Discovery of a Novel Class of Dimeric Smac Mimetics as Potent IAP Antagonists Resulting in a Clinical Candidate for the Treatment of Cancer (AZD5582) by Hennessy, Edward J, Adam, Ammar, Aquila, Brian M, Castriotta, Lillian M, Cook, Donald, Hattersley, Maureen, Hird, Alexander W, Huntington, Christopher, Kamhi, Victor M, Laing, Naomi M, Li, Danyang, MacIntyre, Terry, Omer, Charles A, Oza, Vibha, Patterson, Troy, Repik, Galina, Rooney, Michael T, Saeh, Jamal C, Sha, Li, Vasbinder, Melissa M, Wang, Haiyun, Whitston, David

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Structure-based design and synthesis of tricyclic IAP (Inhibitors of Apoptosis Proteins) inhibitors by Hird, Alexander W., Aquila, Brian M., Block, Michael H., Hennessy, Edward J., Kamhi, Victor M., Omer, Charles A., Laing, Naomi M., Saeh, Jamal C., Sha, Li, Yang, Bin

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Identification and Optimization of Benzimidazole Sulfonamides as Orally Bioavailable Sphingosine 1‑Phosphate Receptor 1 Antagonists with in Vivo Activity by Hennessy, Edward J., Oza, Vibha, Adam, Ammar, Byth, Kate, Castriotta, Lillian, Grewal, Gurmit, Hamilton, Geraldine A., Kamhi, Victor M., Lewis, Paula, Li, Danyang, Lyne, Paul, Öster, Linda, Rooney, Michael T., Saeh, Jamal C., Sha, Li, Su, Qibin, Wen, Shengua, Xue, Yafeng, Yang, Bin

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Discovery of heterocyclic sulfonamides as sphingosine 1-phosphate receptor 1 (S1P1) antagonists by Hennessy, Edward J., Grewal, Gurmit, Byth, Kate, Kamhi, Victor M., Li, Danyang, Lyne, Paul, Oza, Vibha, Ronco, Lucienne, Rooney, Michael T., Saeh, Jamal C., Su, Qibin

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