Small-molecule p21-activated kinase inhibitor PF-3758309 is a potent inhibitor of oncogenic signaling and tumor growth by Murray, Brion W, Guo, Chuangxing, Piraino, Joseph, Westwick, John K, Zhang, Cathy, Lamerdin, Jane, Dagostino, Eleanor, Knighton, Daniel, Loi, Cho-Ming, Zager, Michael, Kraynov, Eugenia, Popoff, Ian, Christensen, James G, Martinez, Ricardo, Kephart, Susan E, Marakovits, Joseph, Karlicek, Shannon, Bergqvist, Simon, Smeal, Tod

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Osteopontin induces growth of metastatic tumors in a preclinical model of non-small lung cancer by Shojaei, Farbod, Scott, Nathan, Kang, Xiaolin, Lappin, Patrick B, Fitzgerald, Amanda A, Karlicek, Shannon, Simmons, Brett H, Wu, Aidong, Lee, Joseph H, Bergqvist, Simon, Kraynov, Eugenia

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SAM-Competitive PRMT5 Inhibitor PF-06939999 Demonstrates Antitumor Activity in Splicing Dysregulated NSCLC with Decreased Liability of Drug Resistance by Jensen-Pergakes, Kristen, Tatlock, John, Maegley, Karen A, McAlpine, Indrawan J, McTigue, Michele, Xie, Tao, Dillon, Christopher P, Wang, Yuli, Yamazaki, Shinji, Spiegel, Noah, Shi, Manli, Nemeth, Amy, Miller, Natalie, Hendrickson, Eleanore, Lam, Hieu, Sherrill, John, Chung, Chi-Yeh, McMillan, Elizabeth A, Bryant, Shannon Karlicek, Palde, Prakash, Braganza, John, Brooun, Alexei, Deng, Ya-Li, Goshtasbi, Vesta, Kephart, Susan E, Kumpf, Robert A, Liu, Wei, Patman, Ryan L, Rui, Eugene, Scales, Stephanie, Tran-Dube, Michelle, Wang, Fen, Wythes, Martin, Paul, Thomas A

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Enzymatic Characterization of c-Met Receptor Tyrosine Kinase Oncogenic Mutants and Kinetic Studies with Aminopyridine and Triazolopyrazine Inhibitors by Timofeevski, Sergei L, McTigue, Michele A, Ryan, Kevin, Cui, Jean, Zou, Helen Y, Zhu, Jeff X, Chau, Fannie, Alton, Gordon, Karlicek, Shannon, Christensen, James G, Murray, Brion W

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Abstract 4456: Biochemical and structural characteristics of crizotinib-resistant ALK mutants by Timofeevski, Sergei, Liu, Wei, Deng, Ya-Li, Brooun, Alexei, Bergqvist, Simon, Karlicek, Shannon, Murray, Brion, Bolaños, Ben, McTigue, Michele

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Comparative analyses of a small molecule/enzyme interaction by multiple users of Biacore technology by Cannon, Michelle J, Papalia, Giuseppe A, Navratilova, Iva, Fisher, Robert J, Roberts, Lindsey R, Worthy, Karen M, Stephen, Andrew G, Marchesini, Gerardo R, Collins, Edward J, Casper, Dave, Qiu, Huawei, Satpaev, Daulet, Liparoto, Stefano F, Rice, Dax A, Gorshkova, Inna I, Darling, Ryan J, Bennett, Donald B, Sekar, Michael, Hommema, Eric, Liang, Amy M, Day, Eric S, Inman, Jean, Karlicek, Shannon M, Ullrich, Stephen J, Hodges, Dianne, Chu, Teresa, Sullivan, Eric, Simpson, Jack, Rafique, Ashique, Luginbühl, Béatrice, Westin, Susanne Nyholm, Bynum, Magdalena, Cachia, Paul, Li, Yue-Jin, Kao, Daniel, Neurauter, Amy, Wong, Melanie, Swanson, Michael, Myszka, David G

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