Structure-guided design of an Hsp90β N-terminal isoform-selective inhibitor by Khandelwal, Anuj, Kent, Caitlin N., Balch, Maurie, Peng, Shuxia, Mishra, Sanket J., Deng, Junpeng, Day, Victor W., Liu, Weiya, Subramanian, Chitra, Cohen, Mark, Holzbeierlein, Jeffery M., Matts, Robert, Blagg, Brian S. J.

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Structure Based Design of a Grp94-Selective Inhibitor: Exploiting a Key Residue in Grp94 To Optimize Paralog-Selective Binding by Que, Nanette L. S, Crowley, Vincent M, Duerfeldt, Adam S, Zhao, Jinbo, Kent, Caitlin N, Blagg, Brian S. J, Gewirth, Daniel T

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Classics in Chemical Neuroscience: Baclofen by Kent, Caitlin N, Park, Charlotte, Lindsley, Craig W

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Back to the Medicinal Chemistry Future by Giustiniano, Mariateresa, Gruber, Christian W, Kent, Caitlin N, Trippier, Paul C

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The Development of Hsp90β-Selective Inhibitors to Overcome Detriments Associated with pan-Hsp90 Inhibition by Mishra, Sanket J, Liu, Weiya, Beebe, Kristin, Banerjee, Monimoy, Kent, Caitlin N, Munthali, Vitumbiko, Koren, John, Taylor, John A, Neckers, Leonard M, Holzbeierlein, Jeffrey, Blagg, Brian S. J

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Structure‐Based Design, Synthesis, and Biological Evaluation of Hsp90β‐Selective Inhibitors by Chaudhury, Subhabrata, Narasimharao Meka, Penchala, Banerjee, Monimoy, Kent, Caitlin N., Blagg, Brian S. J.

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VU6036720: The First Potent and Selective In Vitro Inhibitor of Heteromeric Kir4.1/5.1 Inward Rectifier Potassium Channels by McClenahan, Samantha J., Kent, Caitlin N., Kharade, Sujay V., Isaeva, Elena, Williams, Jade C., Han, Changho, Terker, Andrew, Gresham III, Robert, Lazarenko, Roman M., Days, Emily L., Romaine, Ian M., Bauer, Joshua A., Boutaud, Olivier, Sulikowski, Gary A., Harris, Raymond, Weaver, C. David, Staruschenko, Alexander, Lindsley, Craig W., Denton, Jerod S.

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Discovery and optimization of a novel CNS penetrant series of mGlu4 PAMs based on a 1,4-thiazepane core with in vivo efficacy in a preclinical Parkinsonian model by Kent, Caitlin N., Fulton, Mark G., Stillwell, Kaylee J., Dickerson, Jonathan W., Loch, Matthew T., Rodriguez, Alice L., Blobaum, Anna L., Boutaud, Olivier, Rook, Jerri L., Niswender, Colleen M., Conn, P. Jeffrey, Lindsley, Craig W.

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Synthesis and Biological Evaluation of Stilbene Analogues as Hsp90 C‐Terminal Inhibitors by Byrd, Katherine M., Kent, Caitlin N., Blagg, Brian S. J.

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Cover Feature: Synthesis and Biological Evaluation of Stilbene Analogues as Hsp90 C‐Terminal Inhibitors (ChemMedChem 24/2017) by Byrd, Katherine M., Kent, Caitlin N., Blagg, Brian S. J.

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Discovery and optimization of a novel CNS penetrant series of mGlu 4 PAMs based on a 1,4-thiazepane core with in vivo efficacy in a preclinical Parkinsonian model by Kent, Caitlin N, Fulton, Mark G, Stillwell, Kaylee J, Dickerson, Jonathan W, Loch, Matthew T, Rodriguez, Alice L, Blobaum, Anna L, Boutaud, Olivier, Rook, Jerri L, Niswender, Colleen M, Conn, P Jeffrey, Lindsley, Craig W

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Comparison of FilmArray and Quantitative Real-Time Reverse Transcriptase PCR for Detection of Zaire Ebolavirus from Contrived and Clinical Specimens by Southern, Timothy R, Racsa, Lori D, Albariño, César G, Fey, Paul D, Hinrichs, Steven H, Murphy, Caitlin N, Herrera, Vicki L, Sambol, Anthony R, Hill, Charles E, Ryan, Emily L, Kraft, Colleen S, Campbell, Shelley, Sealy, Tara K, Schuh, Amy, Ritchie, James C, Lyon, 3rd, G Marshall, Mehta, Aneesh K, Varkey, Jay B, Ribner, Bruce S, Brantly, Kent P, Ströher, Ute, Iwen, Peter C, Burd, Eileen M

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Variation of the aryl substituent on the piperazine ring within the 4-(piperazin-1-yl)-2,6-di(pyrrolidin-1-yl)pyrimidine scaffold unveils potent, non-competitive inhibitors of the... by Kent, Courtney R., Bryja, Magdalena, Gustafson, Helen A., Kawarski, Margaret Y., Lenti, Gena, Pierce, Emily N., Knopp, Rachel C., Ceja, Victor, Pati, Bhabna, Walters, D. Eric, Karver, Caitlin E.

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