Diphenylsulfone muscarinic antagonists: piperidine derivatives with high m 2 selectivity and improved potency by Billard, William, Binch, Herbert, Bratzler, Kristen, Chen, Lian-Yong, Crosby, Gordon, Duffy, Ruth A, Dugar, Sundeep, Lachowicz, Jean, McQuade, Robert, Pushpavanam, Pradeep, Ruperto, Vilma B, Taylor, Lisa A, Clader, John W

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Metabolism and structure activity data based drug design: discovery of (−) SCH 53079 an analog of the potent cholesterol absorption inhibitor (−) SCH 48461 by Dugar, Syndeep, Yumibe, Nathan, Clader, John W., Vizziano, Monica, Huie, Keith, Van Heek, Margaret, Compton, Douglas S., Davis, Harry R.

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Metabolic stabilization of benzylidene ketal M 2 muscarinic receptor antagonists via halonaphthoic acid substitution by Boyle, Craig D., Chackalamannil, Samuel, Clader, John W., Greenlee, William J., Josien, Hubert B., Kaminski, James J., Kozlowski, Joseph A., McCombie, Stuart W., Nazareno, Dennis V., Tagat, Jayaram R., Wang, Yuguang, Zhou, Guowei, Billard, William, Binch, Herbert, Crosby, Gordon, Cohen-Williams, Mary, Coffin, Vicki L., Cox, Kathleen A., Grotz, Diane E., Duffy, Ruth A., Ruperto, Vilma, Lachowicz, Jean E.

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Stereoselective synthesis and biological activity of cis azetidinones as cholesterol absorption inhibitors by McKittrick, Brian A., Ma, Ke, Dugar, Sundeep, Clader, John W., Davis, Harry, Czarniecki, Michael, McPhail, Andrew T.

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(−)-SCH 57939: synthesis and pharmacological properties of a potent, metabolically stable cholesterol absorption inhibitor by Kirkup, Michael P., Rizvi, Razia, Shankar, Bandarpalle B., Dugar, Sundeep, Clader, John W., McCombie, Stuart W., Lin, Sue-Ing, Yumibe, Nathan, Huie, Keith, Van Heek, Margaret, Compton, Douglas S., Davis, Harry R., McPhail, Andrew T.

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Diphenylsulfone muscarinic antagonists: Piperidine derivatives with high M2 selectivity and improved potency by BILLARD, William, BINCH, Herbert III, RUPERTO, Vilma B, TAYLOR, Lisa A, CLADER, John W, BRATZLER, Kristen, CHEN, Lian-Yong, CROSBY, Gordon JR, DUFFY, Ruth A, DUGAR, Sundeep, LACHOWICZ, Jean, MCQUADE, Robert, PUSHPAVANAM, Pradeep

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N-oleoyl-1,2,3,4-tetrahydroisoquinolines as conformationally restricted inhibitors of acyl-CoA:cholesterol acyl transferase (ACAT) by Dugar, Sundeep, Clader, John W., Burrier, Robert E., Kogan, Timothy P.

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Rabbit and human liver contain a novel pentacyclic triterpene ester with acyl-CoA: cholesterol acyltransferase inhibitory activity by TABAS, I, LI-LING CHEN, ZIPKIN, R. E, BOYKOW, G, VITA, G, TALL, A. R, CLADER, J. W, MCPHAIL, A. T, BURNETT, D. A, BARTNER, P, DAS, P. R, PRAMANIK, B. N, PUAR, M. S, FEINMARK, S. J

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Gamma-lactams and related compounds as cholesterol absorption inhibitors: homologs of the beta-lactam cholesterol absorption inhibitor SCH 484611 by Dugar, Sundeep, Kirkup, Michael P., Clader, John W., Lin, Sue-Ing, Rizvi, Razia, Snow, Mark E., Davis, Harry R., McCombie, Stuart W.

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Facilitation of acetylcholine release and improvement in cognition by a selective M 2 muscarinic antagonist, SCH 72788 by Lachowicz, Jean E., Duffy, Ruth A., Ruperto, Vilma, Kozlowski, Joseph, Zhou, Guowei, Clader, John, Billard, William, Binch, Herbert, Crosby, Gordon, Cohen-Williams, Mary, Strader, Catherine D., Coffin, Victoria

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Design and synthesis of tricyclic sulfones as y-secretase inhibitors with greatly reduced Notch toxicity by RUO XU, COLE, David, JOSIEN, Hubert, HONGMEI LI, MCBRIAR, Mark, MCKITTRICK, Brian, MCPHAIL, Andrew T, PISSARNITSKI, Dmitri, LI QIANG, RAJAGOPALAN, Murali, SASILCUMAR, Thavalakulamgar, JING SU, ASBEROM, Ted, HAIQUN TANG, WU, Wen-Lian, LILI ZHANG, ZHIQIANG ZHAO, BARA, Tom, BENNETT, Chad, BURNETT, Duane A, CLADER, John, DOMALSKI, Martin, GREENLEE, William, HYDE, Lynn

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Improving the Oral Efficacy of CNS Drug Candidates:  Discovery of Highly Orally Efficacious Piperidinyl Piperidine M 2 Muscarinic Receptor Antagonists by Wang, Yuguang, Chackalamannil, Samuel, Hu, Zhiyong, Greenlee, William J., Clader, John, Boyle, Craig D., Kaminski, James J., Billard, William, Binch, Crosby, Gordon, Ruperto, Vilma, Duffy, Ruth A., Cohen-Williams, Mary, Coffin, Vicki L., Cox, Kathleen A., Grotz, Diane E., Lachowicz, Jean E.

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Inhibitors of Acyl CoA:Cholesterol Acyltransferase by Vaccaro, Wayne, Amore, Cindy, Berger, Joel, Burrier, Robert, Clader, John, Davis, Harry, Domalski, Martin, Fevig, Tom, Salisbury, Brian, Sher, Rosy

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Facilitation of acetylcholine release and improvement in cognition by a selective M2 muscarinic antagonist, SCH 72788 by Lachowicz, J E, Duffy, R A, Ruperto, V, Kozlowski, J, Zhou, G, Clader, J, Billard, W, Binch, 3rd, H, Crosby, G, Cohen-Williams, M, Strader, C D, Coffin, V

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