Characterization of the cellular and antitumor effects of MPI-0479605, a small-molecule inhibitor of the mitotic kinase Mps1 by Tardif, Keith D, Rogers, Aaron, Cassiano, Jared, Roth, Bruce L, Cimbora, Daniel M, McKinnon, Rena, Peterson, Ashley, Douce, Thomas B, Robinson, Rosann, Dorweiler, Irene, Davis, Thaylon, Hess, Mark A, Ostanin, Kirill, Papac, Damon I, Baichwal, Vijay, McAlexander, Ian, Willardsen, J Adam, Saunders, Michael, Christophe, Hoarau, Kumar, D Vijay, Wettstein, Daniel A, Carlson, Robert O, Williams, Brandi L

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Discovery of (2S)‑1-[4-(2-{6-Amino-8-[(6-bromo-1,3-benzodioxol-5-yl)sulfanyl]‑9H‑purin-9-yl}ethyl)piperidin-1-yl]-2-hydroxypropan-1-one (MPC-3100), a Purine-Based Hsp90 Inhibitor... by Kim, Se-Ho, Bajji, Ashok, Tangallapally, Rajendra, Markovitz, Benjamin, Trovato, Richard, Shenderovich, Mark, Baichwal, Vijay, Bartel, Paul, Cimbora, Daniel, McKinnon, Rena, Robinson, Rosann, Papac, Damon, Wettstein, Daniel, Carlson, Robert, Yager, Kraig M

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The Human Endosomal Sorting Complex Required for Transport (ESCRT-I) and Its Role in HIV-1 Budding by Stuchell, Melissa D, Garrus, Jennifer E, Mueller, Barbara, Stray, Kirsten M, Ghaffarian, Sanaz, Mckinnon, Rena, Kraeusslich, Hans-Georg, Morham, Scott G, Sundquist, Wesley I

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Lead optimization of purine based orally bioavailable Mps1 (TTK) inhibitors by Vijay Kumar, D., Hoarau, Christophe, Bursavich, Matthew, Slattum, Paul, Gerrish, David, Yager, Kraig, Saunders, Michael, Shenderovich, Mark, Roth, Bruce L., McKinnon, Rena, Chan, Ashley, Cimbora, Daniel M., Bradford, Chad, Reeves, Leslie, Patton, Scott, Papac, Damon I., Williams, Brandi L., Carlson, Robert O.

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Triterpene based compounds with potent anti-maturation activity against HIV-1 by Gerrish, David, Kim, In Chul, Kumar, Dange V., Austin, Harry, Garrus, Jennifer E., Baichwal, Vijay, Saunders, Michael, McKinnon, Rena S., Anderson, Mark B., Carlson, Robert, Arranz-Plaza, Esther, Yager, Kraig M.

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Discovery of (2 S )-1-[4-(2-{6-Amino-8-[(6-bromo-1,3-benzodioxol-5-yl)sulfanyl]-9 H -purin-9-yl}ethyl)piperidin-1-yl]-2-hydroxypropan-1-one (MPC-3100), a Purine-Based Hsp90 Inhibit... by Kim, Se-Ho, Bajji, Ashok, Tangallapally, Rajendra, Markovitz, Benjamin, Trovato, Richard, Shenderovich, Mark, Baichwal, Vijay, Bartel, Paul, Cimbora, Daniel, McKinnon, Rena, Robinson, Rosann, Papac, Damon, Wettstein, Daniel, Carlson, Robert, Yager, Kraig M.

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Design and characterization of ebolavirus GP prehairpin intermediate mimics as drug targets by Clinton, Tracy R., Weinstock, Matthew T., Jacobsen, Michael T., Szabo‐Fresnais, Nicolas, Pandya, Maya J., Whitby, Frank G., Herbert, Andrew S., Prugar, Laura I., McKinnon, Rena, Hill, Christopher P., Welch, Brett D., Dye, John M., Eckert, Debra M., Kay, Michael S.

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Analogues of 4-[(7-Bromo-2-methyl-4-oxo-3H-quinazolin-6-yl)methylprop-2-ynylamino]-N-(3-pyridylmethyl)benzamide (CB-30865) as Potent Inhibitors of Nicotinamide Phosphoribosyltransf... by Lockman, Jeffrey W, Murphy, Brett R, Zigar, Daniel F, Judd, Weston R, Slattum, Paul M, Gao, Zhong-Hua, Ostanin, Kirill, Green, Jeremy, McKinnon, Rena, Terry-Lorenzo, Ryan T, Fleischer, Tracey C, Boniface, J. Jay, Shenderovich, Mark, Willardsen, J. Adam

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Abstract A77: Inhibition of TTK promotes chromosome segregation defects in a manner distinct from inhibitors of Aurora or PLK mitotic kinases by Williams, Brandi L., Roth, Bruce L., Cassiano, Jared, McKinnon, Rena S., Brown, Brita, Hoarau, Christophe, Saunders, Michael, Kumar, D. Vijay

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Abstract LB-288: MPI-0486348: A novel inhibitor of nicotinamide phosphoribosyltransferase (Nampt) induces tumor regression in a preclinical model by Fleischer, Tracey C., Baichwal, Vijay R., Bradford, Chad L., Demie, Lynn, Green, Jeremy P., Hess, Mark A., Lockman, Jeffrey W., McKinnon, Rena, Ostanin, Kirill, Papac, Damon I., Reeves, Leslie F., Terry-Lorenzo, Ryan T., Willardsen, J Adam

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