In vitro and in vivo activities of the diazabicyclooctane OP0595 against AmpC-derepressed Pseudomonas aeruginosa by Morinaka, Akihiro, Tsutsumi, Yuko, Yamada, Keiko, Takayama, Yoshihiro, Sakakibara, Shiro, Takata, Toshihiko, Abe, Takao, Furuuchi, Takeshi, Inamura, Seiichi, Sakamaki, Yoshiaki, Tsujii, Nakako, Ida, Takashi

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OP0595, a new diazabicyclooctane: mode of action as a serine β-lactamase inhibitor, antibiotic and β-lactam 'enhancer' by Morinaka, Akihiro, Tsutsumi, Yuko, Yamada, Mototsugu, Suzuki, Kenji, Watanabe, Takashi, Abe, Takao, Furuuchi, Takeshi, Inamura, Seiichi, Sakamaki, Yoshiaki, Mitsuhashi, Nakako, Ida, Takashi, Livermore, David M

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X-ray crystallographic analysis of IMP-1 metallo-β-lactamase complexed with a 3-aminophthalic acid derivative, structure-based drug design, and synthesis of 3,6-disubstituted phtha... by Hiraiwa, Yukiko, Saito, Jun, Watanabe, Takashi, Yamada, Mototsugu, Morinaka, Akihiro, Fukushima, Takayoshi, Kudo, Toshiaki

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Metallo-β-lactamase inhibitory activity of 3-alkyloxy and 3-amino phthalic acid derivatives and their combination effect with carbapenem by Hiraiwa, Yukiko, Morinaka, Akihiro, Fukushima, Takayoshi, Kudo, Toshiaki

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Discovery of 2-hydroxyarbekacin, a new aminoglycoside antibiotic with reduced nephrotoxicity by Takahashi, Yoshiaki, Umemura, Eijiro, Kobayashi, Yoshihiko, Murakami, Shoichi, Nawa, Toru, Morinaka, Akihiro, Miyake, Toshiaki, Shibasaki, Masakatsu

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Structural Insights into the TLA-3 Extended-Spectrum β-Lactamase and Its Inhibition by Avibactam and OP0595 by Jin, Wanchun, Wachino, Jun-Ichi, Yamaguchi, Yoshihiro, Kimura, Kouji, Kumar, Anupriya, Yamada, Mototsugu, Morinaka, Akihiro, Sakamaki, Yoshiaki, Yonezawa, Minoru, Kurosaki, Hiromasa, Arakawa, Yoshichika

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In Vitro and In Vivo Activities of OP0595, a New Diazabicyclooctane, against CTX-M-15-Positive Escherichia coli and KPC-Positive Klebsiella pneumoniae by Morinaka, Akihiro, Tsutsumi, Yuko, Yamada, Keiko, Takayama, Yoshihiro, Sakakibara, Shiro, Takata, Toshihiko, Abe, Takao, Furuuchi, Takeshi, Inamura, Seiichi, Sakamaki, Yoshiaki, Tsujii, Nakako, Ida, Takashi

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Metallo-β-lactamase inhibitory activity of phthalic acid derivatives by Hiraiwa, Yukiko, Morinaka, Akihiro, Fukushima, Takayoshi, Kudo, Toshiaki

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Activity of carbapenems with ME1071 (disodium 2,3-diethylmaleate) against Enterobacteriaceae and Acinetobacter spp. with carbapenemases, including NDM enzymes by Livermore, David M, Mushtaq, Shazad, Morinaka, Akihiro, Ida, Takashi, Maebashi, Kazunori, Hope, Russell

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OP0595, a new diazabicyclooctane: mode of action as a serine [Beta]-lactamase inhibitor, antibiotic and [Beta]-lactam 'enhancer' by Morinaka, Akihiro, Tsutsumi, Yuko, Yamada, Mototsugu, Suzuki, Kenji, Watanabe, Takashi, Abe, Takao, Furuuchi, Takeshi, Inamura, Seiichi, Sakamaki, Yoshiaki, Mitsuhashi, Nakako, Ida, Takashi, Livermore, David M

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Metallo-b-lactamase inhibitory activity of phthalic acid derivatives by Hiraiwa, Yukiko, Morinaka, Akihiro, Fukushima, Takayoshi, Kudo, Toshiaki

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Small G protein Ral and its downstream molecules regulate endocytosis of EGF and insulin receptors by Nakashima, Shintaro, Morinaka, Kenji, Koyama, Shinya, Ikeda, Masahiro, Kishida, Michiko, Okawa, Katsuya, Iwamatsu, Akihiro, Kishida, Shosei, Kikuchi, Akira

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Design and syntheses of 4-acylaminopyridine derivatives: Novel high affinity choline uptake enhancers II by Chaki, Haruyuki, Yamabe, Haruko, Sugano, Mamoru, Morita, Shuji, Bessho, Tomoko, Tabata, Reiko, Saito, Ken-Ichi, Egawa, Mitsuo, Tobe, Akihiro, Morinaka, Yasuhiro

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Design and syntheses of 4-acylaminopyridine derivatives: Novel high affinity choline uptake enhancers I by Chaki, Haruyuki, Yamabe, Haruko, Sugano, Mamoru, Morita, Shuji, Bessho, Tomoko, Tabata, Reiko, Saito, Ken-Ichi, Egawa, Mitsuo, Tobe, Akihiro, Morinaka, Yasuhiro

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