Synthesis and Biological Evaluation of Novel Analogues of the Pan Class I Phosphatidylinositol 3-Kinase (PI3K) Inhibitor 2-(Difluoromethyl)-1-[4,6-di(4-morpholinyl)-1,3,5-triazin-2... by Rewcastle, Gordon W, Gamage, Swarna A, Flanagan, Jack U, Frederick, Raphael, Denny, William A, Baguley, Bruce C, Kestell, Philip, Singh, Ripudaman, Kendall, Jackie D, Marshall, Elaine S, Lill, Claire L, Lee, Woo-Jeong, Kolekar, Sharada, Buchanan, Christina M, Jamieson, Stephen M. F, Shepherd, Peter R

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Novel pyrazolo[1,5-a]pyridines with improved aqueous solubility as p110α-selective PI3 kinase inhibitors by Kendall, Jackie D., Giddens, Anna C., Tsang, Kit Yee, Marshall, Elaine S., Lill, Claire L., Lee, Woo-Jeong, Kolekar, Sharada, Chao, Mindy, Malik, Alisha, Yu, Shuqiao, Chaussade, Claire, Buchanan, Christina, Jamieson, Stephen M.F., Rewcastle, Gordon W., Baguley, Bruce C., Denny, William A., Shepherd, Peter R.

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Exploring the isoform selectivity of TGX-221 related pyrido[1,2-a]pyrimidinone-based Class IA PI 3-kinase inhibitors: Synthesis, biological evaluation and molecular modelling by Marshall, Andrew J., Lill, Claire L., Chao, Mindy, Kolekar, Sharada V., Lee, Woo-Jeong, Marshall, Elaine S., Baguley, Bruce C., Shepherd, Peter R., Denny, William A., Flanagan, Jack U., Rewcastle, Gordon W.

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Discovery of pyrazolo[1,5-a]pyridines as p110α-selective PI3 kinase inhibitors by Kendall, Jackie D., O’Connor, Patrick D., Marshall, Andrew J., Frédérick, Raphaël, Marshall, Elaine S., Lill, Claire L., Lee, Woo-Jeong, Kolekar, Sharada, Chao, Mindy, Malik, Alisha, Yu, Shuqiao, Chaussade, Claire, Buchanan, Christina, Rewcastle, Gordon W., Baguley, Bruce C., Flanagan, Jack U., Jamieson, Stephen M.F., Denny, William A., Shepherd, Peter R.

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Novel pyrazolo[1,5-a]pyridines as p110α-selective PI3 kinase inhibitors: Exploring the benzenesulfonohydrazide SAR by Kendall, Jackie D., Giddens, Anna C., Tsang, Kit Yee, Frédérick, Raphaël, Marshall, Elaine S., Singh, Ripudaman, Lill, Claire L., Lee, Woo-Jeong, Kolekar, Sharada, Chao, Mindy, Malik, Alisha, Yu, Shuqiao, Chaussade, Claire, Buchanan, Christina, Rewcastle, Gordon W., Baguley, Bruce C., Flanagan, Jack U., Jamieson, Stephen M.F., Denny, William A., Shepherd, Peter R.

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Synthesis and biological evaluation of novel phosphatidylinositol 3-kinase inhibitors: Solubilized 4-substituted benzimidazole analogs of 2-(difluoromethyl)-1-[4,6-di(4-morpholinyl... by Rewcastle, Gordon W., Gamage, Swarna A., Flanagan, Jack U., Kendall, Jackie D., Denny, William A., Baguley, Bruce C., Buchanan, Christina M., Chao, Mindy, Kestell, Philip, Kolekar, Sharada, Lee, Woo-Jeong, Lill, Claire L., Malik, Alisha, Singh, Ripudaman, Jamieson, Stephen M.F., Shepherd, Peter R.

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Synthesis and Biological Evaluation of Novel Analogues of the Pan Class I Phosphatidylinositol 3-Kinase (PI3K) Inhibitor 2-(Difluoromethyl)-1-[4,6-di(4-morpholinyl)-1,3,5-triazin-2... by Rewcastle, Gordon W., Gamage, Swarna A., Flanagan, Jack U., Frederick, Raphael, Denny, William A., Baguley, Bruce C., Kestell, Philip, Singh, Ripudaman, Kendall, Jackie D., Marshall, Elaine S., Lill, Claire L., Lee, Woo-Jeong, Kolekar, Sharada, Buchanan, Christina M., Jamieson, Stephen M. F., Shepherd, Peter R.

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Novel pyrazolo[1,5-a]pyridines as PI3K inhibitors: variation of the central linker group by Kendall, Jackie D., Marshall, Andrew J., Giddens, Anna C., Tsang, Kit Yee, Boyd, Maruta, Frédérick, Raphaël, Lill, Claire L., Lee, Woo-Jeong, Kolekar, Sharada, Chao, Mindy, Malik, Alisha, Yu, Shuqiao, Chaussade, Claire, Buchanan, Christina M., Rewcastle, Gordon W., Baguley, Bruce C., Flanagan, Jack U., Denny, William A., Shepherd, Peter R.

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Discovery of pyrazolo[1,5-a]pyridines as p110I+/--selective PI3 kinase inhibitors by Kendall, Jackie D, O'Connor, Patrick D, Marshall, Andrew J, Frederick, Raphaeel, Marshall, Elaine S, Lill, Claire L, Lee, Woo-Jeong, Kolekar, Sharada, Chao, Mindy, Malik, Alisha, Yu, Shuqiao, Chaussade, Claire, Buchanan, Christina, Rewcastle, Gordon W, Baguley, Bruce C, Flanagan, Jack U, Jamieson, Stephen MF, Denny, William A, Shepherd, Peter R

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Novel pyrazolo[1,5-a]pyridines as p110I+/--selective PI3 kinase inhibitors: Exploring the benzenesulfonohydrazide SAR by Kendall, Jackie D, Giddens, Anna C, Tsang, Kit Yee, Frederick, Raphaeel, Marshall, Elaine S, Singh, Ripudaman, Lill, Claire L, Lee, Woo-Jeong, Kolekar, Sharada, Chao, Mindy, Malik, Alisha, Yu, Shuqiao, Chaussade, Claire, Buchanan, Christina, Rewcastle, Gordon W, Baguley, Bruce C, Flanagan, Jack U, Jamieson, Stephen MF, Denny, William A, Shepherd, Peter R

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Novel pyrazolo[1,5-a]pyridines as PI3K inhibitors: variation of the central linker groupElectronic supplementary information (ESI) available. See DOI: 10.1039/c3md00221g by Kendall, Jackie D, Marshall, Andrew J, Giddens, Anna C, Tsang, Kit Yee, Boyd, Maruta, Frédérick, Raphaël, Lill, Claire L, Lee, Woo-Jeong, Kolekar, Sharada, Chao, Mindy, Malik, Alisha, Yu, Shuqiao, Chaussade, Claire, Buchanan, Christina M, Rewcastle, Gordon W, Baguley, Bruce C, Flanagan, Jack U, Denny, William A, Shepherd, Peter R

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Global changes in DNA methylation and hydroxymethylation in Alzheimer's disease human brain by Coppieters, Natacha, Dieriks, Birger V, Lill, Claire, Faull, Richard L.M, Curtis, Maurice A, Dragunow, Mike

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Effects of race and ethnicity on perinatal outcomes in high-income and upper-middle-income countries: an individual participant data meta-analysis of 2 198 655 pregnancies by Allotey, John, Kew, Tania, Fernández-Félix, Borja M, Thangaratinam, Shakila, Abdollahain, Mali, Savitri, Ary I., Salvesen, Kjell Åsmund, Bhattacharya, Sohinee, Olive, Elisa Llurba, Daskalakis, George, Macleod, Maureen, Thilaganathan, Baskaran, Ramírez, Javier Arenas, Massé, Jacques, Magnus, Per Minor, Sletner, Line, Baschat, Ahmet, Ohkuchi, Akihide, McAuliffe, Fionnuala M., West, Jane, Farrar, Diane, Riddell, Catherine, van de Post, Joris, Illanes, Sebastián E., Holzman, Claudia, van Kuijk, Sander M.J., Carbillon, Lionel, Villa, Pia M., Eskild, Anne, Chappell, Lucy, Prefumo, Federico, Seed, Paul, van Oostwaard, Miriam, Verlohren, Stefan, Poston, Lucilla, Ferrazzi, Enrico, Vinter, Christina A., Nagata, Chie, Brown, Mark, Vollebregt, Karlijn C., Takeda, Satoru, Langenveld, Josje, Widmer, Mariana, Haavaldsen, Camilla, Olsen, Jørn, Wolf, Hans, Zavaleta, Nelly, Lumbiganon, Pisake, Sequeira, Evan, Gibson, Robert, Ferrazzani, Sergio, Frusca, Tiziana, Figueiró-Filho, Ernesto A., Lapaire, Olav, Laivuori, Hannele, Conde-Agudelo, Agustin, Galindo, Alberto, Mbah, Alfred, Herraiz, Ignacio, Trogstad, Lill, Steegers, Eric A.P., Salim, Read, Huang, Tianhua, Adank, Annemarijne, Meschino, Wendy S., Browne, Joyce L., Da Silva Costa, Fabricio, Jørgensen, Jan Stener, Forest, Jean-Claude, Rumbold, Alice R., Mol, Ben W., Giguère, Yves, Ganzevoort, Wessel, Odibo, Anthony O., Myers, Jenny, Teede, Helena J., Goffinet, Francois, McCowan, Lesley, Pajkrt, Eva, Dekker, Gustaaf, Kleinrouweler, Emily C., Roberts, Claire T., Groen, Henk, Skråstad, Ragnhild Bergene, Heinonen, Seppo, Eero, Kajantie, Kenny, Louise C., Souka, Athena, Monterio, Ilza, Coomarasamy, Arri, Smuk, Melanie, Pillalis, Athanasios, Crovetto, Francesca, Ann Hawkins, Lee, Gabbay- Benziv, Rinat, Riley, Richard, Snell, Kym, Archer, Lucinda, Figuera, Francesc, van Gelder, Marleen

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Applications of crystal structure prediction - organic molecular structures: general discussion by Adjiman, Claire S, Brandenburg, Jan Gerit, Braun, Doris E, Cole, Jason, Collins, Christopher, Cooper, Andrew I, Cruz-Cabeza, Aurora J, Day, Graeme M, Dudek, Marta, Hare, Alan, Iuzzolino, Luca, McKay, David, Mitchell, John B. O, Mohamed, Sharmarke, Neelamraju, Sridhar, Neumann, Marcus, Nilsson Lill, Sten, Nyman, Jonas, Oganov, Artem R, Price, Sarah L, Pulido, Angeles, Reutzel-Edens, Susan, Rietveld, Ivo, Ruggiero, Michael T, Schön, J. Christian, Tsuzuki, Seiji, van den Ende, Joost, Woollam, Grahame, Zhu, Qiang

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Structure searching methods: general discussion by Addicoat, Matthew, Adjiman, Claire S, Arhangelskis, Mihails, Beran, Gregory J. O, Brandenburg, Jan Gerit, Braun, Doris E, Burger, Virginia, Burow, Asbjoern, Collins, Christopher, Cooper, Andrew, Day, Graeme M, Deringer, Volker L, Dyer, Matthew S, Hare, Alan, Jelfs, Kim E, Keupp, Julian, Konstantinopoulos, Stefanos, Li, Yi, Ma, Yanming, Marom, Noa, McKay, David, Mellot-Draznieks, Caroline, Mohamed, Sharmarke, Neumann, Marcus, Nilsson Lill, Sten, Nyman, Jonas, Oganov, Artem R, Price, Sarah L, Reutzel-Edens, Susan, Ruggiero, Michael, Sastre, German, Schmid, Rochus, Schmidt, Julia, Schön, J. Christian, Spackman, Peter, Tsuzuki, Seiji, Woodley, Scott M, Yang, Shiyue, Zhu, Qiang

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Assessing fibrinogen extravasation into Alzheimer's disease brain using high-content screening of brain tissue microarrays by Narayan, Pritika J., Kim, Sue-Ling, Lill, Claire, Feng, Sheryl, Faull, Richard L.M., Curtis, Maurice A., Dragunow, Michael

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Crystal structure evaluation: calculating relative stabilities and other criteria: general discussion by Addicoat, Matthew, Adjiman, Claire S, Arhangelskis, Mihails, Beran, Gregory J. O, Bowskill, David, Brandenburg, Jan Gerit, Braun, Doris E, Burger, Virginia, Cole, Jason, Cruz-Cabeza, Aurora J, Day, Graeme M, Deringer, Volker L, Guo, Rui, Hare, Alan, Helfferich, Julian, Hoja, Johannes, Iuzzolino, Luca, Jobbins, Samuel, Marom, Noa, McKay, David, Mitchell, John B. O, Mohamed, Sharmarke, Neumann, Marcus, Nilsson Lill, Sten, Nyman, Jonas, Oganov, Artem R, Piaggi, Pablo, Price, Sarah L, Reutzel-Edens, Susan, Rietveld, Ivo, Ruggiero, Michael, Ryder, Matthew R, Sastre, German, Schön, J. Christian, Taylor, Christopher, Tkatchenko, Alexandre, Tsuzuki, Seiji, van den Ende, Joost, Woodley, Scott M, Woollam, Grahame, Zhu, Qiang

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