Lead optimization of 2-hydroxymethyl imidazoles as non-hydroxamate LpxC inhibitors: Discovery of TP0586532 by Ushiyama, Fumihito, Takashima, Hajime, Matsuda, Yohei, Ogata, Yuya, Sasamoto, Naoki, Kurimoto-Tsuruta, Risa, Ueki, Kaori, Tanaka-Yamamoto, Nozomi, Endo, Mayumi, Mima, Masashi, Fujita, Kiyoko, Takata, Iichiro, Tsuji, Satoshi, Yamashita, Haruhiro, Okumura, Hirotoshi, Otake, Katsumasa, Sugiyama, Hiroyuki

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Fragment-Based Discovery of Novel Non-Hydroxamate LpxC Inhibitors with Antibacterial Activity by Yamada, Yousuke, Takashima, Hajime, Walmsley, David Lee, Ushiyama, Fumihito, Matsuda, Yohei, Kanazawa, Harumi, Yamaguchi-Sasaki, Toru, Tanaka-Yamamoto, Nozomi, Yamagishi, Junya, Kurimoto-Tsuruta, Risa, Ogata, Yuya, Ohtake, Norikazu, Angove, Hayley, Baker, Lisa, Harris, Richard, Macias, Alba, Robertson, Alan, Surgenor, Allan, Watanabe, Hayato, Nakano, Koichiro, Mima, Masashi, Iwamoto, Kunihiko, Okada, Atsushi, Takata, Iichiro, Hitaka, Kosuke, Tanaka, Akihiro, Fujita, Kiyoko, Sugiyama, Hiroyuki, Hubbard, Roderick E

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Discovery of a potent dual inhibitor of wild-type and mutant respiratory syncytial virus fusion proteins through the modulation of atropisomer interconversion properties by Yamaguchi-Sasaki, Toru, Kawaguchi, Takanori, Okada, Atsushi, Tokura, Seiken, Tanaka-Yamamoto, Nozomi, Takeuchi, Tomoki, Ogata, Yuya, Takahashi, Ryo, Kurimoto-Tsuruta, Risa, Tamaoki, Tomokazu, Sugaya, Yutaka, Abe-Kumasaka, Tomoko, Arikawa, Kaho, Yoshida, Ippei, Sugiyama, Hiroyuki, Kanuma, Kosuke, Yoshinaga, Mitsukane

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