AZD8931, an Equipotent, Reversible Inhibitor of Signaling by Epidermal Growth Factor Receptor, ERBB2 (HER2), and ERBB3: A Unique Agent for Simultaneous ERBB Receptor Blockade in Ca... by HICKINSON, D. Mark, KLINOWSKA, Teresa, MILLS, Elizabeth, GROSIOS, Konstantina, SMITH, Paul, BARLAAM, Bernard, WILKINSON, Robert W, OGILVIE, Donald, SPEAKE, Georgina, VINCENT, John, TRIGWELL, Cath, ANDERTON, Judith, BECK, Sarah, MARSHALL, Gayle, DAVENPORT, Sara, CALLIS, Rowena

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Preclinical anticancer activity of the potent, oral Src inhibitor AZD0530 by Green, Tim P., Fennell, Mike, Whittaker, Robin, Curwen, Jon, Jacobs, Vivien, Allen, Jack, Logie, Armelle, Hargreaves, Judith, Hickinson, D. Mark, Wilkinson, Robert W., Elvin, Paul, Boyer, Brigitte, Carragher, Neil, Plé, Patrick A., Bermingham, Alun, Holdgate, Geoffrey A., Ward, Walter H.J., Hennequin, Laurent F., Davies, Barry R., Costello, Gerard F.

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Novel 3-alkoxy-1H-pyrazolo[3,4-d]pyrimidines as EGFR and erbB2 receptor tyrosine kinase inhibitors by DUCRAY, Richard, BALLARD, Peter, BARLAAM, Bernard C, HICKINSON, Mark D, KETTLE, Jason G, OGILVIE, Donald J, TRIGWELL, Catherine B

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Discovery of AZD8931, an Equipotent, Reversible Inhibitor of Signaling by EGFR, HER2, and HER3 Receptors by Barlaam, Bernard, Anderton, Judith, Ballard, Peter, Bradbury, Robert H, Hennequin, Laurent F. A, Hickinson, D. Mark, Kettle, Jason G, Kirk, George, Klinowska, Teresa, Lambert-van der Brempt, Christine, Trigwell, Cath, Vincent, John, Ogilvie, Donald

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5-Substituted 4-anilinoquinazolines as potent, selective and orally active inhibitors of erbB2 receptor tyrosine kinase by Ballard, Peter, Bradbury, Robert H., Hennequin, Laurent F.A., Hickinson, D. Mark, Johnson, Paul D., Kettle, Jason G., Klinowska, Teresa, Morgentin, Remy, Ogilvie, Donald J., Olivier, Annie

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Neutral 5-substituted 4-anilinoquinazolines as potent, orally active inhibitors of erbB2 receptor tyrosine kinase by Ballard, Peter, Barlaam, Bernard C., Bradbury, Robert H., Dishington, Allan, Hennequin, Laurent F.A., Hickinson, D. Mark, Hollingsworth, Ian M., Kettle, Jason G., Klinowska, Teresa, Ogilvie, Donald J., Pearson, Stuart E., Scott, James S., Suleman, Abid, Whittaker, Robin, Williams, Emma J., Wood, Robin, Wright, Lindsay

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Src Family Kinase Inhibitor Saracatinib (AZD0530) Impairs Oxaliplatin Uptake in Colorectal Cancer Cells and Blocks Organic Cation Transporters by MORROW, Christopher J, GHATTAS, Mohammad, SMITH, Christopher, BÖNISCH, Heinz, BRYCE, Richard A, HICKINSON, D. Mark, GREEN, Tim P, DIVE, Caroline

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A new series of neutral 5-substituted 4-anilinoquinazolines as potent, orally active inhibitors of erbB2 receptor tyrosine kinase by Barlaam, Bernard, Ballard, Peter, Bradbury, Robert H., Ducray, Richard, Germain, Hervé, Hickinson, D. Mark, Hudson, Kevin, Kettle, Jason G., Klinowska, Teresa, Magnien, Françoise, Ogilvie, Donald J., Olivier, Annie, Pearson, Stuart E., Scott, James S., Suleman, Abid, Trigwell, Cath B., Vautier, Michel, Whittaker, Robin D., Wood, Robin

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Identification of Biomarkers in Human Head and Neck Tumor Cell Lines That Predict For In Vitro Sensitivity to Gefitinib by Hickinson, D. Mark, Marshall, Gayle B., Beran, Garry J., Varella-Garcia, Marileila, Mills, Elizabeth A., South, Marie C., Cassidy, Andrew M., Acheson, Kerry L, McWalter, Gael, McCormack, Rose M., Bunn, Paul A., French, Tim, Graham, Alex, Holloway, Brian R., Hirsch, Fred R., Speake, Georgina

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Inhibitors of epidermal growth factor receptor tyrosine kinase: Novel C-5 substituted anilinoquinazolines designed to target the ribose pocket by Ballard, Peter, Bradbury, Robert H., Harris, Craig S., Hennequin, Laurent F.A., Hickinson, Mark, Johnson, Paul D., Kettle, Jason G., Klinowska, Teresa, Leach, Andrew G., Morgentin, Remy, Pass, Martin, Ogilvie, Donald J., Olivier, Annie, Warin, Nicolas, Williams, Emma J.

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Inhibitors of epidermal growth factor receptor tyrosine kinase: Optimisation of potency and in vivo pharmacokinetics by Ballard, Peter, Bradbury, Robert H., Harris, Craig S., Hennequin, Laurent F.A., Hickinson, Mark, Kettle, Jason G., Kendrew, Jane, Klinowska, Teresa, Ogilvie, Donald J., Pearson, Stuart E., Williams, Emma J., Wilson, Ingrid

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Novel 3-alkoxy-1 H-pyrazolo[3,4- d]pyrimidines as EGFR and erbB2 receptor tyrosine kinase inhibitors by Ducray, Richard, Ballard, Peter, Barlaam, Bernard C., Hickinson, Mark D., Kettle, Jason G., Ogilvie, Donald J., Trigwell, Catherine B.

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