(2R)-4-Oxo-4-[3-(Trifluoromethyl)-5,6-dihydro[1,2,4]triazolo[4,3-a]pyrazin- 7(8H)-yl]-1-(2,4,5-trifluorophenyl)butan-2-amine:  A Potent, Orally Active Dipeptidyl Peptidase IV Inhib... by Kim, Dooseop, Wang, Liping, Beconi, Maria, Eiermann, George J, Fisher, Michael H, He, Huaibing, Hickey, Gerard J, Kowalchick, Jennifer E, Leiting, Barbara, Lyons, Kathryn, Marsilio, Frank, McCann, Margaret E, Patel, Reshma A, Petrov, Aleksandr, Scapin, Giovanna, Patel, Sangita B, Roy, Ranabir Sinha, Wu, Joseph K, Wyvratt, Matthew J, Zhang, Bei B, Zhu, Lan, Thornberry, Nancy A, Weber, Ann E

Get full text

Discovery of Potent and Selective Dipeptidyl Peptidase IV Inhibitors Derived from β-Aminoamides Bearing Subsituted Triazolopiperazines by Kim, Dooseop, Kowalchick, Jennifer E, Brockunier, Linda L, Parmee, Emma R, Eiermann, George J, Fisher, Michael H, He, Huaibing, Leiting, Barbara, Lyons, Kathryn, Scapin, Giovanna, Patel, Sangita B, Petrov, Aleksandr, Pryor, KellyAnn D, Roy, Ranabir Sinha, Wu, Joseph K, Zhang, Xiaoping, Wyvratt, Matthew J, Zhang, Bei B, Zhu, Lan, Thornberry, Nancy A, Weber, Ann E

Get full text

Triazolopiperazine-amides as dipeptidyl peptidase IV inhibitors: Close analogs of JANUVIA™ (sitagliptin phosphate) by Kim, Dooseop, Kowalchick, Jennifer E., Edmondson, Scott D., Mastracchio, Anthony, Xu, Jinyou, Eiermann, George J., Leiting, Barbara, Wu, Joseph K., Pryor, KellyAnn D., Patel, Reshma A., He, Huaibing, Lyons, Kathryn A., Thornberry, Nancy A., Weber, Ann E.

Get full text

Design, synthesis, and biological evaluation of triazolopiperazine-based β-amino amides as potent, orally active dipeptidyl peptidase IV (DPP-4) inhibitors by Kowalchick, Jennifer E., Leiting, Barbara, Pryor, KellyAnn D., Marsilio, Frank, Wu, Joseph K., He, Huaibing, Lyons, Kathryn A., Eiermann, George J., Petrov, Aleksandr, Scapin, Giovanna, Patel, Reshma A., Thornberry, Nancy A., Weber, Ann E., Kim, Dooseop

Get full text

Cyclization of unsaturated amides with triflic anhydride and samarium diiodide by McDonald, Chriss E, Galka, Amy M, Green, Ahren I, Keane, Joseph M, Kowalchick, Jennifer E, Micklitsch, Christopher M, Wisnoski, David D

Get full text

2-Arylbenzoxazoles as CETP inhibitors: Raising HDL-C in cynoCETP transgenic mice by Kallashi, Florida, Kim, Dooseop, Kowalchick, Jennifer, Park, You Jung, Hunt, Julianne A., Ali, Amjad, Smith, Cameron J., Hammond, Milton L., Pivnichny, James V., Tong, Xinchun, Xu, Suoyu S., Anderson, Matt S., Chen, Ying, Eveland, Suzanne S., Guo, Qiu, Hyland, Sheryl A., Milot, Denise P., Cumiskey, Anne-Marie, Latham, Melanie, Peterson, Laurence B., Rosa, Raymond, Sparrow, Carl P., Wright, Samuel D., Sinclair, Peter J.

Get full text

(2R)-4-Oxo-4[3-(Trifluoromethyl)-5,6-diihydro:1,2,4}triazolo[4,3-a}pyrazin-7(8H)-y1]-1-(2,4,5-trifluorophenyl)butan-2-amine: A Potent, Orally Active Dipeptidyl Peptidase IV Inhibit... by Kim, D., Wang, L., Beconi, M., Eiermann, G., Fisher, M., He, H., Hickey, G., Kowalchick, Jennifer, Leiting, Barbara, Lyons, K., Marsilio, F., McCann, F., Patel, R., Petrov, A., Scapin, G., Patel, S., Roy, R., Wu, J., Wyvratt, M., Zhang, B., Zhu, L., Thornberry, N., Weber, A.

Get full text

Discovery of Potent and Selective Dipeptidyl Peptidase IV Inhibitors Derived from [beta]-Aminoamides Bearing Subsituted Triazolopiperazines by Kim, Dooseop, Kowalchick, Jennifer E., Brockunier, Linda L., Parmee, Emma R., Eiermann, George J., Fisher, Michael H., He, Huaibing, Leiting, Barbara, Lyons, Kathryn, Scapin, Giovanna, Patel, Sangita B., Petrov, Aleksandr, Pryor, KellyAnn D., Roy, Ranabir Sinha, Wu, Joseph K., Zhang, Xiaoping, Wyvratt, Matthew J., Zhang, Bei B., Zhu, Lan, Thornberry, Nancy A., Weber, Ann E.

Get full text

Discovery of Potent and Selective Dipeptidyl Peptidase IV Inhibitors Derived from β-Aminoaimdes Bearing Subsituted Triazolopiperazines by KIM, Dooseop, KOWALCHICK, Jennifer E, PATEL, Sangita B, PETROV, Aleksandr, PRYOR, Kellyann D, ROY, Ranabir Sinha, WU, Joseph K, XIAOPING ZHANG, WYVRATT, Matthew J, ZHANG, Bei B, LAN ZHU, THOMBERRY, Nancy A, BROCKUNIER, Linda L, WEBER, Ann E, PARMEE, Emma R, EIERMANN, George J, FISHER, Michael H, HUAIBING HE, LEITING, Barbara, LYONS, Kathryn, SCAPIN, Giovanna

Get full text

Design, synthesis, and biological evaluation of triazolopiperazine-based SS-amino amides as potent, orally active dipeptidyl peptidase IV (DPP-4) inhibitors by KOWALCHICK, Jennifer E, LEITING, Barbara, PATEL, Reshma A, THORNBERRY, Nancy A, WEBER, Ann E, KIM, Dooseop, PRYOR, Kellyann D, MARSILIO, Frank, WU, Joseph K, HUAIBING HE, LYONS, Kathryn A, EIERMANN, George J, PETROV, Aleksandr, SCAPIN, Giovanna

Get full text