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Search Results - Koblet, Andreas
Search Results - Koblet, Andreas
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The discovery and unique pharmacological profile of RO4938581 and RO4882224 as potent and selective GABAA α5 inverse agonists for the treatment of cognitive dysfunction
by
Knust, Henner
,
Achermann, Guido
,
Ballard, Theresa
,
Buettelmann, Bernd
,
Gasser, Rodolfo
,
Fischer, Holger
,
Hernandez, Maria-Clemencia
,
Knoflach, Frédéric
,
Koblet, Andreas
,
Stadler, Heinz
,
Thomas, Andrew W.
,
Trube, Gerhard
,
Waldmeier, Pius
Published in
Bioorganic & medicinal chemistry letters
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Discovery of the imidazo[1,5-α][1,2,4].triazolo[1,5-d][1,4]benzodiazepine scaffold as a novel, potent and selective GABAA α5 inverse agonist series
by
ACHERMANN, Guido
,
BALLARD, Theresa M
,
KOBLET, Andreas
,
KNUST, Henner
,
KURT, Anke
,
MARTIN, James R
,
MASCIADRI, Raffaello
,
PORTER, Richard H. P
,
STADLER, Heinz
,
THOMAS, Andrew W
,
TRUBE, Gerhard
,
WICHMANN, Jürgen
,
BLASCO, Francesca
,
BROUTIN, Pierre-Emmanuel
,
BÜTTELMANN, Bernd
,
FISCHER, Holger
,
GRAF, Martin
,
HERNANDEZ, Maria-Clemencia
,
HILTY, Peter
,
KNOFLACH, Frédéric
Published in
Bioorganic & medicinal chemistry letters
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Identification of Three Novel Radiotracers for Imaging Aggregated Tau in Alzheimer’s Disease with Positron Emission Tomography
by
Gobbi, Luca C
,
Knust, Henner
,
Körner, Matthias
,
Honer, Michael
,
Czech, Christian
,
Belli, Sara
,
Muri, Dieter
,
Edelmann, Martin R
,
Hartung, Thomas
,
Erbsmehl, Isabella
,
Grall-Ulsemer, Sandra
,
Koblet, Andreas
,
Rueher, Marianne
,
Steiner, Sandra
,
Ravert, Hayden T
,
Mathews, William B
,
Holt, Daniel P
,
Kuwabara, Hiroto
,
Valentine, Heather
,
Dannals, Robert F
,
Wong, Dean F
,
Borroni, Edilio
Published in
Journal of medicinal chemistry
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Discovery of potent, balanced and orally active dual NK1/NK3 receptor ligands
by
Peters, Jens-Uwe
,
Hoffmann, Torsten
,
Schnider, Patrick
,
Stadler, Heinz
,
Koblet, Andreas
,
Alker, André
,
Poli, Sonia Maria
,
Ballard, Theresa M.
,
Spooren, Will
,
Steward, Lucinda
,
Sleight, Andrew J.
Published in
Bioorganic & medicinal chemistry letters
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Discovery of potent, balanced and orally active dual NK sub(1)/NK sub(3) receptor ligands
by
Peters, Jens-Uwe
,
Hoffmann, Torsten
,
Schnider, Patrick
,
Stadler, Heinz
,
Koblet, Andreas
,
Alker, Andre
,
Poli, Sonia Maria
,
Ballard, Theresa M
,
Spooren, Will
,
Steward, Lucinda
,
Sleight, Andrew J
Published in
Bioorganic & medicinal chemistry letters
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The discovery and unique pharmacological profile of RO4938581 and RO4882224 as potent and selective GABA sub(A) alpha 5 inverse agonists for the treatment of cognitive dysfunction
by
Knust, Henner
,
Achermann, Guido
,
Ballard, Theresa
,
Buettelmann, Bernd
,
Gasser, Rodolfo
,
Fischer, Holger
,
Hernandez, Maria-Clemencia
,
Knoflach, Frederic
,
Koblet, Andreas
,
Stadler, Heinz
,
Thomas, Andrew W
,
Trube, Gerhard
,
Waldmeier, Pius
Published in
Bioorganic & medicinal chemistry letters
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7
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The discovery and unique pharmacological profile of RO4938581 and RO4882224 as potent and selective GABA A α5 inverse agonists for the treatment of cognitive dysfunction
by
Knust, Henner
,
Achermann, Guido
,
Ballard, Theresa
,
Buettelmann, Bernd
,
Gasser, Rodolfo
,
Fischer, Holger
,
Hernandez, Maria-Clemencia
,
Knoflach, Frédéric
,
Koblet, Andreas
,
Stadler, Heinz
,
Thomas, Andrew W.
,
Trube, Gerhard
,
Waldmeier, Pius
Published in
Bioorganic & medicinal chemistry letters
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8
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The discovery and unique pharmacological profile of RO4938581 and R04882224 as potent and selective GABAA α5 inverse agonists for the treatment of cognitive dysfunction
by
KNUST, Henner
,
ACHERMANN, Guido
,
THOMAS, Andrew W
,
TRUBE, Gerhard
,
WALDMEIER, Pius
,
BALLARD, Theresa
,
BUETTELMANN, Bernd
,
GASSER, Rodolfo
,
FISCHER, Holger
,
HERNANDEZ, Maria-Clemencia
,
KNOFLACH, Frédéric
,
KOBLET, Andreas
,
STADLER, Heinz
Published in
Bioorganic & medicinal chemistry letters
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9
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Discovery of the imidazo[1,5-a][1,2,4]-triazolo[1,5-d][1,4]benzodiazepine scaffold as a novel, potent and selective GABA sub(A) alpha 5 inverse agonist series
by
Achermann, Guido
,
Ballard, Theresa M
,
Blasco, Francesca
,
Broutin, Pierre-Emmanuel
,
Buettelmann, Bernd
,
Fischer, Holger
,
Graf, Martin
,
Hernandez, Maria-Clemencia
,
Hilty, Peter
,
Knoflach, Frederic
,
Koblet, Andreas
,
Knust, Henner
,
Kurt, Anke
,
Martin, James R
,
Masciadri, Raffaello
,
Porter, Richard HP
,
Stadler, Heinz
,
Thomas, Andrew W
,
Trube, Gerhard
,
Wichmann, Juergen
Published in
Bioorganic & medicinal chemistry letters
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Article
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10
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Discovery of the imidazo[1,5- a][1,2,4]-triazolo[1,5- d][1,4]benzodiazepine scaffold as a novel, potent and selective GABA A α5 inverse agonist series
by
Achermann, Guido
,
Ballard, Theresa M.
,
Blasco, Francesca
,
Broutin, Pierre-Emmanuel
,
Büttelmann, Bernd
,
Fischer, Holger
,
Graf, Martin
,
Hernandez, Maria-Clemencia
,
Hilty, Peter
,
Knoflach, Frédéric
,
Koblet, Andreas
,
Knust, Henner
,
Kurt, Anke
,
Martin, James R.
,
Masciadri, Raffaello
,
Porter, Richard H.P.
,
Stadler, Heinz
,
Thomas, Andrew W.
,
Trube, Gerhard
,
Wichmann, Jürgen
Published in
Bioorganic & medicinal chemistry letters
Get full text
Article
Save to List
Saved in:
11
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The discovery and unique pharmacological profile of RO4938581 and RO4882224 as potent and selective GABAA alpha5 inverse agonists for the treatment of cognitive dysfunction
by
Knust, Henner
,
Achermann, Guido
,
Ballard, Theresa
,
Buettelmann, Bernd
,
Gasser, Rodolfo
,
Fischer, Holger
,
Hernandez, Maria-Clemencia
,
Knoflach, Frédéric
,
Koblet, Andreas
,
Stadler, Heinz
,
Thomas, Andrew W
,
Trube, Gerhard
,
Waldmeier, Pius
Published in
Bioorganic & medicinal chemistry letters
Get full text
Article
Save to List
Saved in:
12
Loading…
Discovery of the imidazo[1,5-a][1,2,4]-triazolo[1,5-d][1,4]benzodiazepine scaffold as a novel, potent and selective GABA(A) alpha5 inverse agonist series
by
Achermann, Guido
,
Ballard, Theresa M
,
Blasco, Francesca
,
Broutin, Pierre-Emmanuel
,
Büttelmann, Bernd
,
Fischer, Holger
,
Graf, Martin
,
Hernandez, Maria-Clemencia
,
Hilty, Peter
,
Knoflach, Frédéric
,
Koblet, Andreas
,
Knust, Henner
,
Kurt, Anke
,
Martin, James R
,
Masciadri, Raffaello
,
Porter, Richard H P
,
Stadler, Heinz
,
Thomas, Andrew W
,
Trube, Gerhard
,
Wichmann, Jürgen
Published in
Bioorganic & medicinal chemistry letters
Get full text
Article
Save to List
Saved in:
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