Design and in vitro characterization of PAC1/VPAC1-selective agonists with potent neuroprotective effects by Doan, Ngoc-Duc, Bourgault, Steve, Dejda, Agnieszka, Létourneau, Myriam, Detheux, Michel, Vaudry, David, Vaudry, Hubert, Chatenet, David, Fournier, Alain

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Abstract LB-291: EOS100850, an insurmountable and non-brain penetrant A2A receptor antagonist, inhibits adenosine-mediated T cell suppression, demonstrates anti-tumor activity and... by Houthuys, Erica, Marillier, Reece, Deregnaucourt, Théo, Brouwer, margreet, Basilico, Paola, Pirson, Romain, Marchante, Joao, Prasad, Shruthi, Hermant, Annelise, Nyawouame, Florence, Preillon, Julie, Frederix, Kim, Michaux, Anne Catherine, Lambolez, Florence, Swiercz, Jakub, Driessens, Gregory, Wald, Noemie, Martinoli, Chiara, Bodo, Veronique, Detheux, Michel, Leroy, Xavier, Crosignani, Stefano

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Distinct recognition of OX1 and OX2 receptors by orexin peptides by Ammoun, Sylwia, Holmqvist, Tomas, Shariatmadari, Ramin, Oonk, Hendrica B, Detheux, Michel, Parmentier, Marc, Akerman, Karl E O, Kukkonen, Jyrki P

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Abstract B030: Development and validation of a phenotypic screening platform for the identification of novel immuno-oncology targets by Rabolli, Virginie, Martini, Murielle, Scoumanne, Ariane, Letellier, Marie-Claire, Crosignani, Stefano, Quéva, Christophe, Detheux, Michel, Swiercz, Jakub M., Cauwenberghs, Sandra

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Design, Synthesis, and Structure−Activity Relationships of Novel Bicyclic Azole-amines as Negative Allosteric Modulators of Metabotropic Glutamate Receptor 5 by Burdi, Douglas F, Hunt, Rachel, Fan, Lei, Hu, Tao, Wang, Jun, Guo, Zihong, Huang, Zhiqiang, Wu, Chengde, Hardy, Larry, Detheux, Michel, Orsini, Michael A, Quinton, Maria S, Lew, Robert, Spear, Kerry

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Preclinical assessment of a novel small molecule inhibitor of indoleamine 2,3-dioxygenase 1 (IDO1) by Driessens, Gregory, Crosignani, Stefano, Detheux, Michel, Van den Eynde, Benoît, Cauwenberghs, Sandra

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Preclinical assessment of a novel small molecule inhibitor of tryptophan 2,3-dioxygenase 2 (TDO2) by Crosignani, Stefano, Driessens, Gregory, Detheux, Michel, Van den Eynde, Benoît, Cauwenberghs, Sandra

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Serotonin 5-HT2B receptor loss of function mutation in a patient with fenfluramine-associated primary pulmonary hypertension by BLANPAIN, Cédric, LE POUL, Emmanuel, PARMA, Jasmine, KNOOP, Christiane, DETHEUX, Michel, PARMENTIER, Marc, VASSART, Gilbert, ABRAMOWICZ, Marc J

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CD26/Dipeptidyl-Peptidase IV Down-Regulates the Eosinophil Chemotactic Potency, But Not the Anti-HIV Activity of Human Eotaxin by Affecting Its Interaction with CC Chemokine Recept... by Struyf, Sofie, Proost, Paul, Schols, Dominique, De Clercq, Erik, Opdenakker, Ghislain, Lenaerts, Jean-Pierre, Detheux, Michel, Parmentier, Marc, De Meester, Ingrid, Scharpe, Simon, Van Damme, Jo

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Significance of N-Terminal Proteolysis of CCL14a to Activity on the Chemokine Receptors CCR1 and CCR5 and the Human Cytomegalovirus-Encoded Chemokine Receptor US28 by Richter, Rudolf, Casarosa, Paola, Standker, Ludger, Munch, Jan, Springael, Jean-Yves, Nijmeijer, Saskia, Forssmann, Wolf-Georg, Vischer, Henry F, Vakili, Jalal, Detheux, Michel, Parmentier, Marc, Leurs, Rob, Smit, Martine J

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Agonist and antagonist activities on human NPFF 2 receptors of the NPY ligands GR231118 and BIBP3226 by Mollereau, Catherine, Gouardères, Christine, Dumont, Yvan, Kotani, Masato, Detheux, Michel, Doods, Henri, Parmentier, Marc, Quirion, Rémi, Zajac, Jean‐Marie

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Urokinase Plasminogen Activator and Plasmin Efficiently Convert Hemofiltrate CC Chemokine 1 into Its Active [9-74] Processed Variant by Vakili, Jalal, Standker, Ludger, Detheux, Michel, Vassart, Gilbert, Forssmann, Wolf-Georg, Parmentier, Marc

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Recombinant aequorin as a reporter for receptor-mediated changes of intracellular Ca 2+ -levels in Drosophila S2 cells by Torfs, Herbert, Poels, Jeroen, Detheux, Michel, Dupriez, Vincent, Van Loy, Tom, Vercammen, Linda, Vassart, Gilbert, Parmentier, Marc, Vanden Broeck, Jozef

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Oxysterols direct immune cell migration through EBI2 by Hannedouche, Sébastien, Zhang, Juan, Yi, Tangsheng, Shen, Weijun, Nguyen, Deborah, Pereira, João P., Guerini, Danilo, Baumgarten, Birgit U., Roggo, Silvio, Wen, Ben, Knochenmuss, Richard, Noël, Sophie, Gessier, Francois, Kelly, Lisa M., Vanek, Mirka, Laurent, Stephane, Preuss, Inga, Miault, Charlotte, Christen, Isabelle, Karuna, Ratna, Li, Wei, Koo, Dong-In, Suply, Thomas, Schmedt, Christian, Peters, Eric C., Falchetto, Rocco, Katopodis, Andreas, Spanka, Carsten, Roy, Marie-Odile, Detheux, Michel, Chen, Yu Alice, Schultz, Peter G., Cho, Charles Y., Seuwen, Klaus, Cyster, Jason G., Sailer, Andreas W.

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Transmembrane Domain V of the Endothelin-A Receptor Is a Binding Domain of ETA-Selective TTA-386-Derived Photoprobes by Tessier, Sophie, Boivin, Stéphane, Aubin, Jacinthe, Lampron, Philipe, Detheux, Michel, Fournier, Alain

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Identification of a Binding Domain of the Endothelin-B Receptor Using a Selective IRL-1620-Derived Photoprobe by Boivin, Stéphane, Tessier, Sophie, Aubin, Jacinthe, Lampron, Philipe, Detheux, Michel, Fournier, Alain

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PTHrP fragments 1-16 and 1-23 do not bind to either the ET sub(A) or the ET sub(B) endothelin receptors by Langlois, Chantal, Letourneau, Myriam, Turcotte, Kathy, Detheux, Michel, Fournier, Alain

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PTHrP fragments 1-16 and 1-23 do not bind to either the ET A or the ET B endothelin receptors by Langlois, Chantal, Létourneau, Myriam, Turcotte, Kathy, Detheux, Michel, Fournier, Alain

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Transmembrane Domain V of the Endothelin-A Receptor Is a Binding Domain of ET A -Selective TTA-386-Derived Photoprobes by Tessier, Sophie, Boivin, Stéphane, Aubin, Jacinthe, Lampron, Philipe, Detheux, Michel, Fournier, Alain

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PTHrP fragments 1-16 and 1-23 do not bind to either the ETA or the ETB endothelin receptors by LANGLOIS, Chantal, LETOURNEAU, Myriam, TURCOTTE, Kathy, DETHEUX, Michel, FOURNIER, Alain

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