Resistance to pyridine-based inhibitor KF116 reveals an unexpected role of integrase in HIV-1 Gag-Pol polyprotein proteolytic processing by Hoyte, Ashley C., Jamin, Augusta V., Koneru, Pratibha C., Kobe, Matthew J., Larue, Ross C., Fuchs, James R., Engelman, Alan N., Kvaratskhelia, Mamuka

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HIV-1 integrase tetramers are the antiviral target of pyridine-based allosteric integrase inhibitors by Koneru, Pratibha C, Francis, Ashwanth C, Deng, Nanjie, Rebensburg, Stephanie V, Hoyte, Ashley C, Lindenberger, Jared, Adu-Ampratwum, Daniel, Larue, Ross C, Wempe, Michael F, Engelman, Alan N, Lyumkis, Dmitry, Fuchs, James R, Levy, Ronald M, Melikyan, Gregory B, Kvaratskhelia, Mamuka

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Identification and Optimization of a Novel HIV‑1 Integrase Inhibitor by Adu-Ampratwum, Daniel, Pan, Yuhan, Koneru, Pratibha C, Antwi, Janet, Hoyte, Ashley C, Kessl, Jacques, Griffin, Patrick R, Kvaratskhelia, Mamuka, Fuchs, James R, Larue, Ross C

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Computational and synthetic approaches for developing Lavendustin B derivatives as allosteric inhibitors of HIV-1 integrase by Agharbaoui, Fatima E., Hoyte, Ashley C., Ferro, Stefania, Gitto, Rosaria, Buemi, Maria Rosa, Fuchs, James R., Kvaratskhelia, Mamuka, De Luca, Laura

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The Competitive Interplay between Allosteric HIV‑1 Integrase Inhibitor BI/D and LEDGF/p75 during the Early Stage of HIV‑1 Replication Adversely Affects Inhibitor Potency by Feng, Lei, Dharmarajan, Venkatasubramanian, Serrao, Erik, Hoyte, Ashley, Larue, Ross C, Slaughter, Alison, Sharma, Amit, Plumb, Matthew R, Kessl, Jacques J, Fuchs, James R, Bushman, Frederic D, Engelman, Alan N, Griffin, Patrick R, Kvaratskhelia, Mamuka

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