Design, Synthesis, and Structure−Activity Relationship of Indole-3-glyoxylamide Libraries Possessing Highly Potent Activity in a Cell Line Model of Prion Disease by Thompson, Mark J, Borsenberger, Vinciane, Louth, Jennifer C, Judd, Katie E, Chen, Beining

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Improved 2,4-Diarylthiazole-Based Antiprion Agents: Switching the Sense of the Amide Group at C5 Leads to an Increase in Potency by Thompson, Mark J., Louth, Jennifer C., Greenwood, Gemma K., Sorrell, Fiona J., Knight, Sandra G., Adams, Nathan B. P., Chen, Beining

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Amyloid binding and beyond: a new approach for Alzheimer's disease drug discovery targeting Aβo-PrP binding and downstream pathways by Grayson, James D, Baumgartner, Matthew P, Santos Souza, Cleide Dos, Dawes, Samuel J, El Idrissi, Imane Ghafir, Louth, Jennifer C, Stimpson, Sasha, Mead, Emma, Dunbar, Charlotte, Wolak, Joanna, Sharman, Gary, Evans, David, Zhuravleva, Anastasia, Roldan, Margarita Segovia, Colabufo, Nicola Antonio, Ning, Ke, Garwood, Claire, Thomas, James A, Partridge, Benjamin M, de la Vega de Leon, Antonio, Gillet, Valerie J, Rauter, Amélia P, Chen, Beining

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Amyloid binding and beyond: a new approach for Alzheimer's disease drug discovery targeting Aβo-PrP C binding and downstream pathways by Grayson, James D, Baumgartner, Matthew P, Santos Souza, Cleide Dos, Dawes, Samuel J, El Idrissi, Imane Ghafir, Louth, Jennifer C, Stimpson, Sasha, Mead, Emma, Dunbar, Charlotte, Wolak, Joanna, Sharman, Gary, Evans, David, Zhuravleva, Anastasia, Roldan, Margarita Segovia, Colabufo, Nicola Antonio, Ning, Ke, Garwood, Claire, Thomas, James A, Partridge, Benjamin M, de la Vega de Leon, Antonio, Gillet, Valerie J, Rauter, Amélia P, Chen, Beining

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Amyloid binding and beyond: a new approach for Alzheimer's disease drug discovery targeting Aβo–PrPC binding and downstream pathways by Grayson, James D, Baumgartner, Matthew P, Cleide Dos Santos Souza, Dawes, Samuel J, Imane Ghafir El Idrissi, Louth, Jennifer C, Stimpson, Sasha, Mead, Emma, Dunbar, Charlotte, Wolak, Joanna, Sharman, Gary, Evans, David, Zhuravleva, Anastasia, Segovia Roldan, Margarita, Colabufo, Nicola Antonio, Ke Ning, Garwood, Claire, Thomas, James A, Partridge, Benjamin M, Antonio de la Vega de Leon, Gillet, Valerie J, Rauter, Amélia P, Chen, Beining

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Synthesis and Evaluation of 1-Amino-6-halo-β-carbolines as Antimalarial and Antiprion Agents by Thompson, Mark J., Louth, Jennifer C., Little, Susan M., Jackson, Matthew P., Boursereau, Yohan, Chen, Beining, Coldham, Iain

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Discovery of 6-substituted indole-3-glyoxylamides as lead antiprion agents with enhanced cell line activity, improved microsomal stability and low toxicity by Thompson, Mark J., Louth, Jennifer C., Ferrara, Steven, Jackson, Matthew P., Sorrell, Fiona J., Cochrane, Edward J., Gever, Joel, Baxendale, Sarah, Silber, B. Michael, Roehl, Henry H., Chen, Beining

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2,4-Diarylthiazole antiprion compounds as a novel structural class of antimalarial leads by Thompson, Mark J., Louth, Jennifer C., Little, Susan M., Chen, Beining, Coldham, Iain

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Structure-Activity Relationship Refinement and Further Assessment of Indole-3-glyoxylamides as a Lead Series against Prion Disease by Thompson, Mark J., Louth, Jennifer C., Ferrara, Steven, Sorrell, Fiona J., Irving, Benjamin J., Cochrane, Edward J., Meijer, Anthony J. H. M., Chen, Beining

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Synthesis and Evaluation of 1-Amino-6-halo-[beta]-carbolines as Antimalarial and Antiprion Agents by Thompson, Mark J, Louth, Jennifer C, Little, Susan M, Jackson, Matthew P, Boursereau, Yohan, Chen, Beining, Coldham, Iain

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Inside Cover: Improved 2,4-Diarylthiazole-Based Antiprion Agents: Switching the Sense of the Amide Group at C5 Leads to an Increase in Potency (ChemMedChem 9/2010) by Thompson, Mark J., Louth, Jennifer C., Greenwood, Gemma K., Sorrell, Fiona J., Knight, Sandra G., Adams, Nathan B. P., Chen, Beining

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