Mechanism-Based Competitive Inhibitors of Glyoxalase I:  Intracellular Delivery, in Vitro Antitumor Activities, and Stabilities in Human Serum and Mouse Serum by Kavarana, Malcolm J, Kovaleva, Elena G, Creighton, Donald J, Wollman, Megan B, Eiseman, Julie L

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Reaction Mechanism of Glyoxalase I Explored by an X-ray Crystallographic Analysis of the Human Enzyme in Complex with a Transition State Analogue by Cameron, Alexander D, Ridderström, Marianne, Olin, Birgit, Kavarana, Malcolm J, Creighton, Donald J, Mannervik, Bengt

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Exploration of amino alcohol derivatives as novel, potent, and highly selective sphingosine-1-phosphate receptor subtype-1 agonists by Evindar, Ghotas, Bernier, Sylvie G., Doyle, Elisabeth, Kavarana, Malcolm J., Satz, Alexander L., Lorusso, Jeanine, Blanchette, Heather S., Saha, Ashis K., Hannig, Gerhard, Morgan, Barry A., Westlin, William F.

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Synthesis and evaluation of alkoxy-phenylamides and alkoxy-phenylimidazoles as potent sphingosine-1-phosphate receptor subtype-1 agonists by Evindar, Ghotas, Bernier, Sylvie G., Kavarana, Malcolm J., Doyle, Elisabeth, Lorusso, Jeanine, Kelley, Michael S., Halley, Keith, Hutchings, Amy, Wright, Albion D., Saha, Ashis K., Hannig, Gerhard, Morgan, Barry A., Westlin, William F.

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Novel Cyclic Templates of α-MSH Give Highly Selective and Potent Antagonists/Agonists for Human Melanocortin-3/4 Receptors by Kavarana, Malcolm J, Trivedi, Dev, Cai, Minying, Ying, Jinfa, Hammer, Matthew, Cabello, Christopher, Grieco, Paolo, Han, Guoxia, Hruby, Victor J

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Synthesis and evaluation of arylalkoxy- and biarylalkoxy-phenylamide and phenylimidazoles as potent and selective sphingosine-1-phosphate receptor subtype-1 agonists by Evindar, Ghotas, Satz, Alexander L., Bernier, Sylvie G., Kavarana, Malcolm J., Doyle, Elisabeth, Lorusso, Jeanine, Taghizadeh, Nazbeh, Halley, Keith, Hutchings, Amy, Kelley, Michael S., Wright, Albion D., Saha, Ashis K., Hannig, Gerhard, Morgan, Barry A., Westlin, William F.

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Solution structures of cyclic melanocortin agonists and antagonists by NMR by Ying, Jinfa, Kövér, Katalin E., Gu, Xuyuan, Han, Guoxia, Trivedi, Dev B., Kavarana, Malcolm J., Hruby, Victor J.

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Role of Hydrophobic Interactions in Binding S-(N-Aryl/Alkyl-N-hydroxy- carbamoyl)glutathiones to the Active Site of the Antitumor Target Enzyme Glyoxalase I by Kalsi, Avinash, Kavarana, Malcolm J, Lu, Tianfen, Whalen, Dale L, Hamilton, Diana S, Creighton, Donald J

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S-(N-Aryl-N-hydroxycarbamoyl)glutathione Derivatives Are Tight-Binding Inhibitors of Glyoxalase I and Slow Substrates for Glyoxalase II by Murthy, Nunna S. R. K, Bakeris, Tina, Kavarana, Malcolm J, Hamilton, Diana S, Lan, Yin, Creighton, Donald J

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A New Method for Rapidly Generating Inhibitors of Glyoxalase I inside Tumor Cells Using S-(N-Aryl-N-hydroxycarbamoyl)ethylsulfoxides by Hamilton, Diana S, Kavarana, Malcolm J, Sharkey, Ellyn M, Eiseman, Julie L, Creighton, Donald J

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Pharmacokinetics and antitumor properties in tumor-bearing mice of an enediol analogue inhibitor of glyoxalase I by SHARKEY, E. M, O'NEILL, H. B, KAVARANA, M. J, HAIBO WANG, CREIGHTON, D. J, SENTZ, D. L, EISEMAN, J. L

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Exploring the Stereostructural Requirements of Peptide Ligands for the Melanocortin Receptors by HRUBY, VICTOR J., CAI, MINYING, GRIECO, PAOLO, HAN, GUOXIA, KAVARANA, MALCOLM, TRIVEDI, DEV

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