John J., Collins, Ian

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Front Cover: A Degron Blocking Strategy Towards Improved CRL4CRBN Recruiting PROTAC Selectivity by Habib Bouguenina, Scarpino, Andrea, O'Hanlon, Jack A, Warne, Justin, Wang, Hannah Z, Laura Chan Wah Hak, Sadok, Amine, McAndrew, P Craig, Stubbs, Mark, Pierrat, Olivier A, Hahner, Tamas, Cabry, Marc P, Yann‐Vaï Le Bihan, Mitsopoulos, Costas, Sialana, Fernando J, Roumeliotis, Theodoros I, Burke, Rosemary, Rob L M van Montfort, Choudhari, Jyoti, Chopra, Rajesh, Caldwell, John J, Collins, Ian

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Determination of Ligand-Binding Affinity ( K d ) Using Transverse Relaxation Rate ( R 2 ) in the Ligand-Observed 1 H NMR Experiment and Applications to Fragment-Based Drug Discover... by Liu, Manjuan, Mirza, Amin, McAndrew, P Craig, Thapaliya, Arjun, Pierrat, Olivier A, Stubbs, Mark, Hahner, Tamas, Chessum, Nicola E A, Innocenti, Paolo, Caldwell, John, Cheeseman, Matthew D, Bellenie, Benjamin R, van Montfort, Rob L M, Newton, Gary K, Burke, Rosemary, Collins, Ian, Hoelder, Swen

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A Degron Blocking Strategy Towards Improved CRL4 CRBN Recruiting PROTAC Selectivity by Bouguenina, Habib, Scarpino, Andrea, O'Hanlon, Jack A, Warne, Justin, Wang, Hannah Z, Wah Hak, Laura Chan, Sadok, Amine, McAndrew, P Craig, Stubbs, Mark, Pierrat, Olivier A, Hahner, Tamas, Cabry, Marc P, Le Bihan, Yann-Vaï, Mitsopoulos, Costas, Sialana, Fernando J, Roumeliotis, Theodoros I, Burke, Rosemary, van Montfort, Rob L M, Choudhari, Jyoti, Chopra, Rajesh, Caldwell, John J, Collins, Ian

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Investigating the phosphinic acid tripeptide mimetic DG013A as a tool compound inhibitor of the M1-aminopeptidase ERAP1 by Wilding, Birgit, Pasqua, A. Elisa, E. A. Chessum, Nicola, Pierrat, Olivier A., Hahner, Tamas, Tomlin, Kathy, Shehu, Erald, Burke, Rosemary, Richards, G. Meirion, Whitton, Bradleigh, Arwert, Esther N., Thapaliya, Arjun, Salimraj, Ramya, van Montfort, Rob, Skawinska, Agi, Hayes, Angela, Raynaud, Florence, Chopra, Rajesh, Jones, Keith, Newton, Gary, Cheeseman, Matthew D.

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