Fast Iterative Synthetic Approach toward Identification of Novel Highly Selective p38 MAP Kinase Inhibitors by Röhm, Sandra, Berger, Benedict-Tilman, Schröder, Martin, Chaikuad, Apirat, Winkel, Rob, Hekking, Koen F. W, Benningshof, Jorg J. C, Müller, Gerhard, Tesch, Roberta, Kudolo, Mark, Forster, Michael, Laufer, Stefan, Knapp, Stefan

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Discovery of 2,4‑1H‑Imidazole Carboxamides as Potent and Selective TAK1 Inhibitors by Veerman, Johan J. N, Bruseker, Yorik B, Damen, Eddy, Heijne, Erik H, van Bruggen, Wendy, Hekking, Koen F. W, Winkel, Rob, Hupp, Christopher D, Keefe, Anthony D, Liu, Julie, Thomson, Heather A, Zhang, Ying, Cuozzo, John W, McRiner, Andrew J, Mulvihill, Mark J, van Rijnsbergen, Peter, Zech, Birgit, Renzetti, Louis M, Babiss, Lee, Müller, Gerhard

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Development of Potent Mcl‑1 Inhibitors: Structural Investigations on Macrocycles Originating from a DNA-Encoded Chemical Library Screen by Hekking, Koen F. W., Maroto, Sergio, van Kekem, Kees, Haasjes, Frank S., Slootweg, Jack C., Oude Alink, Patrick G. B., Dirks, Ron, Sardana, Malvika, Bolster, Marjon G., Kuijpers, Brian, Smith, Dennis, Doodeman, Robin, Scheepstra, Marcel, Zech, Birgit, Mulvihill, Mark, Renzetti, Louis M., Babiss, Lee, Centrella, Paolo A., Clark, Matthew A., Cuozzo, John W., Guié, Marie-Aude, Sigel, Eric, Habeshian, Sevan, Hupp, Christopher D., Liu, Julie, Thomson, Heather A., Zhang, Ying, Keefe, Anthony D., Müller, Gerhard, Gremmen, Stijn

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An In-Depth Study on Ring-Closing Metathesis of Carbohydrate-Derived α-Alkoxyacrylates:  Efficient Syntheses of DAH, KDO, and 2-Deoxy-β-KDO by Hekking, Koen F. W, Moelands, Marcel A. H, van Delft, Floris L, Rutjes, Floris P. J. T

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A Ring-Closing Metathesis Approach to Cyclic α,β-Dehydroamino Acids by Hekking, Koen F. W., Waalboer, Dennis C. J., Moelands, Marcel A. H., van Delft, Floris L., Rutjes, Floris P. J. T.

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Discovery of 2,4-1 H -Imidazole Carboxamides as Potent and Selective TAK1 Inhibitors by Veerman, Johan J N, Bruseker, Yorik B, Damen, Eddy, Heijne, Erik H, van Bruggen, Wendy, Hekking, Koen F W, Winkel, Rob, Hupp, Christopher D, Keefe, Anthony D, Liu, Julie, Thomson, Heather A, Zhang, Ying, Cuozzo, John W, McRiner, Andrew J, Mulvihill, Mark J, van Rijnsbergen, Peter, Zech, Birgit, Renzetti, Louis M, Babiss, Lee, Müller, Gerhard

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Synthesis of Versatile Building Blocks through Asymmetric Hydrogenation of Functionalized Itaconic Acid Mono-Esters by Hekking, Koen F. W., Lefort, Laurent, de Vries, André H. M., van Delft, Floris L., Schoemaker, Hans E., de Vries, Johannes G., Rutjes, Floris P. J. T.

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Bivalent Ligands for Protein Degradation in Drug Discovery by Scheepstra, Marcel, Hekking, Koen F.W., van Hijfte, Luc, Folmer, Rutger H.A.

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Effects of Extended Aryl-Substituted Bisoxazoline Ligands in Asymmetric Synthesis - Efficient Synthesis and Application of 4,4′-Bis(1-Naphthyl)-, 4,4′-Bis(2-Naphthyl)- and 4,4′-Bis... by van Lingen, Hester L., van Delft, Floris L., Storcken, Roy P. M., Hekking, Koen F. W., Klaassen, Anouk, Smits, Jan J. M., Ruskowska, Patrycja, Frelek, Jadwiga, Rutjes, Floris P. J. T.

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Cobalt Chloride Complexes of N3 and N4 Donor Ligands by Kooistra, T. Martijn, Hekking, Koen F. W., Knijnenburg, Quinten, de Bruin, Bas, Budzelaar, Peter H. M., de Gelder, René, Smits, Jan M. M., Gal, Anton W.

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Cobalt Chloride Complexes of N 3 and N 4 Donor Ligands by Kooistra, T. Martijn, Hekking, Koen F. W., Knijnenburg, Quinten, de Bruin, Bas, Budzelaar, Peter H. M., de Gelder, René, Smits, Jan M. M., Gal, Anton W.

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An Efficient Synthesis of 1-Naphthylbis(oxazoline) and Exploration of the Scope in Asymmetric Catalysis by van Lingen, Hester L., van de Mortel, Jeroen K. W., Hekking, Koen F. W., van Delft, Floris L., Sonke, Theo, Rutjes, Floris P. J. T.

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