Pyronaridine-artesunate Shows Promise as an Effective and Well-tolerated Treatment for Artemisinin-resistant Plasmodium falciparum Malaria by Okombo, John, Fidock, David A

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Correction: Recent updates in the discovery and development of novel antimalarial drug candidates by Okombo, John, Chibale, Kelly

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Structure and drug resistance of the Plasmodium falciparum transporter PfCRT by Kim, Jonathan, Tan, Yong Zi, Wicht, Kathryn J., Erramilli, Satchal K., Dhingra, Satish K., Okombo, John, Vendome, Jeremie, Hagenah, Laura M., Giacometti, Sabrina I., Warren, Audrey L., Nosol, Kamil, Roepe, Paul D., Potter, Clinton S., Carragher, Bridget, Kossiakoff, Anthony A., Quick, Matthias, Fidock, David A., Mancia, Filippo

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Structure-activity relationship analyses of fusidic acid derivatives highlight crucial role of the C-21 carboxylic acid moiety to its anti-mycobacterial activity by Singh, Kawaljit, Kaur, Gurminder, Shanika, Petrus Siningu, Dziwornu, Godwin Akpeko, Okombo, John, Chibale, Kelly

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Malaria in the Era of Food Fortification With Folic Acid by Nzila, Alexis, Okombo, John, Hyde, John

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A Variant PfCRT Isoform Can Contribute to Plasmodium falciparum Resistance to the First-Line Partner Drug Piperaquine by Dhingra, Satish K, Redhi, Devasha, Combrinck, Jill M, Yeo, Tomas, Okombo, John, Henrich, Philipp P, Cowell, Annie N, Gupta, Purva, Stegman, Matthew L, Hoke, Jonathan M, Cooper, Roland A, Winzeler, Elizabeth, Mok, Sachel, Egan, Timothy J, Fidock, David A

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Impact of folate supplementation on the efficacy of sulfadoxine/pyrimethamine in preventing malaria in pregnancy: the potential of 5-methyl-tetrahydrofolate by Nzila, Alexis, Okombo, John, Molloy, Anne M

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Novel Antimalarial Tetrazoles and Amides Active against the Hemoglobin Degradation Pathway in Plasmodium falciparum by Lawong, Aloysus, Gahalawat, Suraksha, Okombo, John, Striepen, Josefine, Yeo, Tomas, Mok, Sachel, Deni, Ioanna, Bridgford, Jessica L, Niederstrasser, Hanspeter, Zhou, Anwu, Posner, Bruce, Wittlin, Sergio, Gamo, Francisco Javier, Crespo, Benigno, Churchyard, Alisje, Baum, Jake, Mittal, Nimisha, Winzeler, Elizabeth, Laleu, Benoît, Palmer, Michael J, Charman, Susan A, Fidock, David A, Ready, Joseph M, Phillips, Margaret A

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Synthesis and biological characterisation of ester and amide derivatives of fusidic acid as antiplasmodial agents by Espinoza-Moraga, Marlene, Singh, Kawaljit, Njoroge, Mathew, Kaur, Gurminder, Okombo, John, De Kock, Carmen, Smith, Peter J., Wittlin, Sergio, Chibale, Kelly

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Cytoplasmic isoleucyl tRNA synthetase as an attractive multistage antimalarial drug target by Istvan, Eva S, Guerra, Francisco, Abraham, Matthew, Huang, Kuo-Sen, Rocamora, Frances, Zhao, Haoshuang, Xu, Lan, Pasaje, Charisse, Kumpornsin, Krittikorn, Luth, Madeline R, Cui, Haissi, Yang, Tuo, Palomo Diaz, Sara, Gomez-Lorenzo, Maria G, Qahash, Tarrick, Mittal, Nimisha, Ottilie, Sabine, Niles, Jacquin, Lee, Marcus C S, Llinas, Manuel, Kato, Nobutaka, Okombo, John, Fidock, David A, Schimmel, Paul, Gamo, Francisco Javier, Goldberg, Daniel E, Winzeler, Elizabeth A

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Antimalarial Pyrido[1,2‑a]benzimidazole Derivatives with Mannich Base Side Chains: Synthesis, Pharmacological Evaluation, and Reactive Metabolite Trapping Studies by Okombo, John, Brunschwig, Christel, Singh, Kawaljit, Dziwornu, Godwin Akpeko, Barnard, Linley, Njoroge, Mathew, Wittlin, Sergio, Chibale, Kelly

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Systematic in vitro evolution in Plasmodium falciparum reveals key determinants of drug resistance by Luth, Madeline R, Godinez-Macias, Karla P, Chen, Daisy, Okombo, John, Thathy, Vandana, Cheng, Xiu, Daggupati, Sindhu, Davies, Heledd, Dhingra, Satish K, Economy, Jan M, Edgar, Rebecca C S, Gomez-Lorenzo, Maria G, Istvan, Eva S, Jado, Juan Carlos, LaMonte, Gregory M, Melillo, Bruno, Mok, Sachel, Narwal, Sunil K, Ndiaye, Tolla, Ottilie, Sabine, Palomo Diaz, Sara, Park, Heekuk, Peña, Stella, Rocamora, Frances, Sakata-Kato, Tomoyo, Small-Saunders, Jennifer L, Summers, Robert L, Tumwebaze, Patrick K, Vanaerschot, Manu, Xia, Guoqin, Yeo, Tomas, You, Ashley, Gamo, Francisco-Javier, Goldberg, Daniel E, Lee, Marcus C S, McNamara, Case W, Ndiaye, Daouda, Rosenthal, Philip J, Schreiber, Stuart L, Serra, Gloria, De Siqueira-Neto, Jair Lage, Skinner-Adams, Tina S, Uhlemann, Anne-Catrin, Kato, Nobutaka, Lukens, Amanda K, Wirth, Dyann F, Fidock, David A, Winzeler, Elizabeth A

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Cytoplasmic Isoleucyl tRNA synthetase as an attractive Multi-stage antimalarial drug target by Istvan, Eva S., Guerra, Francisco, Abraham, Matthew, Huang, Kuo-Sen, Rocamora, Frances, Zhao, Haoshuang, Xu, Lan, Pasaje, Charisse, Kumpornsin, Krittikorn, Luth, Madeline R., Cui, Haissi, Yang, Tuo, Diaz, Sara Palomo, Gomez-Lorenzo, Maria G., Qahash, Tarrick, Mittal, Nimisha, Ottilie, Sabine, Niles, Jacquin, Lee, Marcus C. S., Llinas, Manuel, Kato, Nobutaka, Okombo, John, Fidock, David A., Schimmel, Paul, Gamo, Francisco Javier, Goldberg, Daniel E., Winzeler, Elizabeth A.

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Advances in malaria pharmacology and the online guide to MALARIA PHARMACOLOGY: IUPHAR review 38 by Armstrong, Jane F., Campo, Brice, Alexander, Stephen P. H., Arendse, Lauren B., Cheng, Xiu, Davenport, Anthony P., Faccenda, Elena, Fidock, David A., Godinez‐Macias, Karla P., Harding, Simon D., Kato, Nobutaka, Lee, Marcus C. S., Luth, Madeline R., Mazitschek, Ralph, Mittal, Nimisha, Niles, Jacquin C., Okombo, John, Ottilie, Sabine, Pasaje, Charisse Flerida A., Probst, Alexandra S., Rawat, Mukul, Rocamora, Frances, Sakata‐Kato, Tomoyo, Southan, Christopher, Spedding, Michael, Tye, Mark A., Yang, Tuo, Zhao, Na, Davies, Jamie A.

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3‑Hydroxy-propanamidines, a New Class of Orally Active Antimalarials Targeting Plasmodium falciparum by Knaab, Tanja C, Held, Jana, Burckhardt, Bjoern B, Rubiano, Kelly, Okombo, John, Yeo, Tomas, Mok, Sachel, Uhlemann, Anne-Catrin, Lungerich, Beate, Fischli, Christoph, Pessanha de Carvalho, Lais, Mordmüller, Benjamin, Wittlin, Sergio, Fidock, David A, Kurz, Thomas

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4‑Aminoquinoline Antimalarials Containing a Benzyl­methyl­pyridyl­methyl­amine Group Are Active against Drug Resistant Plasmodium falciparum and Exhibit Oral Activity in Mice by Joshi, Mukesh C, Okombo, John, Nsumiwa, Samkele, Ndove, Jeffrey, Taylor, Dale, Wiesner, Lubbe, Hunter, Roger, Chibale, Kelly, Egan, Timothy J

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Antimalarial Pyrido[1,2‑a]benzimidazoles: Lead Optimization, Parasite Life Cycle Stage Profile, Mechanistic Evaluation, Killing Kinetics, and in Vivo Oral Efficacy in a Mouse Model... by Singh, Kawaljit, Okombo, John, Brunschwig, Christel, Ndubi, Ferdinand, Barnard, Linley, Wilkinson, Chad, Njogu, Peter M, Njoroge, Mathew, Laing, Lizahn, Machado, Marta, Prudêncio, Miguel, Reader, Janette, Botha, Mariette, Nondaba, Sindisiwe, Birkholtz, Lyn-Marie, Lauterbach, Sonja, Churchyard, Alisje, Coetzer, Theresa L, Burrows, Jeremy N, Yeates, Clive, Denti, Paolo, Wiesner, Lubbe, Egan, Timothy J, Wittlin, Sergio, Chibale, Kelly

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Mono- and polynuclear ferrocenylthiosemicarbazones: Synthesis, characterisation and antimicrobial evaluation by Baartzes, Nadia, Stringer, Tameryn, Okombo, John, Seldon, Ronnett, Warner, Digby F., de Kock, Carmen, Smith, Peter J., Smith, Gregory S.

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Pharmacokinetics and Organ Distribution of C‑3 Alkyl Esters as Potential Antimycobacterial Prodrugs of Fusidic Acid by Strydom, Natasha, Kaur, Gurminder, Dziwornu, Godwin Akpeko, Okombo, John, Wiesner, Lubbe, Chibale, Kelly

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Update on genetic markers of quinine resistance in Plasmodium falciparum by Okombo, John, Ohuma, Eric, Picot, Stephane, Nzila, Alexis

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