Aryl Amination Using Soluble Weak Base Enabled by a Water-Assisted Mechanism by Lau, Sii Hong, Yu, Peng, Chen, Liye, Madsen-Duggan, Christina B, Williams, Michael J, Carrow, Brad P

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Discovery of N-[(4R)-6-(4-Chlorophenyl)-7-(2,4-dichlorophenyl)-2,2-dimethyl-3,4-dihydro-2H-pyrano[2,3-b]pyridin-4-yl]-5-methyl-1H-pyrazole-3-carboxamide (MK-5596) as a Novel Cannab... by Yan, Lin, Huo, Pei, Debenham, John S, Madsen-Duggan, Christina B, Lao, Julie, Chen, Richard Z, Xiao, Jing Chen, Shen, Chun-Pyn, Stribling, D. Sloan, Shearman, Lauren P, Strack, Alison M, Tsou, Nancy, Ball, Richard G, Wang, Junying, Tong, Xinchun, Bateman, Thomas J, Reddy, Vijay B. G, Fong, Tung M, Hale, Jeffrey J

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Furo[2,3- b]pyridine-based cannabinoid-1 receptor inverse agonists: Synthesis and biological evaluation. Part 1 by Debenham, John S., Madsen-Duggan, Christina B., Toupence, Richard B., Walsh, Thomas F., Wang, Junying, Tong, Xinchun, Kumar, Sanjeev, Lao, Julie, Fong, Tung M., Xiao, Jing Chen, Huang, Cathy R.-R.C., Shen, Chun-Pyn, Feng, Yue, Marsh, Donald J., Stribling, D. Sloan, Shearman, Lauren P., Strack, Alison M., Goulet, Mark T.

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Dihydro-pyrano[2,3-b]pyridines and tetrahydro-1,8-naphthyridines as CB1 receptor inverse agonists: Synthesis, SAR and biological evaluation by Madsen-Duggan, Christina B., Debenham, John S., Walsh, Thomas F., Yan, Lin, Huo, Pei, Wang, Junying, Tong, Xinchun, Lao, Julie, Fong, Tung M., Xiao, Jing Chen, Huang, Cathy R.-R.C., Shen, Chun-Pyn, Stribling, D.Sloan, Shearman, Lauren P., Strack, Alison M., Goulet, Mark T., Hale, Jeffrey J.

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Pyridopyrimidine based cannabinoid-1 receptor inverse agonists: Synthesis and biological evaluation by Debenham, John S., Madsen-Duggan, Christina B., Wang, Junying, Tong, Xinchun, Lao, Julie, Fong, Tung M., Schaeffer, Marie-Therese, Xiao, Jing Chen, Huang, Cathy C.R.-R., Shen, Chun-Pyn, Sloan Stribling, D., Shearman, Lauren P., Strack, Alison M., Euan MacIntyre, D., Hale, Jeffrey J., Walsh, Thomas F.

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Synthesis of functionalized 1,8-naphthyridinones and their evaluation as novel, orally active CB1 receptor inverse agonists by Debenham, John S., Madsen-Duggan, Christina B., Walsh, Thomas F., Wang, Junying, Tong, Xinchun, Doss, George A., Lao, Julie, Fong, Tung M., Schaeffer, Marie-Therese, Xiao, Jing Chen, Huang, Cathy R.-R.C., Shen, Chun-Pyn, Feng, Yue, Marsh, Donald J., Stribling, D. Sloan, Shearman, Lauren P., Strack, Alison M., MacIntyre, D. Euan, Van der Ploeg, Lex H.T., Goulet, Mark T.

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Lead optimization of 5,6-diarylpyridines as CB1 receptor inverse agonists by Madsen-Duggan, Christina B., Debenham, John S., Walsh, Thomas F., Toupence, Richard B., Huang, Song X., Wang, Junying, Tong, Xinchun, Lao, Julie, Fong, Tung M., Schaeffer, Marie-Therese, Xiao, Jing Chen, Huang, Cathy R.-R.C., Shen, Chun-Pyn, Stribling, D. Sloan, Shearman, Lauren P., Strack, Alison M., MacIntyre, D. Euan, Van der Ploeg, Lex H.T., Goulet, Mark T.

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Diastereoselectivity during 2-pyridone photo-[4+4] cycloaddition. The tribenzylsilyl protecting group by Sieburth, Scott McN, Madsen-Duggan, Christina B, Zhang, Fangning

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Discovery of N -[(4 R )-6-(4-Chlorophenyl)-7-(2,4-dichlorophenyl)-2,2-dimethyl-3,4-dihydro-2 H -pyrano[2,3- b ]pyridin-4-yl]-5-methyl-1 H -pyrazole-3-carboxamide (MK-5596) as a Nov... by Yan, Lin, Huo, Pei, Debenham, John S., Madsen-Duggan, Christina B., Lao, Julie, Chen, Richard Z., Xiao, Jing Chen, Shen, Chun-Pyn, Stribling, D. Sloan, Shearman, Lauren P., Strack, Alison M., Tsou, Nancy, Ball, Richard G., Wang, Junying, Tong, Xinchun, Bateman, Thomas J., Reddy, Vijay B. G., Fong, Tung M., Hale, Jeffrey J.

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Discovery of N‑[Bis(4-methoxyphenyl)methyl]-4-hydroxy-2-(pyridazin-3-yl)pyrimidine-5-carboxamide (MK-8617), an Orally Active Pan-Inhibitor of Hypoxia-Inducible Factor Prolyl Hydrox... by Debenham, John S, Madsen-Duggan, Christina, Clements, Matthew J, Walsh, Thomas F, Kuethe, Jeffrey T, Reibarkh, Mikhail, Salowe, Scott P, Sonatore, Lisa M, Hajdu, Richard, Milligan, James A, Visco, Denise M, Zhou, Dan, Lingham, Russell B, Stickens, Dominique, DeMartino, Julie A, Tong, Xinchun, Wolff, Michael, Pang, Jianmei, Miller, Randy R, Sherer, Edward C, Hale, Jeffrey J

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