A destabilizing Y891D mutation in activated EGFR impairs sensitivity to kinase inhibition by Lenchner, Daniel S., Petrova, Zaritza O., Hunihan, Lisa, Ashtekar, Kumar D., Walther, Zenta, Wilson, Frederick H.

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Identification and characterization of a MAPT-targeting locked nucleic acid antisense oligonucleotide therapeutic for tauopathies by Easton, Amy, Jensen, Marianne L., Wang, Congwei, Hagedorn, Peter H., Li, Yuwen, Weed, Michael, Meredith, Jere E., Guss, Valerie, Jones, Kelli, Gill, Martin, Krause, Carol, Brown, Jeffrey M., Hunihan, Lisa, Natale, Joanne, Fernandes, Alda, Lu, Yifeng, Polino, Joe, Bookbinder, Mark, Cadelina, Greg, Benitex, Yulia, Sane, Ramola, Morrison, John, Drexler, Dieter, Mercer, Stephen E., Bon, Charlotte, Pandya, Nikhil J., Jagasia, Ravi, Ou Yang, Tai-Hsien, Distler, Tania, Grüninger, Fiona, Meldgaard, Michael, Terrigno, Marco, Macor, John E., Albright, Charles F., Loy, James, Hoeg, Anja M., Olson, Richard E., Cacace, Angela M.

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Generation of a clonal induced pluripotent stem cell (iPSC) line expressing the mutant MECP2 allele from a Rett Syndrome patient fibroblast line by Hunihan, Lisa, Brown, Jeffrey, Cacace, Angela, Fernandes, Alda, Weston, Andrea

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RASGRF1 Fusions Activate Oncogenic RAS Signaling and Confer Sensitivity to MEK Inhibition by Hunihan, Lisa, Zhao, Dejian, Lazowski, Heather, Li, Man, Qian, Yuping, Abriola, Laura, Surovtseva, Yulia V, Muthusamy, Viswanathan, Tanoue, Lynn T, Rothberg, Bonnie E Gould, Schalper, Kurt A, Herbst, Roy S, Wilson, Frederick H

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Identification and Characterization of Compounds That Potentiate NT-3-Mediated Trk Receptor Activity by Lewis, Martin A., Hunihan, Lisa, Franco, Diana, Robertson, Barbara, Palmer, Jane, Laurent, Denis R. St, Balasubramanian, Balu N., Li, Yi, Westphal, Ryan S.

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A general liquid chromatography/mass spectroscopy-based assay for detection and quantitation of methyltransferase activity by Salyan, Mary Ellen K., Pedicord, Donna L., Bergeron, Laurie, Mintier, Gabe A., Hunihan, Lisa, Kuit, Kathy, Balanda, Lynn A., Robertson, Barbara J., Feder, John N., Westphal, Ryan, Shipkova, Petia A., Blat, Yuval

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Discovery, Structure–Activity Relationships, and In Vivo Evaluation of Novel Aryl Amides as Brain Penetrant Adaptor Protein 2‑Associated Kinase 1 (AAK1) Inhibitors for the Treatmen... by Hartz, Richard A, Ahuja, Vijay T, Nara, Susheel J, Kumar, C.M. Vijaya, Brown, Jeffrey M, Bristow, Linda J, Rajamani, Ramkumar, Muckelbauer, Jodi K, Camac, Daniel, Kiefer, Susan E, Hunihan, Lisa, Gulianello, Michael, Lewis, Martin, Easton, Amy, Lippy, Jonathan S, Surti, Neha, Pattipati, Sreenivasulu N, Dokania, Manoj, Elavazhagan, Saravanan, Dandapani, Kumaran, Hamman, Brian D, Allen, Jason, Kostich, Walter, Bronson, Joanne J, Macor, John E, Dzierba, Carolyn D

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Bicyclic Heterocyclic Replacement of an Aryl Amide Leading to Potent and Kinase-Selective Adaptor Protein 2‑Associated Kinase 1 Inhibitors by Hartz, Richard A, Ahuja, Vijay T, Nara, Susheel J, Kumar, C. M. Vijaya, Manepalli, Raju K. V. L. P, Sarvasiddhi, Sarat Kumar, Honkhambe, Swarnamba, Patankar, Vidya, Dasgupta, Bireshwar, Rajamani, Ramkumar, Muckelbauer, Jodi K, Camac, Daniel M, Ghosh, Kaushik, Pokross, Matthew, Kiefer, Susan E, Brown, Jeffrey M, Hunihan, Lisa, Gulianello, Michael, Lewis, Martin, Lippy, Jonathan S, Surti, Neha, Hamman, Brian D, Allen, Jason, Kostich, Walter A, Bronson, Joanne J, Macor, John E, Dzierba, Carolyn D

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In vitro Characterization of a small molecule inhibitor of the alanine serine cysteine transporter ‐1 (SLC7A10) by Brown, Jeffrey M., Hunihan, Lisa, Prack, Margaret M., Harden, David G., Bronson, Joanne, Dzierba, Carolyn D., Gentles, Robert G., Hendricson, Adam, Krause, Rudy, Macor, John E., Westphal, Ryan S.

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Molecular characterization and identification of surrogate substrates for diacylglycerol lipase α by Pedicord, Donna L., Flynn, Michael J., Fanslau, Caroline, Miranda, Maricar, Hunihan, Lisa, Robertson, Barbara J., Pearce, Bradley C., Yu, Xuan-Chuan, Westphal, Ryan S., Blat, Yuval

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A DNA-Binding Activity, TRAC, Specific for the TRA Element of the Transferrin Receptor Gene Copurifies with the Ku Autoantigen by Roberts, Margo R., Han, Young, Fienberg, Alan, Hunihan, Lisa, Ruddle, Francis H.

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Hydroxamic Acid-Based Bisubstrate Analog Inhibitors of Ras Farnesyl Protein Transferase by Patel, Dinesh V, Young, Marian G, Robinson, Simon P, Hunihan, Lisa, Dean, Brenda J, Gordon, Eric M

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Rational design of potent carboxylic acid based bisubstrate inhibitors of ras farnesyl protein transferase by Bhide, Rajeev S., Patel, Dinesh V., Patel, Manorama M., Robinson, Simon P., Hunihan, Lisa W., Gordon, Eric M.

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Phosphinyl Acid-Based Bisubstrate Analog Inhibitors of Farnesyl Protein Transferase by Patel, Dinesh V, Gordon, Eric M, Schmidt, Robert J, Weller, Harold N, Young, Marian G, Zahler, Robert, Barbacid, Mariano, Carboni, Joan M, Gullo-Brown, Johnni L, Hunihan, Lisa, Ricca, Carol, Robinson, Simon, Seizinger, Bernd R, Tuomari, Anne V, Manne, Veeraswamy

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