Pharmacology of Novel Heteroaromatic Polycycle Antibacterials by GROSS, M, BÜRLI, R, TANAKA, R, JOHNSON, K. W, JONES, P, GARCIA, M, BATISTE, B, KAIZERMAN, J, MOSER, H, JIANG, V, HOCH, U, DUAN, J.-X

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DNA binding ligands targeting drug-resistant Gram-positive bacteria. Part 1: Internal benzimidazole derivatives by Bürli, Roland W, McMinn, Dustin, Kaizerman, Jacob A, Hu, Wenhao, Ge, Yigong, Pack, Quinn, Jiang, Vernon, Gross, Matthew, Garcia, Martin, Tanaka, Richard, Moser, Heinz E

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DNA binding ligands targeting drug-resistant Gram-positive bacteria. Part 2: C-terminal benzimidazoles and derivatives by Bürli, Roland W, Jones, Peter, McMinn, Dustin, Le, Quan, Duan, Jian-Xin, Kaizerman, Jacob A, Difuntorum, Stacey, Moser, Heinz E

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DNA Binding Ligands with Improved in Vitro and in Vivo Potency against Drug-Resistant Staphylococcus aureus by Hu, Wenhao, Bürli, Roland W, Kaizerman, Jacob A, Johnson, Kirk W, Gross, Matthew I, Iwamoto, Mari, Jones, Peter, Lofland, Denene, Difuntorum, Stacey, Chen, Hsiu, Bozdogan, Bülent, Appelbaum, Peter C, Moser, Heinz E

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DNA Binding Ligands with Excellent Antibiotic Potency Against Drug-Resistant Gram-Positive Bacteria by Bürli, Roland W., Ge, Yigong, White, Sarah, Baird, Eldon E., Touami, Sofia M., Taylor, Matthew, Kaizerman, Jacob A., Moser, Heinz E.

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DNA Binding Ligands Targeting Drug-Resistant Bacteria:  Structure, Activity, and Pharmacology by Kaizerman, Jacob A, Gross, Matthew I, Ge, Yigong, White, Sarah, Hu, Wenhao, Duan, Jian-Xin, Baird, Eldon E, Johnson, Kirk W, Tanaka, Richard D, Moser, Heinz E, Bürli, Roland W

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DNA binding ligands with in vivo efficacy in murine models of bacterial infection: optimization of internal aromatic amino acids by BÜRLI, Roland W, KAIZERMAN, Jacob A, TOUAMI, Sofia, GROSS, Matthew, JIANG, Vernon, YIGONG GE, MOSER, Heinz E, DUAN, Jian-Xin, JONES, Peter, JOHNSON, Kirk W, IWAMOTO, Mari, TRUONG, Kiet, WENHAO HU, STANTON, Timothy, CHEN, Alfred

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Discovery of AMG 925, a FLT3 and CDK4 Dual Kinase Inhibitor with Preferential Affinity for the Activated State of FLT3 by Li, Zhihong, Wang, Xianghong, Eksterowicz, John, Gribble, Michael W, Alba, Grace Q, Ayres, Merrill, Carlson, Timothy J, Chen, Ada, Chen, Xiaoqi, Cho, Robert, Connors, Richard V, DeGraffenreid, Michael, Deignan, Jeffrey T, Duquette, Jason, Fan, Pingchen, Fisher, Benjamin, Fu, Jiasheng, Huard, Justin N, Kaizerman, Jacob, Keegan, Kathleen S, Li, Cong, Li, Kexue, Li, Yunxiao, Liang, Lingming, Liu, Wen, Lively, Sarah E, Lo, Mei-Chu, Ma, Ji, McMinn, Dustin L, Mihalic, Jeffrey T, Modi, Kriti, Ngo, Rachel, Pattabiraman, Kanaka, Piper, Derek E, Queva, Christophe, Ragains, Mark L, Suchomel, Julia, Thibault, Steve, Walker, Nigel, Wang, Xiaodong, Wang, Zhulun, Wanska, Malgorzata, Wehn, Paul M, Weidner, Margaret F, Zhang, Alex J, Zhao, Xiaoning, Kamb, Alexander, Wickramasinghe, Dineli, Dai, Kang, McGee, Lawrence R, Medina, Julio C

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Discovery of amide replacements that improve activity and metabolic stability of a bis-amide smoothened antagonist hit by Brown, Matthew L., Aaron, Wade, Austin, Richard J., Chong, Angela, Huang, Tom, Jiang, Ben, Kaizerman, Jacob A., Lee, Gary, Lucas, Brian S., McMinn, Dustin L., Orf, Jessica, Rong, Minqing, Toteva, Maria M., Xu, Guifen, Ye, Qiuping, Zhong, Wendy, DeGraffenreid, Michael R., Wickramasinghe, Dineli, Powers, Jay P., Hungate, Randall, Johnson, Michael G.

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Design of 1-piperazinyl-4-arylphthalazines as potent Smoothened antagonists by Lucas, Brian S., Aaron, Wade, An, Songzhu, Austin, Richard J., Brown, Matthew, Chan, Hon, Chong, Angela, Hungate, Randall, Huang, Tom, Jiang, Ben, Johnson, Michael G., Kaizerman, Jacob A., Lee, Gary, McMinn, Dustin L., Orf, Jessica, Powers, Jay P., Rong, Minqing, Toteva, Maria M., Uyeda, Craig, Wickramasinghe, Dineli, Xu, Guifen, Ye, Qiuping, Zhong, Wendy

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