Pyrazole-Based Thrombin Inhibitors with a Serine-Trapping Mechanism of Action: Synthesis and Biological Activity by Dunker, Calvin, Imberg, Lukas, Siutkina, Alena I, Erbacher, Catharina, Daniliuc, Constantin G, Karst, Uwe, Kalinin, Dmitrii V

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N‐Pyrazolyl‐ and N‐Triazolylamines and ‐Ureas as Antileishmanial and Antitrypanosomal Drugs by Winge, Tobias, Imberg, Lukas, Perry, Ben, Matheeussen, An, Caljon, Guy, Kalinin, Dmitrii, Wünsch, Bernhard

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Microscale Parallel Synthesis of Acylated Aminotriazoles Enabling the Development of Factor XIIa and Thrombin Inhibitors by Platte, Simon, Korff, Marvin, Imberg, Lukas, Balicioglu, Ilker, Erbacher, Catharina, Will, Jonas M., Daniliuc, Constantin G., Karst, Uwe, Kalinin, Dmitrii V.

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Acylated 1 H -1,2,4-Triazol-5-amines Targeting Human Coagulation Factor XIIa and Thrombin: Conventional and Microscale Synthesis, Anticoagulant Properties, and Mechanism of Action by Korff, Marvin, Imberg, Lukas, Will, Jonas M, Bückreiß, Nico, Kalinina, Svetlana A, Wenzel, Benjamin M, Kastner, Gregor A, Daniliuc, Constantin G, Barth, Maximilian, Ovsepyan, Ruzanna A, Butov, Kirill R, Humpf, Hans-Ulrich, Lehr, Matthias, Panteleev, Mikhail A, Poso, Antti, Karst, Uwe, Steinmetzer, Torsten, Bendas, Gerd, Kalinin, Dmitrii V

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An automated analysis method enabling the screening of covalent thrombin and factor XIIa inhibitors via liquid chromatography‐mass spectrometry by Erbacher, Catharina, Athmer, Mathis, Kröger, Erik, Dahrendorf, Laureen, Imberg, Lukas, Kalinin, Dmitrii V., Karst, Uwe

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Acylated 1H‑1,2,4-Triazol-5-amines Targeting Human Coagulation Factor XIIa and Thrombin: Conventional and Microscale Synthesis, Anticoagulant Properties, and Mechanism of Action by Korff, Marvin, Imberg, Lukas, Will, Jonas M, Bückreiß, Nico, Kalinina, Svetlana A, Wenzel, Benjamin M, Kastner, Gregor A, Daniliuc, Constantin G, Barth, Maximilian, Ovsepyan, Ruzanna A, Butov, Kirill R, Humpf, Hans-Ulrich, Lehr, Matthias, Panteleev, Mikhail A, Poso, Antti, Karst, Uwe, Steinmetzer, Torsten, Bendas, Gerd, Kalinin, Dmitrii V

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Cover Feature: Microscale Parallel Synthesis of Acylated Aminotriazoles Enabling the Development of Factor XIIa and Thrombin Inhibitors (ChemMedChem 24/2021) by Platte, Simon, Korff, Marvin, Imberg, Lukas, Balicioglu, Ilker, Erbacher, Catharina, Will, Jonas M., Daniliuc, Constantin G., Karst, Uwe, Kalinin, Dmitrii V.

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Amide-functionalized 1,2,4-Triazol-5-amines as Covalent Inhibitors of Blood Coagulation Factor XIIa and Thrombin by Imberg, Lukas, Platte, Simon, Erbacher, Catharina, Daniliuc, Constantin G., Kalinina, Svetlana A., Dörner, Wolfgang, Poso, Antti, Karst, Uwe, Kalinin, Dmitrii V.

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Pyrazinyl-Substituted Aminoazoles as Covalent Inhibitors of Thrombin: Synthesis, Structure, and Anticoagulant Properties by Imberg, Lukas, Siutkina, Alena I., Erbacher, Catharina, Schmidt, Judith, Broekmans, Darius F., Ovsepyan, Ruzanna A., Daniliuc, Constantin G., Gonçalves de Oliveira, Ellen, Serafim, Mateus Sá Magalhães, O’Donoghue, Anthony J., Pillaiyar, Thanigaimalai, Panteleev, Mikhail A., Poso, Antti, Kalinina, Svetlana A., Bermúdez, Marcel, Nekipelov, Katrin, Bendas, Gerd, Karst, Uwe, Kalinin, Dmitrii V.

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