Discovery and Optimization of Tetramethylpiperidinyl Benzamides as Inhibitors of EZH2 by Nasveschuk, Christopher G, Gagnon, Alexandre, Garapaty-Rao, Shivani, Balasubramanian, Srividya, Campbell, Robert, Lee, Christina, Zhao, Feng, Bergeron, Louise, Cummings, Richard, Trojer, Patrick, Audia, James E, Albrecht, Brian K, Harmange, Jean-Christophe P

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Design and Synthesis of Styrenylcyclopropylamine LSD1 Inhibitors by Gehling, Victor S, McGrath, John P, Duplessis, Martin, Khanna, Avinash, Brucelle, Francois, Vaswani, Rishi G, Côté, Alexandre, Stuckey, Jacob, Watson, Venita, Cummings, Richard T, Balasubramanian, Srividya, Iyer, Priyadarshini, Sawant, Priyanka, Good, Andrew C, Albrecht, Brian K, Harmange, Jean-Christophe, Audia, James E, Bellon, Steven F, Trojer, Patrick, Levell, Julian R

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Novel 2,3-Dihydro-1,4-Benzoxazines as Potent and Orally Bioavailable Inhibitors of Tumor-Driven Angiogenesis by La, Daniel S, Belzile, Julie, Bready, James V, Coxon, Angela, DeMelfi, Thomas, Doerr, Nicholas, Estrada, Juan, Flynn, Julie C, Flynn, Shaun R, Graceffa, Russell F, Harriman, Shawn P, Larrow, Jay F, Long, Alexander M, Martin, Matthew W, Morrison, Michael J, Patel, Vinod F, Roveto, Philip M, Wang, Ling, Weiss, Matthew M, Whittington, Douglas A, Teffera, Yohannes, Zhao, Zhiyang, Polverino, Anthony J, Harmange, Jean-Christophe

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Naphthamides as Novel and Potent Vascular Endothelial Growth Factor Receptor Tyrosine Kinase Inhibitors: Design, Synthesis, and Evaluation by Harmange, Jean-Christophe, Weiss, Matthew M, Germain, Julie, Polverino, Anthony J, Borg, George, Bready, James, Chen, Danlin, Choquette, Deborah, Coxon, Angela, DeMelfi, Tom, DiPietro, Lucian, Doerr, Nicholas, Estrada, Juan, Flynn, Julie, Graceffa, Russell F, Harriman, Shawn P, Kaufman, Stephen, La, Daniel S, Long, Alexander, Martin, Matthew W, Neervannan, Sesha, Patel, Vinod F, Potashman, Michele, Regal, Kelly, Roveto, Phillip M, Schrag, Michael L, Starnes, Charlie, Tasker, Andrew, Teffera, Yohannes, Wang, Ling, White, Ryan D, Whittington, Douglas A, Zanon, Roger

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Collagen IVα345 dysfunction in glomerular basement membrane diseases. III. A functional framework for α345 hexamer assembly by Pedchenko, Vadim, Boudko, Sergei P., Barber, Mary, Mikhailova, Tatiana, Saus, Juan, Harmange, Jean-Christophe, Hudson, Billy G.

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Evaluation of indazole-based compounds as a new class of potent KDR/VEGFR-2 inhibitors by Bauer, David, Whittington, Douglas A., Coxon, Angela, Bready, James, Harriman, Shawn P., Patel, Vinod F., Polverino, Anthony, Harmange, Jean-Christophe

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Evaluation of a Series of Naphthamides as Potent, Orally Active Vascular Endothelial Growth Factor Receptor-2 Tyrosine Kinase Inhibitors by Weiss, Matthew M, Harmange, Jean-Christophe, Polverino, Anthony J, Bauer, David, Berry, Loren, Berry, Virginia, Borg, George, Bready, James, Chen, Danlin, Choquette, Deborah, Coxon, Angela, DeMelfi, Tom, Doerr, Nicholas, Estrada, Juan, Flynn, Julie, Graceffa, Russell F, Harriman, Shawn P, Kaufman, Stephen, La, Daniel S, Long, Alexander, Neervannan, Sesha, Patel, Vinod F, Potashman, Michele, Regal, Kelly, Roveto, Phillip M, Schrag, Michael L, Starnes, Charlie, Tasker, Andrew, Teffera, Yohannes, Whittington, Douglas A, Zanon, Roger

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Discovery of 2,4-bis-arylamino-1,3-pyrimidines as insulin-like growth factor-1 receptor (IGF-1R) inhibitors by Buchanan, John L., Newcomb, John R., Carney, David P., Chaffee, Stuart C., Chai, Lilly, Cupples, Rod, Epstein, Linda F., Gallant, Paul, Gu, Yan, Harmange, Jean-Christophe, Hodge, Kathy, Houk, Brett E., Huang, Xin, Jona, Janan, Joseph, Smriti, Jun, H. Toni, Kumar, Rakesh, Li, Chun, Lu, John, Menges, Tom, Morrison, Michael J., Novak, Perry M., van der Plas, Simon, Radinsky, Robert, Rose, Paul E., Sawant, Satin, Sun, Ji-Rong, Surapaneni, Sekhar, Turci, Susan M., Xu, Keyang, Yanez, Evelyn, Zhao, Huilin, Zhu, Xiaotian

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