Discovery of the Irreversible Covalent FGFR Inhibitor 8‑(3-(4-Acryloyl­piperazin-1-yl)propyl)-6-(2,6-dichloro-3,5-dimethoxyphenyl)-2-(methylamino)­pyrido[2,3‑d]­pyrimidin-7(8H)‑one... by Brameld, Ken A, Owens, Timothy D, Verner, Erik, Venetsanakos, Eleni, Bradshaw, J. Michael, Phan, Vernon T, Tam, Danny, Leung, Kwan, Shu, Jin, LaStant, Jacob, Loughhead, David G, Ton, Tony, Karr, Dane E, Gerritsen, Mary E, Goldstein, David M, Funk, Jens Oliver

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Novel hexahydropyrrolo[3,4- c]pyrrole CCR5 antagonists by Rotstein, David M., Melville, Chris R., Padilla, Fernando, Cournoyer, Dick, Lee, Eun K., Lemoine, Remy, Petersen, Ann C., Setti, Lina Q., Wanner, Jutta, Chen, Lijing, Filonova, Lubov, Loughhead, David G., Manka, Jason, Lin, Xiao-Fa, Gleason, Shelley, Sankuratri, Surya, Ji, Changhua, deRosier, Andre, Dioszegi, Marianna, Heilek, Gabrielle, Jekle, Andreas, Berry, Pamela, Mau, Cheng-I, Weller, Paul

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Asymmetric Synthesis and Stereochemical Assignment of RS-97613, a Potent Immunosuppressive and Antiinflammatory Agent by Smith, David B, Waltos, Ann Marie, Loughhead, David G, Weikert, Robert J, Morgans, David J, Rohloff, John C, Link, John O, Zhu, Rong-rong

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Structures and Total Synthesis of 2-Aminoimidazoles from a Notodoris Nudibranch by Alvi, K. A, Crews, Phillip, Loughhead, David G

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Synthesis of des-N-methylacronycine and acronycine by Loughhead, David G

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Synthesis of Mexiletine Stereoisomers and Related Compounds via SNAr Nucleophilic Substitution of a Cr(CO)3-Complexed Aromatic Fluoride by Loughhead, David G, Flippin, Lee A, Weikert, Robert J

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2,2-Dimethylcyclopropyl-benzamides: Novel positive allosteric modulators of α7 nAChRs by Maag, Hans, Bois, Daisy Joe Du, Loughhead, David G., Manka, Jason, Misner, Dinah, Sahdeo, Sunil, Smith, David B.

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Synthesis and anthelmintic activity of 3'-benzoylurea derivatives of 6-phenyl-2,3,5,6-tetrahydroimidazo[2,1-b]thiazole by Weikert, Robert J, Bingham, Stanford, Emanuel, Mark A, Fraser-Smith, Elizabeth B, Loughhead, David G, Nelson, Peter H, Poulton, Anthony L

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Preparation and acid-catalyzed rearrangement of a carbon-17 isopropylidene and a carbon-17 isopropenyl sterol by Loughhead, David G

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Synthesis of Mexiletine Stereoisomers and Related Compounds via S(N)Ar Nucleophilic Substitution of a Cr(CO)(3)-Complexed Aromatic Fluoride by Loughhead, David G., Flippin, Lee A., Weikert, Robert J.

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Structure−Activity Relationships for Inhibition of Inosine Monophosphate Dehydrogenase by Nuclear Variants of Mycophenolic Acid by Nelson, Peter H, Carr, Stephen F, Devens, Bruce H, Eugui, Elsie M, Franco, Fidencio, Gonzalez, Carlos, Hawley, Ronald C, Loughhead, David G, Milan, David J, Papp, Eva, Patterson, John W, Rouhafza, Sussan, Sjogren, Eric B, Smith, David B, Stephenson, Rebecca A, Talamas, Francisco X, Waltos, Ann-Marie, Weikert, Robert J, Wu, John C

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Synthesis of Mexiletine Stereoisomers and Related Compounds via S N Ar Nucleophilic Substitution of a Cr(CO) 3 -Complexed Aromatic Fluoride by Loughhead, David G., Flippin, Lee A., Weikert, Robert J.

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The Florisil ® catalyzed [1,3]-sigmatropic shift of allyl phenyl ethers — An entryway into novel mycophenolic acid analogues by Talamás, Francisco X., Smith, David B., Cervantes, Alicia, Franco, Fidencio, Cutler, Serena T., Loughhead, David G., Morgans, David J., Weikert, Robert J.

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Preparation and acid-catalyzed rearrangement of C-17 isopropylidene and a C-17 isopropenyl sterol by LOUGHHEAD, D. G

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