PD-1 derived CA-170 is an oral immune checkpoint inhibitor that exhibits preclinical anti-tumor efficacy by Sasikumar, Pottayil G., Sudarshan, Naremaddepalli S., Adurthi, Srinivas, Ramachandra, Raghuveer K., Samiulla, Dodderi S., Lakshminarasimhan, Anirudha, Ramanathan, Anuradha, Chandrasekhar, Talapaneni, Dhudashiya, Amit A., Talapati, Sumalatha R., Gowda, Nagesh, Palakolanu, Sreenivasulareddy, Mani, Jiju, Srinivasrao, Bandi, Joseph, David, Kumar, Nigam, Nair, Rashmi, Atreya, Hanudatta S., Gowda, Nagaraj, Ramachandra, Murali

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Abstract 4148: An orally bioavailable small molecule antagonist of TIM-3 signaling pathway shows potent anti-tumor activity by Sasikumar, Pottayil G., Naremaddepalli, Sudarshan S., Ramachandra, Raghuveer K., Gowda, Nagesh, Devarapalli, Srinivaskumar, Adurthi, Sreenivas, Mani, Jiju, Nair, Rashmi, Dhudashiya, Amit A., Samiulla, Dodheri S., Gowda, Nagaraj M., Ramachandra, Murali

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Abstract A96: First-in-class orally available immune checkpoint antagonists for cancer therapy by Sasikumar, Pottayil G., Naremaddepalli, Sudarshan S., Gowda, Nagaraj, Adurthi, Sreenivas, Dhodheri, Samiulla, Dhudashia, Amit, Ramachandra, Raghuveer, Ramachandra, Murali

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Abstract B006: Functional antagonism of VSIG8-mediated immune suppression by oral VISTA agents by Sasikumar, Pottayil G., Naremaddepalli, Sudarshan S., Ramachandra, Raghuveer K., Gowda, Nagesh, Yerramsetti, Manikyala Rao, Bandireddy, Srinivasa Rao, Adurthi, Sreenivas, Mani, Jiju, Nair, Rashmi, Dhudashia, Amit A., Dodheri, Samiulla S., Gowda, Nagaraj M., Ramachandra, Murali

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Abstract B007: Potent antitumor activity of a novel and orally available small-molecule antagonist targeting the CD47/SIRPα pathway by Sasikumar, Pottayil G., Gundala, Chennakrishnareddy, Balasubramanian, Wesley R., Naremaddepalli, Sudarshan S., Bhumireddy, Archana, Patil, Sandeep S., Dhudashiya, Amit A., Rayavarapu, Vijaysai, Lakshminarasimhan, Anirudha, Samiulla, Dodheri S., Aithal, Kiran, Daginakatte, Girish, Ramachandra, Murali

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Abstract 1650: Targeting CD47- SIRPα interaction by novel peptide-based antagonists by Sasikumar, Pottayil G., Gundala, Chennakrishnareddy, Gowda, Nagaraj M., Naremaddepalli, Sudarshan S., Bhumireddy, Archana, Nair, Rashmi, Balasubramanian, Wesley Roy, Lakshminarasimhan, Anirudha, Dodheri, Samiulla S., Aithal, Kiran, Ramachandra, Raghuveer K., Daginakatte, Girish, Ramachandra, Murali

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Efficient Synthesis of O-Succinimidyl-(tert-Butoxycarbonylamino)methyl Carbamates Derived from α-Amino Acids Accelerated by Ultrasound: Application to the Synthesis of Ureidodipept... by Sureshbabu, Vommina V., Sudarshan, Naremaddepalli S., Kantharaju

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Abstract A36: CA-170, an oral small molecule PD-L1 and VISTA immune checkpoint antagonist, promotes T cell immune activation and inhibits tumor growth in pre-clinical models of can... by Lazorchak, Adam S., Patterson, Troy, Ding, Yueyun, Sasikumar, Pottayil G., Sudarshan, Naremaddepalli S., Gowda, Nagaraj M., Ramachandra, Raghuveer K., Samiulla, Dodheri S., Giri, Sanjeev, Eswarappa, Rajesh, Ramachandra, Murali, Tuck, David, Wyant, Timothy

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HOBt·DCHA-Mediated Synthesis of Sterically Hindered Peptides employing Fmoc-Amino Acid Chlorides in Both Solution-Phase and Solid Phase Methods by Sureshbabu, Vommina V., Sudarshan, Naremaddepalli S., Chenna Krishna, G.

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Microwave Assisted Alcoholysis of Isocyanates Derived from Nα-[(9-fluorenylmethyl)oxy]carbonyl Amino Acids: Synthesis of N-Fmoc-N1-Z-/Boc-/Alloc-/Bsmoc-gem-diamines by Venkataramanarao, Rao, Sudarshan, Naremaddepalli S, Sureshbabu, Vommina V

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Microwave Assisted Alcoholysis of Isocyanates Derived from N[alpha]-[(9-fluorenylmethyl)oxy]carbonyl Amino Acids: Synthesis of N-Fmoc-N1-Z-/Boc-/Alloc-/Bsmoc-gem-diamines by Venkataramanarao, Rao, Sudarshan, Naremaddepalli S, Sureshbabu, Vommina V

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Abstract 3852: Combination efficacy and safety profile of an orally bioavailable small molecule agent targeting CD47/SIRPα axis by Daginakatte, Girish, Pottayil, Sasikumar, Chennakrishna, Gundala, Balasubramanian, Wesley Roy, Naremaddepalli, Sudarshan, Bhumireddy, Archana, Patil, Sandeep, Nellore, Kavitha, Chand, Priyabrata, Aithal, Kiran, Dhudashiya, Amit, DS, Samiulla, Eswarappa, Rajesh, Ramachandra, Murali

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Abstract 3500: AUR103 an oral small molecule CD47 antagonist in combination with azacytidine and bortezomib exhibits potent anti-tumor activity in myeloma and leukemia models in vi... by Daginakatte, Girish C., Pottayil, Sasikumar, Naremaddepalli, Sudarshan, Chennakrishnareddy, Gundala, Bilugudi, Prasad, Tangella, Sai Krishna, Patil, Sandeep, Gowda, Nagesh, Aithal, Kiran, Balasubramanian, Wesley Roy, Dhudashiya, Amit, Dodheri, Samiulla, Nellore, Kavitha, Samajdar, Susanta, Ramachandra, Murali

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