Discovery of 7‑Methyl-5-(1-{[3-(trifluoromethyl)phenyl]acetyl}-2,3-dihydro‑1H‑indol-5-yl)‑7H‑pyrrolo[2,3‑d]pyrimidin-4-amine (GSK2606414), a Potent and Selective First-in-Class Inh... by Axten, Jeffrey M, Medina, Jesús R, Feng, Yanhong, Shu, Arthur, Romeril, Stuart P, Grant, Seth W, Li, William Hoi Hong, Heerding, Dirk A, Minthorn, Elisabeth, Mencken, Thomas, Atkins, Charity, Liu, Qi, Rabindran, Sridhar, Kumar, Rakesh, Hong, Xuan, Goetz, Aaron, Stanley, Thomas, Taylor, J. David, Sigethy, Scott D, Tomberlin, Ginger H, Hassell, Annie M, Kahler, Kirsten M, Shewchuk, Lisa M, Gampe, Robert T

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Discovery of GSK2656157: An Optimized PERK Inhibitor Selected for Preclinical Development by Axten, Jeffrey M, Romeril, Stuart P, Shu, Arthur, Ralph, Jeffrey, Medina, Jesús R, Feng, Yanhong, Li, William Hoi Hong, Grant, Seth W, Heerding, Dirk A, Minthorn, Elisabeth, Mencken, Thomas, Gaul, Nathan, Goetz, Aaron, Stanley, Thomas, Hassell, Annie M, Gampe, Robert T, Atkins, Charity, Kumar, Rakesh

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Structures of human DPP7 reveal the molecular basis of specific inhibition and the architectural diversity of proline-specific peptidases by Bezerra, Gustavo Arruda, Dobrovetsky, Elena, Dong, Aiping, Seitova, Almagul, Crombett, Lissete, Shewchuk, Lisa M, Hassell, Annie M, Sweitzer, Sharon M, Sweitzer, Thomas D, McDevitt, Patrick J, Johanson, Kyung O, Kennedy-Wilson, Karen M, Cossar, Doug, Bochkarev, Alexey, Gruber, Karl, Dhe-Paganon, Sirano

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Exploration of the P1 SAR of aldehyde cathepsin K inhibitors by CATALANO, John G, DEATON, David N, FURFINE, Eric S, HASSELL, Annie M, MCFADYEN, Robert B, MILLER, Aaron B, MILLER, Larry R, SHEWCHUK, Lisa M, WILLARD, Derril H, WRIGHT, Lois L

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Discovery of 7-Methyl-5-(1-{[3-(trifluoromethyl)phenyl]acetyl}-2,3-dihydro-1 H -indol-5-yl)-7 H -pyrrolo[2,3- d ]pyrimidin-4-amine (GSK2606414), a Potent and Selective First-in-Cla... by Axten, Jeffrey M., Medina, Jesús R., Feng, Yanhong, Shu, Arthur, Romeril, Stuart P., Grant, Seth W., Li, William Hoi Hong, Heerding, Dirk A., Minthorn, Elisabeth, Mencken, Thomas, Atkins, Charity, Liu, Qi, Rabindran, Sridhar, Kumar, Rakesh, Hong, Xuan, Goetz, Aaron, Stanley, Thomas, Taylor, J. David, Sigethy, Scott D., Tomberlin, Ginger H., Hassell, Annie M., Kahler, Kirsten M., Shewchuk, Lisa M., Gampe, Robert T.

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Exploration of the P 1 SAR of aldehyde cathepsin K inhibitors by Catalano, John G., Deaton, David N., Furfine, Eric S., Hassell, Annie M., McFadyen, Robert B., Miller, Aaron B., Miller, Larry R., Shewchuk, Lisa M., Willard, Derril H., Wright, Lois L.

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The Drosophila Orphan Nuclear Receptor DHR38 Mediates an Atypical Ecdysteroid Signaling Pathway by Baker, Keith D., Shewchuk, Lisa M., Kozlova, Tatiana, Makishima, Makoto, Hassell, Annie, Wisely, Bruce, Caravella, Justin A., Lambert, Millard H., Reinking, Jeffrey L., Krause, Henry, Thummel, Carl S., Willson, Timothy M., Mangelsdorf, David J.

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Investigating the viability of genetic screening/testing for RA susceptibility using combinations of five confirmed risk loci by McClure, Annie, Lunt, Mark, Eyre, Steve, Ke, Xiayi, Thomson, Wendy, Hinks, Anne, Bowes, John, Gibbons, Laura, Plant, Darren, Wilson, Anthony G., Marinou, Ioanna, Morgan, Ann W., Emery, Paul, Steer, Sophia, Hocking, Lynne J., Reid, David M., Wordsworth, Paul, Harrison, Pille, Worthington, Jane, Barton, Anne

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