Design and synthesis of morpholine derivatives. SAR for dual serotonin & noradrenaline reuptake inhibition by Fish, Paul V., Deur, Christopher, Gan, Xinmin, Greene, Keri, Hoople, David, Mackenny, Malcolm, Para, Kimberly S., Reeves, Keith, Ryckmans, Thomas, Stiff, Cory, Stobie, Alan, Wakenhut, Florian, Whitlock, Gavin A.

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Synthetic Studies on a Nonsteroidal Progesterone Metabolite: Regioselective N-Alkylation of an Activated Pyrazole by Bradley, Paul A., de Koning, Pieter D., Gibson, Karl R., Lecouturier, Yann C., MacKenny, Malcolm C., Morao, Inaki, Poinsard, Cedric, Underwood, Toby J.

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Serendipity in drug-discovery: A new series of 2-(benzyloxy)benzamides as TRPM8 antagonists by Brown, Alan, Ellis, David, Favor, David A., Kirkup, Tony, Klute, Wolfgang, MacKenny, Malcolm, McMurray, Gordon, Stennett, Adam

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Sulfonamides as selective oestrogen receptor β agonists by Roberts, Lee R., Armor, Duncan, Barker, Carolyn, Bent, Andrew, Bess, Kirstin, Brown, Alan, Favor, David A., Ellis, David, Irving, Stephen L., MacKenny, Malcolm, Phillips, Chris, Pullen, Nick, Stennett, Adam, Strand, Linda, Styles, Michelle

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Design and optimization of selective serotonin re-uptake inhibitors with high synthetic accessibility Part 1 by Andrews, Mark, Brown, Alan, Chiva, Jean-Yves, Fradet, David, Gordon, David, Lansdell, Mark, MacKenny, Malcolm

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Design and optimisation of selective serotonin re-uptake inhibitors with high synthetic accessibility: Part 2 by Andrews, Mark, Brown, Alan, Chiva, Jean-Yves, Fradet, David, Gordon, David, Lansdell, Mark, MacKenny, Malcolm

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Sulfonamides as selective oestrogen receptor [beta] agonists by Roberts, Lee R, Armor, Duncan, Barker, Carolyn, Bent, Andrew, Bess, Kirstin, Brown, Alan, Favor, David A, Ellis, David, Irving, Stephen L, MacKenny, Malcolm, Phillips, Chris, Pullen, Nick, Stennett, Adam, Strand, Linda, Styles, Michelle

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Enantioselective synthesis of ( R)- and ( S)- N-Boc-morpholine-2-carboxylic acids by enzyme-catalyzed kinetic resolution: application to the synthesis of reboxetine analogs by Fish, Paul V., Mackenny, Malcolm, Bish, Gerwyn, Buxton, Timothy, Cave, Russell, Drouard, David, Hoople, David, Jessiman, Alan, Miller, Duncan, Pasquinet, Christelle, Patel, Bhairavi, Reeves, Keith, Ryckmans, Thomas, Skerten, Melanie, Wakenhut, Florian

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Designing rapid onset selective serotonin re-uptake inhibitors. Part 3: Site-directed metabolism as a strategy to avoid active circulating metabolites: Structure–activity relations... by Middleton, Donald S., Andrews, Mark, Glossop, Paul, Gymer, Geoffrey, Hepworth, David, Jessiman, Alan, Johnson, Patrick S., MacKenny, Malcolm, Stobie, Alan, Tang, Kim, Morgan, Paul, Jones, Barry

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Designing rapid onset selective serotonin re-uptake inhibitors. 2: Structure–activity relationships of substituted (aryl)benzylamines by Middleton, Donald S., Andrews, Mark, Glossop, Paul, Gymer, Geoffrey, Hepworth, David, Jessiman, Alan, Johnson, Patrick S., MacKenny, Malcolm, Pitcher, Michael J., Rooker, Tony, Stobie, Alan, Tang, Kim, Morgan, Paul

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Designing rapid onset selective serotonin re-uptake inhibitors. Part 1: Structure–activity relationships of substituted (1 S,4 S)-4-(3,4-dichlorophenyl)- N-methyl-1,2,3,4-tetrahydr... by Middleton, Donald S., Andrews, Mark, Glossop, Paul, Gymer, Geoffrey, Jessiman, Alan, Johnson, Patrick S., MacKenny, Malcolm, Pitcher, Michael J., Rooker, Tony, Stobie, Alan, Tang, Kim, Morgan, Paul

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Facile Decarboxylation of Nitrobenzeneacetic Acids as a Convenient Route to Alkylnitrobenzenes by Bull, David J., Fray, M. Jonathan, Mackenny, Malcolm C., Malloy, Kerry A.

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