The discovery of 2-substituted phenol quinazolines as potent RET kinase inhibitors with improved KDR selectivity by Newton, Rebecca, Bowler, Katherine A., Burns, Emily M., Chapman, Philip J., Fairweather, Emma E., Fritzl, Samantha J.R., Goldberg, Kristin M., Hamilton, Niall M., Holt, Sarah V., Hopkins, Gemma V., Jones, Stuart D., Jordan, Allan M., Lyons, Amanda J., Nikki March, H., McDonald, Neil Q., Maguire, Laura A., Mould, Daniel P., Purkiss, Andrew G., Small, Helen F., Stowell, Alexandra I.J., Thomson, Graeme J., Waddell, Ian D., Waszkowycz, Bohdan, Watson, Amanda J., Ogilvie, Donald J.

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Identification of selective inhibitors of RET and comparison with current clinical candidates through development and validation of a robust screening cascade by Watson, Amanda J, Hopkins, Gemma V, Hitchin, Samantha, Begum, Habiba, Jones, Stuart, Jordan, Allan, Holt, Sarah, March, H Nikki, Newton, Rebecca, Small, Helen, Stowell, Alex, Waddell, Ian D, Waszkowycz, Bohdan, Ogilvie, Donald J

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Identification of selective inhibitors of RET and comparison with current clinical candidates through development and validation of a robust screening cascade [version 1; peer revi... by Watson, Amanda J, Hopkins, Gemma V, Hitchin, Samantha, Begum, Habiba, Jones, Stuart, Jordan, Allan, Holt, Sarah, March, H. Nikki, Newton, Rebecca, Small, Helen, Stowell, Alex, Waddell, Ian D, Waszkowycz, Bohdan, Ogilvie, Donald J

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ERK1/2, but not ERK5, is necessary and sufficient for phosphorylation and activation of c-Fos by Gilley, Rebecca, March, H. Nikki, Cook, Simon J.

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Nuclear receptor binding protein 1 regulates intestinal progenitor cell homeostasis and tumour formation by Wilson, Catherine H, Crombie, Catriona, van der Weyden, Louise, Poulogiannis, George, Rust, Alistair G, Pardo, Mercedes, Gracia, Tannia, Yu, Lu, Choudhary, Jyoti, Poulin, Gino B, McIntyre, Rebecca E, Winton, Douglas J, March, H Nikki, Arends, Mark J, Fraser, Andrew G, Adams, David J

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Anilinoquinazoline inhibitors of the RET kinase domain—Elaboration of the 7-position by Jordan, Allan M., Begum, Habiba, Fairweather, Emma, Fritzl, Samantha, Goldberg, Kristin, Hopkins, Gemma V., Hamilton, Niall M., Lyons, Amanda J., March, H. Nikki, Newton, Rebecca, Small, Helen F., Vishwanath, Swamy, Waddell, Ian D., Waszkowycz, Bohdan, Watson, Amanda J., Ogilvie, Donald J.

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Abstract B05: Discovery, validation and targeting of novel synthetic lethal interactions in academic drug discovery by March, H. Nikki, Chapman, Phil, Blaikley, Elizabeth, Eberlein, Catherine A., Cockerill, Mark, Hitchin, Samantha, Waddell, Ian D., Ogilvie, Donald

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Abstract 1139: Novel, cellular active inhibitors of G6PD, a key mediator of ROS-induced cellular stress by Jordan, Allan M., Hamilton, Niall M., Hamilton, Nicola S., Hitchin, James R., James, Dominic I., Jones, Stuart D., Lyons, Amanda J., March, H. Nikki, Thomson, Graeme J., Waddell, Ian D., Ogilvie, Donald J.

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Nuclear receptor binding protein 1 regulates intestinal progenitor cell homeostasis and tumour formation: Nrbp1 regulates cell fate and tumourigenesis by Wilson, Catherine H, Crombie, Catriona, van der Weyden, Louise, Poulogiannis, George, Rust, Alistair G, Pardo, Mercedes, Gracia, Tannia, Yu, Lu, Choudhary, Jyoti, Poulin, Gino B, McIntyre, Rebecca E, Winton, Douglas J, March, H Nikki, Arends, Mark J, Fraser, Andrew G, Adams, David J

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